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Volumn 152, Issue 2, 1997, Pages 165-178

Percutaneous absorption of bendroflumethiazide from gel and membrane-controlled gel systems: An in vitro and in vivo study

Author keywords

Bendroflumethiazide; Gel; Hairless mouse skin; Membrane controlled; Percutaneous absorption; Rabbit

Indexed keywords

1 METHYL 2 PYRROLIDINONE; 2 PYRROLIDINONE; ALCOHOL; BENDROFLUMETHIAZIDE; CELLULOSE; ETHYLENE VINYL ACETATE COPOLYMER; MACROGOL 400; POLYACRYLIC ACID; POLYPROPYLENE; POLYURETHAN; SILICONE;

EID: 0030858822     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-5173(97)00088-4     Document Type: Article
Times cited : (5)

References (56)
  • 2
    • 0022000863 scopus 로고
    • Absorption through human skin of ibuprofen and flurbiprofen: Effect of dose variation, deposited drug films, occlusion and the penetration enhancer N-methyl 2-pyrrolidone
    • Akhter, S.A., Barry, B.W., 1985. Absorption through human skin of ibuprofen and flurbiprofen: effect of dose variation, deposited drug films, occlusion and the penetration enhancer N-methyl 2-pyrrolidone. J. Pharm. Pharmacol. 37, 27-37.
    • (1985) J. Pharm. Pharmacol. , vol.37 , pp. 27-37
    • Akhter, S.A.1    Barry, B.W.2
  • 3
    • 0017253868 scopus 로고
    • Effect of dimethyl sulfoxide on permeability of human skin in vitro
    • Astley, J.P., Levine, M., 1976. Effect of dimethyl sulfoxide on permeability of human skin in vitro. J. Pharm. Sci. 65, 210-215.
    • (1976) J. Pharm. Sci. , vol.65 , pp. 210-215
    • Astley, J.P.1    Levine, M.2
  • 4
    • 0023597397 scopus 로고
    • Mode of action of penetration enhancers in human skin
    • Barry, B.W., 1987. Mode of action of penetration enhancers in human skin. J. Cont. Rel. 6, 85.
    • (1987) J. Cont. Rel. , vol.6 , pp. 85
    • Barry, B.W.1
  • 5
    • 0023235207 scopus 로고
    • Effect of penetration enhancers on the skin permeation of mannitol, hydrocortisone and progesterone through human skin
    • Barry, B.W., Bennett, S.L., 1987. Effect of penetration enhancers on the skin permeation of mannitol, hydrocortisone and progesterone through human skin. J. Pharm. Pharmacol. 39, 535-546.
    • (1987) J. Pharm. Pharmacol. , vol.39 , pp. 535-546
    • Barry, B.W.1    Bennett, S.L.2
  • 6
    • 0019429646 scopus 로고
    • The effect of cosmetic vehicles on the permeation of N-nitrosodiethanolamine through excised human skin
    • Bronaugh, R.L., Congdon, E.R., Scheuplein, R.J., 1981. The effect of cosmetic vehicles on the permeation of N-nitrosodiethanolamine through excised human skin. J. Invest. Dermatol. 76, 94-96.
    • (1981) J. Invest. Dermatol. , vol.76 , pp. 94-96
    • Bronaugh, R.L.1    Congdon, E.R.2    Scheuplein, R.J.3
  • 8
    • 0009912609 scopus 로고
    • Transdermal therapeutic systems
    • Robinson, J.R., Lee, V.H. (Eds.), Marcel Dekker, New York
    • Chien, Y.W., 1987. Transdermal therapeutic systems. In: Robinson, J.R., Lee, V.H. (Eds.), Controlled Drug Delivery: Fundamentals and Applications, vol. 29. Marcel Dekker, New York, pp. 524-552.
