Application of tumbling melt granulation (TMG) method for controlled enteric-release beads by coating mixture of hydrogenated castor oil and higher fatty acid

Chemical and Pharmaceutical Bulletin

Volumn 45, Issue 8, 1997, Pages 1332-1338

  Maejima, Toru ^a   Osawa, Takashi ^a   Nakajima, Kingo ^a   Kobayashi, Masao ^a  

^a MITSUBISHI TANABE PHARMA CORPORATION   (Japan)

Author keywords

Beads; Centrifugal fluidizing granulator; Controlled release; Entero soluble; Tumbling melt granulation; Wax

Indexed keywords

FATTY ACID; HYDROGENATED CASTOR OIL; ISONIAZID; ORGANIC SOLVENT; SALICYLIC ACID; STEARIC ACID; THEOPHYLLINE;

ARTICLE; DRUG BIOAVAILABILITY; DRUG PENETRATION; DRUG SOLUBILITY; ENTERIC COATED TABLET; STOMACH PH; SUSTAINED RELEASE PREPARATION;

EID: 0030867925     PISSN: 00092363     EISSN: None     Source Type: Journal    
DOI: 10.1248/cpb.45.1332     Document Type: Article

References (20)

1. Kobayashi M., Pharm. Tech. Jpn., 7, 711-718 (1991).
2. Miyajima M., Akatsu S., Satoh H., Pharm. Tech. Jpn, 8 1021-1027 (1992).
3. Fischer W., Boertz A., Davis S. S., Khosla R., Cawello W., Sandrock K., Cordes G., Pharm. Res., 4, 480-485 (1987).
4. Wilding I. R., Hardy J. G., Maccari M., Ravelli V., Davis S. S., Int. J. Pharm., 76, 133-143 (1991).
5. Evans D. F., Pye G., Bramley R., Clark A. G., Tyson T. J., Hardcastle J. D., Gut, 29, 1035-1041 (1988).
6. Suzuki Y., Tsukada T., Nagafuji N., Tomoda Y., Hayashi T., Tanaka H., Fujimoto A., Nakajima C., Shima K. Ogura T., Takagishi Y., Yakuzaigaku, 53, 201-209 (1993).
7. Shimano K., Kondo O., Miwa A., Higashi Y., Koyama I., Yoshida T., Ito Y., Hirose J., Goto S., Yakuzaigaku, 54, 135-148 (1994).
8. Suzuki Y., Takeyama T., Fujii T., Noda K., Sakamoto T., Abstracts of Papers, The 108th Annual Meeting of Pharmaceutical Society of Japan, Hiroshima, April 1988.
9. Maki T., Ueki N., Ozawa Y., J. Soc. Technol. Jpn., 25, 338-343 (1988).
10. Akiyama Y., Yoshioka M., Horibe H., Hirai S., Kitamori N., Toguchi H., J. Controlled Release, 26, 1-10 (1993).
11. Yoshitomi H., Kawamoto M., Masuda Y., Takahashi K., Yakuzaigaku, 50, 156-165 (1990).
12. Maejima T., Osawa T., Nakajima K., Kobayashi M., Chem. Pharm. Bull., 45, 904-910 (1997).
13. Maejima T., Osawa T., Nakajima K., Kobayashi M., Chem. Pharm. Bull., 40, 488-492 (1992).
14. Ozturk A. G., Ozturk S. S., Palsson B. O., Wheatley T. A., Dressman J. B., J. Controlled. Release, 14, 203-213 (1990).
15. Donbrow M., Friedman M., J. Pharm. Pharmacol., 27, 633-646 (1975).
16. Koida Y., Kobayashi M., Samejima M., Chem. Pharm. Bull., 35, 1538-1545 (1987).
17. Narisawa S., Yoshino H., Hirakawa Y., Noda K., Int. J. Pharm., 104, 95-106 (1994).
18. Madan P. L., Luzzi L. A., Price J. C., J. Pharm. Sci., 63, 280-284 (1974).
19. Haramiishi Y., Hishida J., Matsumoto N., Kataoka K., Abstracts of Papers, The 107th Annual Meeting of Pharmaceutical Society of Japan, Kyoto, April 1987.
20. The Association of Oil Chemistry, Japan (ed.), "Yushikagakubinran," Maruzen Company, Tokyo, 1990, p. 252.