Inhibition by protein kinase C of the 86Rb+ efflux and vasorelaxation induced by P1075, a K(ATP) channel opener, in rat isolated aorta

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 356, Issue 3, 1997, Pages 425-432

  Linde, Claudia ^a   Löffler, Cornelia ^a   Quast, Ulrich ^a  

^a UNIVERSITY OF TÜBINGEN   (Germany)

Author keywords

86Rb+ efflux; Glibenclamide; P1075; P1075 binding; Phorbol ester; Potassium channel openers; Protein kinase C; Staurosporine; Vasorelaxation

Indexed keywords

1 (5 ISOQUINOLINESULFONYL) 2 METHYLPIPERAZINE; 2 [1 (3 DIMETHYLAMINOPROPYL) 3 INDOLYL] 3 (3 INDOLYL)MALEIMIDE; 2 CYANO 1 (1,1 DIMETHYLPROPYL) 3 (3 PYRIDYL)GUANIDINE; 4ALPHA PHORBOL DIBUTYRATE; CHELERYTHRINE; GLIBENCLAMIDE; PHORBOL 13 ACETATE 12 MYRISTATE; PHORBOL DIBUTYRATE; POTASSIUM CHANNEL; POTASSIUM CHANNEL STIMULATING AGENT; PROTEIN KINASE C; PROTEIN KINASE C ACTIVATOR; PROTEIN KINASE C INHIBITOR; RUBIDIUM 86; STAUROSPORINE;

ANIMAL TISSUE; AORTA; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG INHIBITION; DRUG POTENTIATION; ION TRANSPORT; MALE; MEMBRANE BINDING; NONHUMAN; RAT; SMOOTH MUSCLE RELAXATION; STEREOISOMERISM; VASCULAR RING; VASODILATATION;

ADENOSINE TRIPHOSPHATE; ANIMALS; AORTA; ENZYME ACTIVATION; ENZYME INHIBITORS; GUANIDINES; MALE; MUSCLE CONTRACTION; MUSCLE RELAXATION; MUSCLE, SMOOTH, VASCULAR; PHORBOL 12,13-DIBUTYRATE; POTASSIUM CHANNELS; PROTEIN BINDING; PROTEIN KINASE C; PYRIDINES; RATS; RATS, SPRAGUE-DAWLEY; RUBIDIUM RADIOISOTOPES; TETRADECANOYLPHORBOL ACETATE;

EID: 0030883208     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/PL00005072     Document Type: Article

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