    • (1987) Controlled Drug Delivery: Fundamentals and Applications , vol.29 , pp. 524-552
    • Chien, Y.W.1
  • 9
    • 0342865675 scopus 로고
    • Transdermal controlled release systems
    • Langer, R.S., Wise, D.L. (Eds.), CRC Press, Boca Raton, FL
    • Cleary, G.W., 1984. Transdermal controlled release systems. In: Langer, R.S., Wise, D.L. (Eds.), Medical Applications of Controlled Release, Classes of Systems, vol. 1. CRC Press, Boca Raton, FL, pp. 203-251.
    • (1984) Medical Applications of Controlled Release, Classes of Systems , vol.1 , pp. 203-251
    • Cleary, G.W.1
  • 10
    • 0021855110 scopus 로고
    • Effect of fatty acids and alcohols on the penetration of acyclovir across human skin in vitro
    • Cooper, E.R., Merritt, E.W., Smith, R.L., 1985. Effect of fatty acids and alcohols on the penetration of acyclovir across human skin in vitro. J. Pharm. Sci. 74, 688.
    • (1985) J. Pharm. Sci. , vol.74 , pp. 688
    • Cooper, E.R.1    Merritt, E.W.2    Smith, R.L.3
  • 11
    • 0019403775 scopus 로고
    • Effect of non-ionic surfactants on penetration of dissolved benzocaine through hairless mouse skin
    • Dalvi, U.G., Zatz, J.L., 1984. Effect of non-ionic surfactants on penetration of dissolved benzocaine through hairless mouse skin. J. Soc. Cosmet. Chem. 32, 87-94.
    • (1984) J. Soc. Cosmet. Chem. , vol.32 , pp. 87-94
    • Dalvi, U.G.1    Zatz, J.L.2
  • 12
    • 0018855548 scopus 로고
    • Vehicle effects in percutaneous absorption: In vitro study of influence of solvent power and microscopic viscosity of vehicle on benzocaine release from suspension hydrogels
    • Di Colo, G., Carelli, V., Giannaccini, B., Serafini, M., Bottari, F., 1980. Vehicle effects in percutaneous absorption: in vitro study of influence of solvent power and microscopic viscosity of vehicle on benzocaine release from suspension hydrogels. J. Pharm. Sci. 69, 387-391.
    • (1980) J. Pharm. Sci. , vol.69 , pp. 387-391
    • Di Colo, G.1    Carelli, V.2    Giannaccini, B.3    Serafini, M.4    Bottari, F.5
  • 14
    • 0019155972 scopus 로고
    • Permeation of hairless mouse skin I: Experimental methods and comparison with human epidermal permeation by alkanols
    • Durrheim, H., Flynn, G.L., Higuchi, W.I., Behl, C.R., 1980. Permeation of hairless mouse skin I: Experimental methods and comparison with human epidermal permeation by alkanols. J. Pharm. Sci. 69, 781-786.
    • (1980) J. Pharm. Sci. , vol.69 , pp. 781-786
    • Durrheim, H.1    Flynn, G.L.2    Higuchi, W.I.3    Behl, C.R.4
  • 15
    • 0002676005 scopus 로고
    • Measurement of drug release from topical gels using two types of apparatus
    • Fares, H.M., Zatz, J.L., 1995. Measurement of drug release from topical gels using two types of apparatus. Pharm. Technol. 19, 52-58.
    • (1995) Pharm. Technol. , vol.19 , pp. 52-58
    • Fares, H.M.1    Zatz, J.L.2
  • 16
    • 0342737088 scopus 로고
    • Bendroflumethiazide
    • Florey, K. (Ed.), Academic Press, New York
    • Florey, K., Russo-Alesi, F.M., 1976. Bendroflumethiazide. In: Florey, K. (Ed.), Analytical Profiles of Drug Substances, vol. 5. Academic Press, New York, pp. 2-19.
    • (1976) Analytical Profiles of Drug Substances , vol.5 , pp. 2-19
    • Florey, K.1    Russo-Alesi, F.M.2
  • 17
    • 0015257617 scopus 로고
    • Membrane diffusion III: Influence of solvent composition and permeant solubility on membrane transport
    • Flynn, G.L., Smith, R.W., 1972. Membrane diffusion III: Influence of solvent composition and permeant solubility on membrane transport. J. Pharm. Sci. 61, 61-66.
