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Volumn 282, Issue 2, 1997, Pages 920-927

WIN 35,428 and mazindol are mutually exclusive in binding to the cloned human dopamine transporter

Author keywords

[No Author keywords available]

Indexed keywords

3BETA (4 FLUOROPHENYL) 2BETA TROPANECARBOXYLIC ACID METHYL ESTER; COCAINE DERIVATIVE; COMPLEMENTARY DNA; DOPAMINE TRANSPORTER; MAZINDOL; RADIOLIGAND;

EID: 0030839892     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (9)

References (45)
  • 3
    • 0026507640 scopus 로고
    • Expression of a single dopamine transporter cDNA can confer two cocaine binding sites
    • BOJA, J. W., MARKHAM, L., PATEL, A., UHL, G. AND KUHAR, M. J.: Expression of a single dopamine transporter cDNA can confer two cocaine binding sites. Neuroreport 3: 247-248, 1992.
    • (1992) Neuroreport , vol.3 , pp. 247-248
    • Boja, J.W.1    Markham, L.2    Patel, A.3    Uhl, G.4    Kuhar, M.J.5
  • 4
    • 0028577297 scopus 로고
    • Chimeric dopamine-norepinephrine transporters delineate structural domains influencing selectivity for catecholamines and 1-methyl-4-phenylpyridinium
    • BUCK, K. J. AND AMARA, S. G.: Chimeric dopamine-norepinephrine transporters delineate structural domains influencing selectivity for catecholamines and 1-methyl-4-phenylpyridinium. Proc. Natl. Acad. Sci. USA 91: 12584-12588, 1994.
    • (1994) Proc. Natl. Acad. Sci. USA , vol.91 , pp. 12584-12588
    • Buck, K.J.1    Amara, S.G.2
  • 5
    • 0023632425 scopus 로고
    • 3H]cocaine in striatum and its relationship to the dopamine transporter
    • 3H]cocaine in striatum and its relationship to the dopamine transporter, Membr. Biochem. 7: 87-106, 1987.
    • (1987) Membr. Biochem. , vol.7 , pp. 87-106
    • Calligaro, D.O.1    Eldefrawi, M.E.2
  • 6
    • 0026566383 scopus 로고
    • Cocaine receptor. Biochemical characterization and structure-activity relationships of cocaine analogues at the dopamine transporter
    • CARROLL, F. I., LEWIN, A. H., BOJA, J. W. AND KUHAR, M. J.: Cocaine receptor. Biochemical characterization and structure-activity relationships of cocaine analogues at the dopamine transporter. J. Med. Chem. 35: 969-981, 1992.
    • (1992) J. Med. Chem. , vol.35 , pp. 969-981
    • Carroll, F.I.1    Lewin, A.H.2    Boja, J.W.3    Kuhar, M.J.4
  • 7
    • 0028180477 scopus 로고
    • 3H]WIN 35,428 binding to the dopamine uptake carrier. I. Effect of tonicity and buffer composition
    • 3H]WIN 35,428 binding to the dopamine uptake carrier. I. Effect of tonicity and buffer composition. J. Neurosci. Methods 51: 23-30, 1994.
    • (1994) J. Neurosci. Methods , vol.51 , pp. 23-30
    • Coffey, L.L.1    Reith, M.E.A.2
  • 8
    • 0018001339 scopus 로고
    • Simultaneous analysis of families of sigmoidal curves: Application to bioassay, radioligand assay, and physiological dose-response curves
    • DELEAN, A., MUNSON, P. J. AND RODBARD, D.: Simultaneous analysis of families of sigmoidal curves: Application to bioassay, radioligand assay, and physiological dose-response curves. Am. J. Physiol. 235: E97-E102, 1978.
    • (1978) Am. J. Physiol. , vol.235
    • Delean, A.1    Munson, P.J.2    Rodbard, D.3
  • 10
    • 0023958554 scopus 로고
    • Estimation of the affinities of allosteric ligands using radioligand binding and pharmacological null methods
    • EHLERT, F. J.: Estimation of the affinities of allosteric ligands using radioligand binding and pharmacological null methods. Mol. Pharmacol. 33: 187-194, 1988.
    • (1988) Mol. Pharmacol. , vol.33 , pp. 187-194
    • Ehlert, F.J.1
  • 12
    • 0029064866 scopus 로고
    • Characterization of a recombinant human dopamine transporter in multiple cell lines
    • ESHLEMAN, A. J., NEVE, R. L., JANOWSKY, A. AND NEVE, K. A.: Characterization of a recombinant human dopamine transporter in multiple cell lines. J. Pharmacol. Exp. Ther. 274: 276-283, 1995.
