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European Journal of Medicinal Chemistry

Volumn 32, Issue 7-8, 1997, Pages 547-570

Synthesis and pharmacological evaluation of new cysLT1 receptor antagonists

(9) Griera, R a Armengol, M a Reyes, A a Alvarez, M a Palomer, A b Cabre F b Pascual, J b Garcia M L b Mauleon D b

a UNIVERSITY OF BARCELONA (Spain)

b Laboratorios Menarini (Spain)

Author keywords

4 quinolons; Acylsulfonamide; Antagonist; Leukotriene D4; Molecular modelling

Indexed keywords

4 QUINOLONE DERIVATIVE; LEUKOTRIENE RECEPTOR BLOCKING AGENT; SULFONAMIDE;

ANIMAL TISSUE; CONTROLLED STUDY; DRUG SYNTHESIS; GUINEA PIG; ILEUM; LUNG; MOLECULAR MODEL; NONHUMAN; REVIEW; SMOOTH MUSCLE RELAXATION;

EID: 0030878984 PISSN: 02235234 EISSN: None Source Type: Journal
DOI: 10.1016/S0223-5234(97)83282-5 Document Type: Article

Times cited : (10)

References (47)

1
- 0018710244
- Borgeat P, Samuelsson B (1979) J Biol Chem 254 (16), 7865-7869
- (1979) J Biol Chem , vol.254 , Issue.16 , pp. 7865-7869
- Borgeat, P.¹ Samuelsson, B.²

2
- 0018803640
- Hammarstrom S, Murphy R, Samuelsson B, Clark DA, Mioskowski CCh, Corey EJ (1979) Biochem Biophys Res Commun 91, 1266-1272
- (1979) Biochem Biophys Res Commun , vol.91 , pp. 1266-1272
- Hammarstrom, S.¹ Murphy, R.² Samuelsson, B.³ Clark, D.A.⁴ Mioskowski, C.Ch.⁵ Corey, E.J.⁶

3
- 0009970260
- Borgeat P, Samuelsson B (1979) Proc Natl Acad Sci USA 76 (5), 2148-2152
- (1979) Proc Natl Acad Sci USA , vol.76 , Issue.5 , pp. 2148-2152
- Borgeat, P.¹ Samuelsson, B.²

4
- 0018418754
- Borgeat P, Samuelsson B (1979) J Biol Chem 254, 2643-2646
- (1979) J Biol Chem , vol.254 , pp. 2643-2646
- Borgeat, P.¹ Samuelsson, B.²

5
- 0027281182
- Ar JP, Lee TH (1993) Clin Sci 84, 501-510
- (1993) Clin Sci , vol.84 , pp. 501-510
- Ar, J.P.¹ Lee, T.H.²

6
- 0029152856
- Hay DWP, Torphy TJ, Undem BJ (1995) Trends Pharmacol Sci 16, 304-311
- (1995) Trends Pharmacol Sci , vol.16 , pp. 304-311
- Hay, D.W.P.¹ Torphy, T.J.² Undem, B.J.³

7
- 0029181278
- Fort-Hutchinson WA (1995) Adv Prostaglandin Thromboxane Leukotriene Res 23, 69-74
- (1995) Adv Prostaglandin Thromboxane Leukotriene Res , vol.23 , pp. 69-74
- Fort-Hutchinson, W.A.¹

8
- 0024453185
- Gardiner PJ (1989) Pharmacol Ther 44, 1-62
- (1989) Pharmacol Ther , vol.44 , pp. 1-62
- Gardiner, P.J.¹

9
- 21144478185
- Von Sprecher A, Beck A, Gerspacher M, Bray MA (1992) Chimia 46, 304-311
- (1992) Chimia , vol.46 , pp. 304-311
- Von Sprecher, A.¹ Beck, A.² Gerspacher, M.³ Bray, M.A.⁴

10
- 0028896048
- Koch K, Burgess E (1995) Expert Opin Ther Pat 5 (2), 127-155
- (1995) Expert Opin Ther Pat , vol.5 , Issue.2 , pp. 127-155
- Koch, K.¹ Burgess, E.²

11
- 0027272829
- Larsen JS, Acosta EP (1993) Ann Pharmacother 27 (7-8), 898-903
- (1993) Ann Pharmacother , vol.27 , Issue.7-8 , pp. 898-903
- Larsen, J.S.¹ Acosta, E.P.²

12
- 0029156140
- Pauwels RA, Joos GF, Kips JC (1995) Leukotrienes Ther Target Asthma Allergy 50 (8), 615-622
- (1995) Leukotrienes Ther Target Asthma Allergy , vol.50 , Issue.8 , pp. 615-622
- Pauwels, R.A.¹ Joos, G.F.² Kips, J.C.³

13
- 0029132046
- Chung KF (1995) Eur Res J 8 (7), 1203-1213
- (1995) Eur Res J , vol.8 , Issue.7 , pp. 1203-1213
- Chung, K.F.¹

14
- 0025300626
- Matassa VG, Maduskuie TP, Shapiro HS et al (1990) J Med Chem 33, 1781-1790
- (1990) J Med Chem , vol.33 , pp. 1781-1790
- Matassa, V.G.¹ Maduskuie, T.P.² Shapiro, H.S.³