    • (1972) J. Pharm. Sci. , vol.61 , pp. 61-66
    • Flynn, G.L.1    Smith, R.W.2
  • 18
    • 0025030097 scopus 로고
    • Oleic acid: Its effect on stratum corneum in relation to transdermal drug delivery
    • Francoeur, M.L., Golden, G.M., Potts, R.O., 1990. Oleic acid: its effect on stratum corneum in relation to transdermal drug delivery. Pharm. Res. 7, 621.
    • (1990) Pharm. Res. , vol.7 , pp. 621
    • Francoeur, M.L.1    Golden, G.M.2    Potts, R.O.3
  • 19
    • 0343171492 scopus 로고
    • The development and in vitro characterization of gelatin films as a uniphasic transdermal drug delivery system
    • Gabriel, D.L., Simonelli, A.P., 1988. The development and in vitro characterization of gelatin films as a uniphasic transdermal drug delivery system. Pharm. Res. 5, 78.
    • (1988) Pharm. Res. , vol.5 , pp. 78
    • Gabriel, D.L.1    Simonelli, A.P.2
  • 21
    • 0023112902 scopus 로고
    • Transdermal drug delivery: A perspective
    • Guy, R.H., Hadgraft, J., 1987. Transdermal drug delivery: a perspective. J. Cont. Rel. 4, 237-251.
    • (1987) J. Cont. Rel. , vol.4 , pp. 237-251
    • Guy, R.H.1    Hadgraft, J.2
  • 22
    • 73049177744 scopus 로고
    • Analysis of data on the medicament release from ointments
    • Higuchi, W.I., 1962. Analysis of data on the medicament release from ointments. J. Pharm. Sci. 51, 802-804.
    • (1962) J. Pharm. Sci. , vol.51 , pp. 802-804
    • Higuchi, W.I.1
  • 23
    • 0001902009 scopus 로고
    • Prodrugs in transdermal delivery
    • Kydonieus, A.F., Berner, B. (Eds.), CRC Press, Boca Raton, FL
    • Higuchi, W.I., Yu, C.D., 1987. Prodrugs in transdermal delivery. In: Kydonieus, A.F., Berner, B. (Eds.), Transdermal Delivery of Drugs, vol. 3. CRC Press, Boca Raton, FL, pp. 43-83.
    • (1987) Transdermal Delivery of Drugs , vol.3 , pp. 43-83
    • Higuchi, W.I.1    Yu, C.D.2
  • 24
    • 0008972454 scopus 로고
    • Mechanism of ethanol effects on the simultaneous transport and metabolism of β-estradiol in hairless mouse skin
    • Controlled Release Society, Lincolnshire, IL
    • Higuchi, W.I., Liu, P., Ghanem, A.H., Song, W., 1987. Mechanism of ethanol effects on the simultaneous transport and metabolism of β-estradiol in hairless mouse skin. In: Proceedings of the International Symposium on Controlled Release and Bioactive Materials, vol. 14. Controlled Release Society, Lincolnshire, IL, pp. 101-102.
    • (1987) Proceedings of the International Symposium on Controlled Release and Bioactive Materials , vol.14 , pp. 101-102
    • Higuchi, W.I.1    Liu, P.2    Ghanem, A.H.3    Song, W.4
  • 25
    • 0022803030 scopus 로고
    • Determination of bendroflumethiazide in plasma by high performance liquid chromatography and fluorescence detection
    • Hikal, A.H., 1986. Determination of bendroflumethiazide in plasma by high performance liquid chromatography and fluorescence detection. J. Liq. Chromat. 9, 2937-2943.
