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0343095203
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+ m/z 382.2130, found 382.2122.
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Mitsunobu, O.1
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0026010908
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The impurity resulted from the incomplete PyBOP coupling reaction due to the electron-withdrawing groups on the aromatic ring. For less nucleophilic substrates, the yield and purity could be improved by using PyBroP, a more reactive coupling reagent. See, Frérot, E.; Coste, J.; Pantaloni, A.; Dufour, M.-N.; Jouin, P. Tetrahedron 1991, 47, 259.
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