    • (1995) J. Pharmacol. Exp. Ther. , vol.274 , pp. 276-283
    • Eshleman, A.J.1    Neve, R.L.2    Janowsky, A.3    Neve, K.A.4
  • 14
    • 0027535205 scopus 로고
    • Molecular characterization of the dopamine transporter
    • GIROS, B. AND CARON, M. G.: Molecular characterization of the dopamine transporter. Trends Pharmacol. Sci. 14: 43-49, 1993.
    • (1993) Trends Pharmacol. Sci. , vol.14 , pp. 43-49
    • Giros, B.1    Caron, M.G.2
  • 15
    • 0027049060 scopus 로고
    • Cloning, pharmacological characterization, and chromosome assignment of the human dopamine transporter
    • GIROS, B., EL MESTIKAWY, S., GODINOT, N., ZHENG, K., HAN, H., YANG-FENG, T. AND CARON, M. G.: Cloning, pharmacological characterization, and chromosome assignment of the human dopamine transporter. Mol. Pharmacol. 42: 383-390, 1992.
    • (1992) Mol. Pharmacol. , vol.42 , pp. 383-390
    • Giros, B.1    El Mestikawy, S.2    Godinot, N.3    Zheng, K.4    Han, H.5    Yang-Feng, T.6    Caron, M.G.7
  • 16
    • 0028341658 scopus 로고
    • Delineation of discrete domains for substrate, cocaine, and tricyclic antidepressant interactions using chimeric dopamine-norepinephrine transporters
    • GIROS, B., WANG, Y. M., SUTER, S., MCLESKEY, S. B., PIFL, C. AND CARON, M. G.: Delineation of discrete domains for substrate, cocaine, and tricyclic antidepressant interactions using chimeric dopamine-norepinephrine transporters. J. Biol. Chem. 269: 15985-15988, 1994.
    • (1994) J. Biol. Chem. , vol.269 , pp. 15985-15988
    • Giros, B.1    Wang, Y.M.2    Suter, S.3    Mcleskey, S.B.4    Pifl, C.5    Caron, M.G.6
  • 17
    • 0028229855 scopus 로고
    • Stable expression of biogenic amine transporters reveals differences in inhibitor sensitivity, kinetics, and ion dependence
    • Gu, H., WALL, S. C. AND RUDNICK, G.: Stable expression of biogenic amine transporters reveals differences in inhibitor sensitivity, kinetics, and ion dependence. J. Biol. Chem. 269: 7124-7130, 1994.
    • (1994) J. Biol. Chem. , vol.269 , pp. 7124-7130
    • Gu, H.1    Wall, S.C.2    Rudnick, G.3
  • 18
    • 0021287012 scopus 로고
    • 3H]Mazindol binding associated with neuronal dopamine and norepinephrine uptake sites
    • 3H]Mazindol binding associated with neuronal dopamine and norepinephrine uptake sites. Mol. Pharmacol. 26: 35-44, 1984.
    • (1984) Mol. Pharmacol. , vol.26 , pp. 35-44
    • Javitch, J.A.1    Blaustein, R.O.2    Snyder, S.H.3
  • 19
    • 0029052914 scopus 로고
    • Comparison of dopamine uptake in the basolateral amygdaloid nucleus, caudate-putamen, and nucleus accumbens of the rat
    • JONES, S. R., GARRIS, P. A., KILTS, C. D. AND WIGHTMAN, R. M.: Comparison of dopamine uptake in the basolateral amygdaloid nucleus, caudate-putamen, and nucleus accumbens of the rat. J. Neurochem. 64: 2581-2589, 1995.
    • (1995) J. Neurochem. , vol.64 , pp. 2581-2589
    • Jones, S.R.1    Garris, P.A.2    Kilts, C.D.3    Wightman, R.M.4
  • 20
    • 0026722234 scopus 로고
    • Dopamine transporter site-directed mutations differentially alter substrate transport and cocaine binding
    • KITAYAMA, S., SHIMADA, S., XU, H., MARKHAM, L., DONOVAN, D. M. AND UHL, G. R.: Dopamine transporter site-directed mutations differentially alter substrate transport and cocaine binding. Proc. Natl. Acad. Sci. USA 89: 7782-7785, 1992.
    • (1992) Proc. Natl. Acad. Sci. USA , vol.89 , pp. 7782-7785
    • Kitayama, S.1    Shimada, S.2    Xu, H.3    Markham, L.4    Donovan, D.M.5    Uhl, G.R.6
  • 21
    • 0025362328 scopus 로고
    • Kinetics and block of dopamine uptake in synaptosomes from rat caudate nucleus
    • KRUEGER, B. K.: Kinetics and block of dopamine uptake in synaptosomes from rat caudate nucleus. J. Neurochem. 55: 260-267, 1990.
    • (1990) J. Neurochem. , vol.55 , pp. 260-267
    • Krueger, B.K.1
  • 23
    • 0023772218 scopus 로고