    • (1986) J. Liq. Chromat. , vol.9 , pp. 2937-2943
    • Hikal, A.H.1
  • 26
    • 0020559714 scopus 로고
    • Polymer matrix considerations for transdermal devices
    • Keith, A.D., 1983. Polymer matrix considerations for transdermal devices. Drug Dev. Ind. Pharm. 9, 604-625.
    • (1983) Drug Dev. Ind. Pharm. , vol.9 , pp. 604-625
    • Keith, A.D.1
  • 29
    • 0030013239 scopus 로고    scopus 로고
    • Formulation development of a transdermal drug delivery system for amlodipine base
    • McDaid, D.M., Deasy, P.B., 1996. Formulation development of a transdermal drug delivery system for amlodipine base. Int. J. Pharm. 133, 71-83.
    • (1996) Int. J. Pharm. , vol.133 , pp. 71-83
    • McDaid, D.M.1    Deasy, P.B.2
  • 30
    • 0027223972 scopus 로고
    • Solubility and in vitro percutaneous absorption of teracaine from solvents of propylene glycol and saline
    • Miller, K.J., Rao, Y.K., Goodwin, S.R., Westermann-Clark, G.B., Shah, D.O., 1993. Solubility and in vitro percutaneous absorption of teracaine from solvents of propylene glycol and saline. Int. J. Pharm. 98, 101.
    • (1993) Int. J. Pharm. , vol.98 , pp. 101
    • Miller, K.J.1    Rao, Y.K.2    Goodwin, S.R.3    Westermann-Clark, G.B.4    Shah, D.O.5
  • 32
    • 0022537849 scopus 로고
    • Penetration enhancing effect of azone on the transport of 5-fluorouracil across hairless mouse skin
    • Morimoto, Y., Sugibayashi, K., Hosoya, K., Higuchi, W.I., 1986. Penetration enhancing effect of azone on the transport of 5-fluorouracil across hairless mouse skin. Int. J. Pharm. 32, 31-38.
    • (1986) Int. J. Pharm. , vol.32 , pp. 31-38
    • Morimoto, Y.1    Sugibayashi, K.2    Hosoya, K.3    Higuchi, W.I.4
  • 33
    • 0343171490 scopus 로고
    • Percutaneous absorption of propranolol from gel ointment
    • Nagai, T., Santoh, Y., Nambu, N., 1983. Percutaneous absorption of propranolol from gel ointment. Acta Pharm. Suec. 20, 47-48.
    • (1983) Acta Pharm. Suec. , vol.20 , pp. 47-48
    • Nagai, T.1    Santoh, Y.2    Nambu, N.3
  • 34
    • 0021845217 scopus 로고
    • Percutaneous absorption of propranolol from gel ointment in rabbits
    • Nagai, T., Santoh, Y., Nambu, N., Machida, Y., 1985. Percutaneous absorption of propranolol from gel ointment in rabbits. J. Cont. Rel. 1, 239-246.
    • (1985) J. Cont. Rel. , vol.1 , pp. 239-246
    • Nagai, T.1    Santoh, Y.2    Nambu, N.3    Machida, Y.4
  • 35
    • 0029944428 scopus 로고    scopus 로고
    • Differences in penetration-enhancing effect of azone through excised rabbit, rat, hairless mouse, guinea pig and human skins
    • Niazy, E.M., 1996. Differences in penetration-enhancing effect of azone through excised rabbit, rat, hairless mouse, guinea pig and human skins. Int. J. Pharm. 130, 225-230.
    • (1996) Int. J. Pharm. , vol.130 , pp. 225-230
    • Niazy, E.M.1
  • 36
    • 0025242631 scopus 로고
    • Mechanism for the enhancement effect of fatty acids on the percutaneous absorption of propranolol
    • Ogiso, T., Shintani, M., 1990. Mechanism for the enhancement effect of fatty acids on the percutaneous absorption of propranolol. J. Pharm. Sci. 79, 235.
