106. Synthesis via a carbohydrate-derived Munchnone of pyrrolopyridines (indolizines) and imidazopyridines, and their evaluation as inhibitors of β- D-glucosidases

Helvetica Chimica Acta

Volumn 80, Issue 5, 1997, Pages 1443-1456

  Granier, Thierry ^a   Gaiser, Florian ^a   Hintermann, Lukas ^a   Vasella, Andrea ^a  

^a ETH ZURICH   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

BETA GLUCOSIDASE; IMIDAZOPYRAZINE DERIVATIVE; PYRROLOPYRIMIDINE DERIVATIVE;

ALKYLATION; ARTICLE; CARBOHYDRATE METABOLISM; DRUG SYNTHESIS; ENZYME INHIBITION; NONHUMAN; REACTION ANALYSIS; SIALYLATION; X RAY ANALYSIS;

EID: 0030873356     PISSN: 0018019X     EISSN: None     Source Type: Journal    
DOI: 10.1002/hlca.19970800509     Document Type: Article

References (12)

1. P. Ermert, A. Vasella, Helv. Chim. Acta 1991, 74, 2043.
2. A. Frankowski, C. Seliga, D. Bur, J. Streith, Helv. Chim. Acta 1991, 74, 934.
3. T. Aoyagi, H. Suda, K. Uotani, F. Kojima, T. Aoyama, K. Horiguchi, M. Hamada, T. Takeuchi, J. Antibiot. 1992, 45, 1404.
4. T. Aoyama, H. Naganawa, H. Suda, K. Uotani, T. Aoyagi, T. Takeuchi, J. Antibiot. 1992, 45, 1557.
5. P. Kefalas, D. S. Grierson, Tetrahedron Lett. 1993, 34, 3555.
6. K. Burgess, D. A. Chaplin, Heterocycles 1994, 37, 673.
7. K. Tatsuta, S. Miura, S. Ohta, H. Gunji, Tetrahedron Lett. 1995, 36, 1085
8. K. Tatsuta, S. Miura, Tetrahedron Lett. 1995, 36, 6721.
9. K. Tatsuta, Y. Ikeda, S. Miura, J. Antibiot. 1996, 49, 836.
10. K. Tatsuta, S. Miura, H. Gunji, Bull. Chem. Soc. Jpn. 1997, 70, 427.
11. T. D. Heightman, M. Locatelli, A. Vasella, Helv. Chim. Acta 1996, 79, 2190.
12. R. Hoos, A. Vasella, K. Rupitz, S. G. Withers, Carbohydr. Res. 1997, 295, 291.