Evaluation of cross-linked amylose press-coated tablets for sustained drug delivery

International Journal of Pharmaceutics

Volumn 149, Issue 2, 1997, Pages 139-149

  Moussa, Iskandar S ^a   Cartilier, Louis H ^a  

^a UNIVERSITÉ DE MONTRÉAL   (Canada)

Author keywords

Acetaminophen; Compression coating; Controlled release; Cross linked amylose; Diltiazem HCl; Hydrophilic matrix

Indexed keywords

AMYLOSE; DILTIAZEM; PARACETAMOL;

ARTICLE; COMPRESSION; CROSS LINKING; DISSOLUTION; DRUG COATING; DRUG RELEASE; PRIORITY JOURNAL; SUSTAINED RELEASE PREPARATION; TABLET COMPRESSION; THERMODYNAMICS;

EID: 0030901087     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-5173(97)04864-3     Document Type: Article

References (17)

1. Baker, R.W. and Lonsdale, H.K., Controlled release: mechanisms and rates. In Tanquary, A.C. and Lacey, R.E. (Eds.), Controlled Release of Biologically Active Agents: Advances in Experimental Medicine and Biology, Plenum Press, New York, 1974, pp. 15-71.
2. Banks, W. and Greenwood, C.T., Starch and its Components, Edinburgh University Press, Edinburgh, 1975.
3. Bogin, R.M. and Ballard, R.D., Treatment of nocturnal asthma with pulsed-release albuterol. Chest, 102 (1992) 362-366.
4. Crank, J., The Mathematics of Diffusion, Oxford University Press, New York, 1970.
5. Dumoulin, Y., Cartilier, L., Preda, M., Alex, S., Lenaerts, V. and Mateescu, M., Cross-linked amylose as matrix for drug controlled release. X-Ray and FT-IR analysis. Proc. Int. Symp. Control. Release Bioact. Mater., 21 (1994a) 660-661.
6. Dumoulin, Y., Clement, P., Mateescu, M.A. and Cartilier, L., Cross-linked amylose as a binder/disintegrant in compressed tablets. S.T.P. Pharma, 5 (1994b) 329-335.
7. Lenaerts, V., Dumoulin, Y. and Mateescu, M.A., Controlled release of theophylline from cross-linked amylose tablets. J. Control. Release, 15 (1991) 39-46.
8. Lenaerts, V., Dumoulin, Y., Cartilier, L. and Mateescu, M., Cross-linked amylose tablets for controlled-release of drugs. Proc. Int. Symp. Control. Release Bioact. Mater., 19 (1992) 30-31.
9. Mateescu, M., Dumoulin, Y., Delmas G., Lenaerts, V. and Cartilier, L., Cross-linked amylose: a new matrix for drug controlled release. Molecular insights. Proc. Int. Symp. Control. Release Bioact. Mater., 20 (1993) 290-291.
10. Mateescu, M., Lenaerts, V. and Dumoulin, Y., Cross-linked material for controlled-release of biologically active compounds, U.S. Patent 618,650, 1991.
11. Moussa, I.S. and Cartilier, L.H., Characterization of moving fronts in cross-linked amylose matrices by image analysis. J. Control. Release, 42 (1996) 47-56.
12. Moussa, I.S. and Cartilier, L.H., The influence of the cross-linking degree on drug dissolution, water uptake and swelling profiles of cross-linked amylose matrices. Proc. 1st World Meeting APGI/APV, 1995, pp. 241-242.
13. Ofner III, C.M. and Schott, H., Swelling studies of gelatin. I. Gelatin without additives. J. Pharm. Sci., 75 (1986) 790-796.
14. Ségot-Chicq, S., Teillaud, E. and Peppas, N.A., Les dispositifs à libération contrôlée pour la délivrance des principes actifs médicamenteux. I. Intérêt et applications. S.T.P. Pharma, 1 (1985) 25-36.
15. Sirkiä, T., Mäkimartti, M., Liukko-Sipi, S. and Marvolla, M., Development and biopharmaceutical evaluations of a new press-coated prolonged-release salbutamol sulphate tablet in man. Eur. J. Pharm. Sci., 1 (1994) 195-201.
16. Thiffault, J., Landriault, H., Gossard, D., Raymond, M., Caillé, G. and Spénard, J., Influence of time of administration of a once-a-day diltiazem formulation on its pharmacokinetics. Pharm. Res., 10 (1993) S-313.
17. Zolia, I., L'amylose réticulé, nouveau polymère pour la libération contrôlée de médicament. Etude du mécanisme de contrôle. Master's Thesis, Faculty of Pharmacy, University of Montreal, 1994.