    • (1990) J. Pharm. Sci. , vol.79 , pp. 235
    • Ogiso, T.1    Shintani, M.2
  • 37
    • 0027223973 scopus 로고
    • Percutaneous absorption of terodiline and the membrane-controlled transdermal therapeutic system
    • Ogiso, T., Iwaki, M., Tanino, T., Yatomi, M., Tsujimoto, C., 1993. Percutaneous absorption of terodiline and the membrane-controlled transdermal therapeutic system. Int. J. Pharm. 98, 113-120.
    • (1993) Int. J. Pharm. , vol.98 , pp. 113-120
    • Ogiso, T.1    Iwaki, M.2    Tanino, T.3    Yatomi, M.4    Tsujimoto, C.5
  • 38
    • 0025733949 scopus 로고
    • Development and evaluation of an intracutaneous depot formulation of corticosteroids using transcutol as a cosolvent: In-vitro, ex-vivo and in-vivo rat studies
    • Panchagnula, R., Ritschel, W.A., 1991. Development and evaluation of an intracutaneous depot formulation of corticosteroids using transcutol as a cosolvent: in-vitro, ex-vivo and in-vivo rat studies. J. Pharm. Pharmacol. 43, 609-614.
    • (1991) J. Pharm. Pharmacol. , vol.43 , pp. 609-614
    • Panchagnula, R.1    Ritschel, W.A.2
  • 39
    • 0028215123 scopus 로고
    • Topical formulation development of a novel thymidylate synthase inhibitor for the treatment of psoriasis
    • Pavliv, L., Freebern, K., Wilke, T., Chiang, C.C., Shetty, B., Tyle, P., 1994. Topical formulation development of a novel thymidylate synthase inhibitor for the treatment of psoriasis. Int. J. Pharm. 105, 227-233.
    • (1994) Int. J. Pharm. , vol.105 , pp. 227-233
    • Pavliv, L.1    Freebern, K.2    Wilke, T.3    Chiang, C.C.4    Shetty, B.5    Tyle, P.6
  • 40
    • 0023004097 scopus 로고
    • The effect of a rate controlling membrane on release from poly-HEMA hydrogels
    • Pywell, E.J., Yalkowsky, S.H., Collett, J.H., 1986. The effect of a rate controlling membrane on release from poly-HEMA hydrogels. Drug Dev. Ind. Pharm. 12, 1767-1775.
    • (1986) Drug Dev. Ind. Pharm. , vol.12 , pp. 1767-1775
    • Pywell, E.J.1    Yalkowsky, S.H.2    Collett, J.H.3
  • 43
    • 0029954232 scopus 로고    scopus 로고
    • Application of kinetic model to in vitro percutaneous permeation of drugs
    • Shah, J.C., 1996. Application of kinetic model to in vitro percutaneous permeation of drugs. Int. J. Pharm. 133, 179-189.
    • (1996) Int. J. Pharm. , vol.133 , pp. 179-189
    • Shah, J.C.1
  • 44
    • 0022645792 scopus 로고
    • The influence of azone, propylene glycol and polyethylene glycol on the in vitro skin permeation of trifluorthymidine
    • Sheth, N.V., Freeman, D.J., Higuchi, W.I., Spruance, S.L., 1986. The influence of azone, propylene glycol and polyethylene glycol on the in vitro skin permeation of trifluorthymidine. Int. J. Pharm. 28, 201-209.
    • (1986) Int. J. Pharm. , vol.28 , pp. 201-209
    • Sheth, N.V.1    Freeman, D.J.2    Higuchi, W.I.3    Spruance, S.L.4
  • 45
    • 0021748490 scopus 로고
    • Penetration enhancement in human skin: Effect of 2-pyrrolidone, dimethylformamide, and increased hydration on finite dose permeation of aspirin and caffeine
    • Southwell, D., Barry, B.W., 1984. Penetration enhancement in human skin: effect of 2-pyrrolidone, dimethylformamide, and increased hydration on finite dose permeation of aspirin and caffeine. Int. J. Pharm. 22, 291-298.