15
- 0023848175
- Nakai H, Konno M, Kosuge S et al (1988) J Med Chem 31, 84-91
- (1988) J Med Chem , vol.31 , pp. 84-91
- Nakai, H.¹ Konno, M.² Kosuge, S.³

16
- 0025879330
- Huang FC, Galemmo RA, Poli GB et al (1991) J Med Chem 34, 1704-1707
- (1991) J Med Chem , vol.34 , pp. 1704-1707
- Huang, F.C.¹ Galemmo, R.A.² Poli, G.B.³

17
- 0029054404
- Glass M (1995) Eur Resp Rev 5 (26), 120-123
- (1995) Eur Resp Rev , vol.5 , Issue.26 , pp. 120-123
- Glass, M.¹

18
- 0010484698
- Grossman J, Bronsky E, Busse W et al (1995) J Allergy Clin Immunol 95 (1), 352
- (1995) J Allergy Clin Immunol , vol.95 , Issue.1 , pp. 352
- Grossman, J.¹ Bronsky, E.² Busse, W.³

19
- 85058206310
- Grossman J, Bronsky E, Busse E et al (1995) Eur Resp J 8 (suppl 19) 288S
- (1995) Eur Resp J , vol.8 , Issue.SUPPL. 19
- Grossman, J.¹ Bronsky, E.² Busse, E.³

20
- 0013541089
- John Wiley and Sons, NY
- Jones G (1977) In: The Chemistry of Heterocyclic Compounds. John Wiley and Sons, NY, vol 32, part I, 143
- (1977) The Chemistry of Heterocyclic Compounds , vol.32 , Issue.PART I , pp. 143
- Jones, G.¹

21
- 0017881232
- Cairns H, Payne AR (1978) J Heterocycl Chem 15, 551-553
- (1978) J Heterocycl Chem , vol.15 , pp. 551-553
- Cairns, H.¹ Payne, A.R.²

22
- 0343902917
- Venturella P, Bellino A, Marino ML, Piozzi F (1990) Gazz Chim Ital 100, 678-681
- (1990) Gazz Chim Ital , vol.100 , pp. 678-681
- Venturella, P.¹ Bellino, A.² Marino, M.L.³ Piozzi, F.⁴

23
- 0025237214
- Huang FC, Galemmo RA, Johnson WH et al (1990) J Med Chem 33, 1194-1200
- (1990) J Med Chem , vol.33 , pp. 1194-1200
- Huang, F.C.¹ Galemmo, R.A.² Johnson, W.H.³

24
- 84943961938
- Cassis R, Tapia R, Valderrama JA (1985) Synth Commun 15, 125-133
- (1985) Synth Commun , vol.15 , pp. 125-133
- Cassis, R.¹ Tapia, R.² Valderrama, J.A.³

25
- 84986369514
- Huang X, Chen B (1987) Synthesis 480-481
- (1987) Synthesis , pp. 480-481
- Huang, X.¹ Chen, B.²

26
- 85082554940
- Chen B, Huang X, Wang J (1987) Synthesis 482-483
- (1987) Synthesis , pp. 482-483
- Chen, B.¹ Huang, X.² Wang, J.³

27
- 0012017104
- Lauer WM, Kaslow CE (1949) Org Synth Coll III, 580-583
- (1949) Org Synth Coll , vol.3 , pp. 580-583
- Lauer, W.M.¹ Kaslow, C.E.²

28
- 0009777389
- Bieber MP (1951) Comptes Rendus Acad Sci Paris 233, 655-657
- (1951) Comptes Rendus Acad Sci Paris , vol.233 , pp. 655-657
- Bieber, M.P.¹

29
- 37049079087
- Alvarez M, Salas M, Rigat LI, de Veciana A, Joule JA (1992) J Chem Soc Perkin Trans I 351-356
- (1992) J Chem Soc Perkin Trans , vol.1 , pp. 351-356
- Alvarez, M.¹ Salas, M.² Rigat, L.I.³ De Veciana, A.⁴ Joule, J.A.⁵

30
- 85030298944
- Jpn Kokai Tokyo Koho 03 95, 144 [9195, 144] (Cl C07C225/22) 19 Apr 1991, appl 89/202, 682, 04 Aug 1989
- Wakatsuka H, Nakai H, Okumoto I (1991) Jpn Kokai Tokyo Koho 03 95, 144 [9195, 144] (Cl C07C225/22) 19 Apr 1991, appl 89/202, 682, 04 Aug 1989
- (1991)
- Wakatsuka, H.¹ Nakai, H.² Okumoto, I.³

31
- 0342597179
- (Sanz F, Manaut F, eds) Prous, Barcelona
- Palomer A, Giolitti A, García ML, Cabré F, Mauleón D, Carganico G (1995) in: Trends in QSAR and Molecular Modelling '94 (Sanz F, Manaut F, eds) Prous, Barcelona
- (1995) Trends in QSAR and Molecular Modelling '94
- Palomer, A.¹ Giolitti, A.² García, M.L.³ Cabré, F.⁴ Mauleón, D.⁵ Carganico, G.⁶