    • Differentiation of dopamine overflow and uptake processes in the extracellular fluid of the rat caudate nucleus with fast-scan in vivo voltammetry
    • MAY, L. J., KUHR, W. G. AND WIGHTMAN, R. M.: Differentiation of dopamine overflow and uptake processes in the extracellular fluid of the rat caudate nucleus with fast-scan in vivo voltammetry. J. Neurochem. 51: 1060-1069, 1988.
    • (1988) J. Neurochem. , vol.51 , pp. 1060-1069
    • May, L.J.1    Kuhr, W.G.2    Wightman, R.M.3
  • 24
    • 0026770299 scopus 로고
    • A multisubstrate mechanism of striatal dopamine uptake and its inhibition by cocaine
    • MCELVAIN, J. S. AND SCHENK, J. O.: A multisubstrate mechanism of striatal dopamine uptake and its inhibition by cocaine. Biochem. Pharmacol. 43: 2189-2199, 1992.
    • (1992) Biochem. Pharmacol. , vol.43 , pp. 2189-2199
    • Mcelvain, J.S.1    Schenk, J.O.2
  • 25
    • 0028072749 scopus 로고
    • Kinetic evaluation of the commonality between the site(s) of action of cocaine and some other structurally similar and dissimilar inhibitors of the striatal transporter for dopamine
    • MEIERGERD, S. M. AND SCHENK, J. O.: Kinetic evaluation of the commonality between the site(s) of action of cocaine and some other structurally similar and dissimilar inhibitors of the striatal transporter for dopamine. J. Neurochem. 63: 1683-1692, 1994.
    • (1994) J. Neurochem. , vol.63 , pp. 1683-1692
    • Meiergerd, S.M.1    Schenk, J.O.2
  • 26
    • 0027454020 scopus 로고
    • Dopamine transporter expression confers cytotoxicity to low doses of the parkinsonism-inducing neurotoxin 1-methyl-4-phenylpyridinium
    • PIFL, C., GIROS, B. AND CARON, M. G.: Dopamine transporter expression confers cytotoxicity to low doses of the parkinsonism-inducing neurotoxin 1-methyl-4-phenylpyridinium. J. Neurosci. 13: 4246-4253, 1993.
    • (1993) J. Neurosci. , vol.13 , pp. 4246-4253
    • Pifl, C.1    Giros, B.2    Caron, M.G.3
  • 28
    • 0027158841 scopus 로고
    • 3H]tropane to the dopamine uptake carrier
    • 3H]tropane to the dopamine uptake carrier. J. Neurochem. 61: 167-177, 1993.
    • (1993) J. Neurochem. , vol.61 , pp. 167-177
    • Reith, M.E.A.1    Coffey, L.L.2
  • 29
    • 0026469609 scopus 로고
    • Evidence for mutually exclusive binding of cocaine, BTCP, GBR 12935, and dopamine to the dopamine transporter
    • REITH, M. E. A., DE COSTA, B., RICE, K. C. AND JACOBSON, A. E.: Evidence for mutually exclusive binding of cocaine, BTCP, GBR 12935, and dopamine to the dopamine transporter. Eur. J. Pharmacol. 227: 417-425, 1992.
    • (1992) Eur. J. Pharmacol. , vol.227 , pp. 417-425
    • Reith, M.E.A.1    De Costa, B.2    Rice, K.C.3    Jacobson, A.E.4
  • 30
    • 0022481325 scopus 로고
    • Structural requirements for cocaine congeners to interact with dopamine and serotonin uptake sites in mouse brain and to induce stereotyped behavior
    • REITH, M. E. A., MEISLER, B. E., SERSHEN, H. AND LAJTHA, A.: Structural requirements for cocaine congeners to interact with dopamine and serotonin uptake sites in mouse brain and to induce stereotyped behavior. Biochem. Pharmacol. 35: 1123-1129, 1986.
    • (1986) Biochem. Pharmacol. , vol.35 , pp. 1123-1129
    • Reith, M.E.A.1    Meisler, B.E.2    Sershen, H.3    Lajtha, A.4
  • 31
    • 0026568962 scopus 로고
    • Radiolabeling of dopamine uptake sites in mouse striatum: Comparison of binding sites for cocaine, mazindol, and GBR 12935
    • REITH, M. E. A. AND SELMECI, G.: Radiolabeling of dopamine uptake sites in mouse striatum: comparison of binding sites for cocaine, mazindol, and GBR 12935. Naunyn Schmiedebergs Arch. Pharmacol. 345: 309-318, 1992.
    • (1992) Naunyn Schmiedebergs Arch. Pharmacol. , vol.345 , pp. 309-318
    • Reith, M.E.A.1    Selmeci, G.2
  • 33
    • 0021149396 scopus 로고
    • Blockade by antidepressants and related compounds of biogenic amine uptake into rat brain synaptosomes: Most antidepressants selectively block norepinephrine uptake