    • (1984) Int. J. Pharm. , vol.22 , pp. 291-298
    • Southwell, D.1    Barry, B.W.2
  • 46
    • 0343607052 scopus 로고
    • Release of drugs from homogenous ointments containing drug in solution
    • Sprang-Brunner, B.H., Speiser, P.P., 1975. Release of drugs from homogenous ointments containing drug in solution. J. Pharm. Pharmacol. 28, 23-28.
    • (1975) J. Pharm. Pharmacol. , vol.28 , pp. 23-28
    • Sprang-Brunner, B.H.1    Speiser, P.P.2
  • 47
    • 0019940117 scopus 로고
    • Enhanced percutaneous penetration with 1-dodecylazacycloheptan-2-one
    • Stoughton, R.B., 1982. Enhanced percutaneous penetration with 1-dodecylazacycloheptan-2-one. Arch. Dermatol. 118, 474-477.
    • (1982) Arch. Dermatol. , vol.118 , pp. 474-477
    • Stoughton, R.B.1
  • 48
    • 0343171487 scopus 로고
    • Azone: A new non-toxic enhancer of cutaneous penetration
    • Stoughton, R.B., McClure, W.O., 1985. Azone: a new non-toxic enhancer of cutaneous penetration. Drug Dev. Ind. Pharm. 37, 578-580.
    • (1985) Drug Dev. Ind. Pharm. , vol.37 , pp. 578-580
    • Stoughton, R.B.1    McClure, W.O.2
  • 49
    • 0342723195 scopus 로고    scopus 로고
    • Collagen membrane controlled transdermal delivery of propanolol hydrochloride
    • Thacharodi, D., Rao, K.P., 1996. Collagen membrane controlled transdermal delivery of propanolol hydrochloride. Int. J. Pharm. 131, 97-99.
    • (1996) Int. J. Pharm. , vol.131 , pp. 97-99
    • Thacharodi, D.1    Rao, K.P.2
  • 50
    • 0018741719 scopus 로고
    • Effects of polyoxypropylene 15 stearyl ether and propylene glycol on percutaneous penetration rate of diflorasone diacetate
    • Turi, J.S., Danielson, D., Woltersom, J.W., 1979. Effects of polyoxypropylene 15 stearyl ether and propylene glycol on percutaneous penetration rate of diflorasone diacetate. J. Pharm. Sci. 68, 275.
    • (1979) J. Pharm. Sci. , vol.68 , pp. 275
    • Turi, J.S.1    Danielson, D.2    Woltersom, J.W.3
  • 52
    • 0025741493 scopus 로고
    • Aspects of the transdermal delivery of prostaglandins
    • Watkinson, A.C., Madgraft, J., Bye, A., 1991. Aspects of the transdermal delivery of prostaglandins. Int. J. Pharm. 74, 229-236.
    • (1991) Int. J. Pharm. , vol.74 , pp. 229-236
    • Watkinson, A.C.1    Madgraft, J.2    Bye, A.3
  • 54
    • 0021916025 scopus 로고
    • In vitro and in vivo release of nitroglycerine from a transdermal therapeutic system
    • Wolff, M., Cordes, G., Luckow, V., 1988. In vitro and in vivo release of nitroglycerine from a transdermal therapeutic system. Pharm. Res. 2, 23-29.
    • (1988) Pharm. Res. , vol.2 , pp. 23-29
    • Wolff, M.1    Cordes, G.2    Luckow, V.3
  • 55
    • 0021922963 scopus 로고
    • Vehicle effect on topical delivery III. Effect of azone on the percutaneous permeation of metronidazole and propylene glycol
    • Wotton, P.K., Mollgaard, B., Hadgraft, J., Hoelgaard, A., 1985. Vehicle effect on topical delivery III. Effect of azone on the percutaneous permeation of metronidazole and propylene glycol. Int. J. Pharm. 24, 19-26.
    • (1985) Int. J. Pharm. , vol.24 , pp. 19-26
    • Wotton, P.K.1    Mollgaard, B.2    Hadgraft, J.3    Hoelgaard, A.4


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