Carbamate linkers as latent N-methylamines in solid phase synthesis

Tetrahedron Letters

Volumn 38, Issue 16, 1997, Pages 2799-2802

  Ho, Chih Y ^a   Kukla, Michael J ^a  

^a JANSSEN RESEARCH AND DEVELOPMENT   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMINE;

ARTICLE; DRUG SYNTHESIS; IN VITRO STUDY; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; REACTION ANALYSIS; TECHNIQUE;

EID: 0030914639     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(97)00510-8     Document Type: Article

References (12)

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2. (b) Fruchtel, J.S.; Jung, G., Angew. Chem. Int. Ed. Engl. 1996, 35, 17-42.
3. (c) Hemkens, P.H.H.; Ottenheijm, H.C.J.; Rees, D., Tetrahedron 1996, 52, 4527-4554.
4. (a) Plunkett, M.J.; Ellman, J.A., J. Org. Chem. 1995, 60, 6006-6007.
5. (b) Chenera, B.; Finkelstein, J.A.; Veber, D.F., J. Amer. Chem. Soc. 1995, 117, 11999-12000.
6. Morphy, J.R.; Rankovic, Z.; Rees, D.C., Tetrahedron Lett. 1996, 37, 3209-3212.
7. (a)Letsinger, R.L.; Kornet, M.J.; Mahadevan, V.; Jerina, D.M., J. Amer. Chem. Soc. 1964, 86, 5163-5165.
8. (b) Dixit, D.M.; Lenzoff, C.C., J. Chem. Soc. Chem. Commun. 1977, 798-799.
9. (c) Letsinger, R.L.; Kornet, M.J., J. Amer. Chem. Soc. 1963, 85, 3045-3046.
10. (d) Felix, A.M.; Merrifield, R.B., J. Amer. Chem. Soc. 1970, 92, 1385-1391.
11. (e) Hauske, J. R.; Dorff, P. Tetrahedron Lett. 1995, 36, 1589-1592.
12. Dressman, B.A.; Spangle, L.A.; Kaldor, S.W., Tetrahedron Lett. 1996, 37, 937-940.