    • RICHELSON, E. AND PFENNING, M.: Blockade by antidepressants and related compounds of biogenic amine uptake into rat brain synaptosomes: Most antidepressants selectively block norepinephrine uptake. Eur. J. Pharmacol. 104: 277-286, 1984.
    • (1984) Eur. J. Pharmacol. , vol.104 , pp. 277-286
    • Richelson, E.1    Pfenning, M.2
  • 34
    • 0023265754 scopus 로고
    • Cocaine receptors on dopamine transporters are related to self-administration of cocaine
    • RITZ, M. C., LAMB, R. J., GOLDBERG, S. R. AND KUHAR, M. J.: Cocaine receptors on dopamine transporters are related to self-administration of cocaine. Science 237: 1219-1223, 1987.
    • (1987) Science , vol.237 , pp. 1219-1223
    • Ritz, M.C.1    Lamb, R.J.2    Goldberg, S.R.3    Kuhar, M.J.4
  • 38
    • 0023769440 scopus 로고
    • Apparent competitive inhibition of radioligand binding to receptors: Experimental and theoretical considerations in the analysis of equilibrium binding data
    • TOMLINSON, G. AND HNATOWICH, M. R.: Apparent competitive inhibition of radioligand binding to receptors: experimental and theoretical considerations in the analysis of equilibrium binding data. J. Recept. Res. 8: 809-830, 1988.
    • (1988) J. Recept. Res. , vol.8 , pp. 809-830
    • Tomlinson, G.1    Hnatowich, M.R.2
  • 40
    • 0026473061 scopus 로고
    • Determination of radioligand specific activity using competition binding assays
    • WIENER, H. L. AND REITH, M. E. A.: Determination of radioligand specific activity using competition binding assays. Anal. Biochem. 207: 58-62, 1992.
    • (1992) Anal. Biochem. , vol.207 , pp. 58-62
    • Wiener, H.L.1    Reith, M.E.A.2
  • 41
    • 0021646463 scopus 로고
    • Neural mechanism of the reinforcing action of cocaine
    • ed. by J. Grabowski, NIDA Research Monograph 50, U.S. Government Printing Office, Washington, D.C. 20402
    • WISE, R. W.: Neural mechanism of the reinforcing action of cocaine. In Cocaine: Pharmacology, Effects and Treatment of Abuse, ed. by J. Grabowski, p. 15. NIDA Research Monograph 50, U.S. Government Printing Office, Washington, D.C. 20402, 1984.
    • (1984) Cocaine: Pharmacology, Effects and Treatment of Abuse , pp. 15
    • Wise, R.W.1
  • 42
    • 0030611085 scopus 로고    scopus 로고
    • 3H] Win 35,428 Binding to the human dopamine transporter in a similar fashion
    • in press
    • 3H] WIN 35,428 Binding to the human dopamine transporter in a similar fashion. J. Neurochemistry, in press, 1997.
    • (1997) J. Neurochemistry
    • Wu, Q.1    Coffey, L.L.2    Reith, M.E.A.3
  • 43
    • 0028797473 scopus 로고
    • Translocation of dopamine and binding of 2β-carbomethoxy-3β-(4-fluorophenyl)tropane (Win 35,428) measured under identical conditions in rat striatal synaptosomal preparations. Inhibition by various blockers
    • XU, C., COFFEY, L. L. AND REITH, M. E. A.: Translocation of dopamine and binding of 2β-carbomethoxy-3β-(4-fluorophenyl)tropane (WIN 35,428) measured under identical conditions in rat striatal synaptosomal preparations. Inhibition by various blockers. Biochem. Pharmacol. 49: 339-350, 1995.
    • (1995) Biochem. Pharmacol. , vol.49 , pp. 339-350
    • Xu, C.1    Coffey, L.L.2    Reith, M.E.A.3
  • 45
    • 0030426646 scopus 로고    scopus 로고
    • Modeling of the pH dependence of the binding of WIN 35,428 to the dopamine transporter in rat striatal membranes: Is the bioactive form positively charged or neutral?
    • XU, C. AND REITH, M. E. A.: Modeling of the pH dependence of the binding of WIN 35,428 to the dopamine transporter in rat striatal membranes: Is the bioactive form positively charged or neutral? J. Pharmacol. Exp. Ther. 278: 1340-1348, 1996.
    • (1996) J. Pharmacol. Exp. Ther. , vol.278 , pp. 1340-1348
    • Xu, C.1    Reith, M.E.A.2


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