32
- 0005123846
- (Müller K, ed) Escom, Leiden
- Sprague P (1995) In: De Novo Design (Müller K, ed) Escom, Leiden, 1-20
- (1995) De Novo Design , pp. 1-20
- Sprague, P.¹

33
- 0023751431
- Cramer III RD, Patterson DE, Bunce JD (1988) J Am Chem Soc 110, 5959-5967
- (1988) J Am Chem Soc , vol.110 , pp. 5959-5967
- Cramer R.D. III¹ Patterson, D.E.² Bunce, J.D.³

34
- 85030292018
- Pascual J, Fos E, García ML et al (1994) Proc XIIIth Int Symp Med Chem Paris, p 184
- (1994) Proc XIIIth Int Symp Med Chem Paris , pp. 184
- Pascual, J.¹ Fos, E.² García, M.L.³

35
- 0028550028
- Greene J, Kahn S, Savoj H, Sprague P, Teig S (1994) J Chem Inf Comput Sci 34 (6), 1297-1308
- (1994) J Chem Inf Comput Sci , vol.34 , Issue.6 , pp. 1297-1308
- Greene, J.¹ Kahn, S.² Savoj, H.³ Sprague, P.⁴ Teig, S.⁵

36
- 0025195923
- Matassa VG, Brown FJ, Bernstein PR et al (1990) J Med Chem 33, 2621-2629
- (1990) J Med Chem , vol.33 , pp. 2621-2629
- Matassa, V.G.¹ Brown, F.J.² Bernstein, P.R.³

37
- 84986512474
- Brooks BR, Bruccoleri RE, Olafson BD, States DJ, Swaninathan S, Karplus M (1983) J Comput Chem 4, 187-217
- (1983) J Comput Chem , vol.4 , pp. 187-217
- Brooks, B.R.¹ Bruccoleri, R.E.² Olafson, B.D.³ States, D.J.⁴ Swaninathan, S.⁵ Karplus, M.⁶

38
- 0029277503
- Smellie AS, Kahn SD, Teig SL (1995) J Chem Inf Comput Sci 35 (2), 285-294
- (1995) J Chem Inf Comput Sci , vol.35 , Issue.2 , pp. 285-294
- Smellie, A.S.¹ Kahn, S.D.² Teig, S.L.³

39
- 0029276206
- Smellie AS, Kahn SD, Teig SL (1995) J Chem Inf Comput Sci 35 (2), 295-304
- (1995) J Chem Inf Comput Sci , vol.35 , Issue.2 , pp. 295-304
- Smellie, A.S.¹ Kahn, S.D.² Teig, S.L.³

40
- 84986522856
- Smellie AS, Teig SL, Towbin P (1995) J Comput Chem 16 (2), 171-187
- (1995) J Comput Chem , vol.16 , Issue.2 , pp. 171-187
- Smellie, A.S.¹ Teig, S.L.² Towbin, P.³

41
- 0343467087
- Liu KC, Lu WC, Lee LC (1979) Taiwan I-Hsueh-Hui Tsa Chih 31, 80-90
- (1979) Taiwan I-Hsueh-Hui Tsa Chih , vol.31 , pp. 80-90
- Liu, K.C.¹ Lu, W.C.² Lee, L.C.³

42
- 0001921558
- Huang X, Chen B (1986) Synthesis 967-968
- (1986) Synthesis , pp. 967-968
- Huang, X.¹ Chen, B.²

43
- 0343031369
- Cidda C, Sleiter G (1980) Gazz Chim Ital 110, 155-162
- (1980) Gazz Chim Ital , vol.110 , pp. 155-162
- Cidda, C.¹ Sleiter, G.²

44
- 0018757383
- Denny WA, Atwell GJ, Baguley BC, Cain BF (1979) J Med Chem 22, 134-150
- (1979) J Med Chem , vol.22 , pp. 134-150
- Denny, W.A.¹ Atwell, G.J.² Baguley, B.C.³ Cain, B.F.⁴

45
- 0342597177
- Imperial Chemical Industries Ltd
- Crowter AF, Hepworth W, Morley JS (1960) Br Pat 835, 474, Imperial Chemical Industries Ltd
- (1960) Br Pat , vol.835 , pp. 474
- Crowter, A.F.¹ Hepworth, W.² Morley, J.S.³

46
- 0021647642
- Mong S, Wu HL, Clark MA, Stadel JM, Gleason JG, Crooke ST (1984) Prostaglandins 28, 805-822
- (1984) Prostaglandins , vol.28 , pp. 805-822
- Mong, S.¹ Wu, H.L.² Clark, M.A.³ Stadel, J.M.⁴ Gleason, J.G.⁵ Crooke, S.T.⁶

47
- 0025195923
- Matassa VG, Brown FJ, Bernstein PR et al (1990) J Med Chem 33, 2621-2629
- (1990) J Med Chem , vol.33 , pp. 2621-2629
- Matassa, V.G.¹ Brown, F.J.² Bernstein, P.R.³

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