One-pot preparation of 1-substituted imidazole-2-thione from isothiocyanate and amino acetal

Synthetic Communications

Volumn 27, Issue 20, 1997, Pages 3565-3571

  Matsuda, Koyo ^a   Yanagisawa, Isao ^a   Isomura, Yasuo ^a   Mase, Toshiyasu ^a   Shibanuma, Tadao ^a  

^a ASTELLAS PHARMA INC   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

ACETAL; IMIDAZOLE 2 THIONE DERIVATIVE; ISOTHIOCYANIC ACID DERIVATIVE; THIOUREA DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CYCLIZATION; DRUG SYNTHESIS; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; REACTION ANALYSIS;

EID: 0030880642     PISSN: 00397911     EISSN: None     Source Type: Journal    
DOI: 10.1080/00397919708007078     Document Type: Article

References (7)

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3. McCarthy, J. R.; Matthews, D. P.; Broersma, R. J.; McDermott, R. D.; Kastner, P. R.; Hornsperger, J. -M.; Demeter, D. A.; Weintraub, H. J. R. and Whitten, J. P. ibid. 1990, 33, 1866.
4. a) Wohl, A. and Marckwald, W. Chem. Ber. 1889, 22, 568;
5. b) Marckwald, W. ibid. 1892, 25, 2354.
6. a) Jones, R. G. J. Am. Chem. Soc. 1949, 71, 383;
7. b) Jones, R. G.; Kornfeld, E. C.; McLaughlin, K. C. and Anderson, R. C. ibid. 1949, 71, 4000.