An efficient and convenient synthesis of formamidines

Tetrahedron Letters

Volumn 38, Issue 31, 1997, Pages 5423-5426

  Han, Ying ^a   Cai, Lisheng ^a  

^a UNIVERSITY OF ILLINOIS AT CHICAGO   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMINE; FORMAMIDINE; N,N DIMETHYLFORMAMIDE; REAGENT;

ARTICLE; DRUG SYNTHESIS; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; REACTION ANALYSIS;

EID: 0030836335     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(97)01206-9     Document Type: Article

References (34)

1. (a) Meyers, A. I.; Hutchings, R. Heterocycles 1996, 42, 475-8.
2. (b) Meyers, A. I.; Gonzalez, M. A.; Struzka, V.; Akahane, A.; Guiles, J.; Warmus, J. S. Tetrahedron Letters 1991, 32, 5501-4.
3. (c) Meyers, A. I.; Hutchings, R. H. Tetrahedron 1993, 49, 1807-20.
4. (d) Meyers, A. I.; Elworthy, T. R. J. Org.Chem. 1992, 57, 4732-40.
5. (e) Meyers, A. I. Tetrahedron 1992, 48, 2589-612.
6. (f) Partridge, M. W.; Smith, A. J. C. S. Perkin 1, 1973, 453-6.
7. (a) Leauza, W. J.; Wildouger, K. J.; Miller, T. W.; Christensen, B. G. J. Med. Chem. 1979, 22, 435.
8. (b) Scott, M. K.; Jacoby, H. J.; Mills, J. E.; Bonfilio, A. C.; Rasmussen, C. R. J. Med. Chem. 1983, 26, 535.
9. (c) Donetti, A.; Cereda, E.; Bellora, E.; Gallazzi, A.; Bazzano, C.; Vanoni, P. C.; Del Soldato, P.; Micheletti, R.; Pagani, F.; Giachetti, A. J. Med. Chem. 1984,27, 380.
10. (d) Beeman, R. W.; Matsumura, F. Nature 1973, 242, 273.
11. (e) Aziz, S. A.; Knowles, C. O. Nature 1973, 242, 417.
12. (f) Gätzi, K.; Fisher, H. Swiss Patent 563 109; C. A. 1975, 83, 189327.
13. (a) Bottomley, W.; Boyd, G. V. J. C. S. Chem. Comm. 1980, 790.
14. (b) Bésán, J.; Kulcsár, L.; Kovács, M. Synthesis 1980, 883-4.
15. (c) Pedersen, E. B. Synthesis 1979, 546-7.
16. (d) Hill, A. J.; Johnson, J. V. J. Am. Chem. Soc. 1954, 76, 920.
17. (e) Mandel, G.; Hill, A. J. J. Am. Chem. Soc. 1954, 76, 3978.
18. (f) Bredereck, H.; Gomper, R.; Klen, H.; Kempfer, M. Chem. Ber. 1959, 92, 837.
19. Cereda, E.; Bellora, E.; Donetti, A. Synthesis 1986, 288-91.
20. (a) De Wolfe, R. H. J. Org. Chem. 1962, 27, 490.
21. (b) Roberts, R. M. J. Org. Chem. 1949, 14, 297.
22. (c) Bradley, W.; Wright, I. J. Chem. Soc. 1956, 640.
23. (d) Taylor, E. C.; Ehrhart, W. A. J. Org. Chem. 1965, 28, 1108.
24. (e) Zupan, M.; Pirc, V.; Pollak, A.; Stanovnik, B.; Tisler, M. J. Heterocycl. Chem. 1974, 525-8.
25. (f) Osek, J.; Oszczapowicz, J.; Drzewinski, W. J. Chem. Soc. Perkin Trans. II 1986, 1961-4.
26. Weiner, M. L. J. Org. Chem. 1960, 2245-6.
27. Ulrich, H.; Tucker, B.; Stuber, F. A.; Sayigh, A. A. R. J. Org. Chem. 1968, 33, 3928-30.
28. Shevchenko, I. V.; Furmanova, M. V.; Kukhar, V. P.; Kolodyazhnyi, O. I. J. Gen. Chem. USSR (Engl. Transl.) 1988, 1289-90.
29. (a) Larizza, A.; Brancaccio, G.; Lettieri, G. J. Org. Chem. 1964, 3697-700.
30. (b) Scott, M.; Rasmussen, C. U. K. Patent 1979, 2017689.
31. (c) McNeil, B. Inc. C. A. 1980, 92, 110826.
32. (d) Kikugawa, Y.; Yamada, S. Tetrahedron Lett. 1969, 699.
33. Hegarty, A. F.; Chandler, A. Tetrahedron Lett. 1980, 21, 885-8.
34. Corey, E. J.; Posner, G. H.; Atkinson, R. F.; Wingard, A. K.; Hallora, D. J.; Radzik, D. M.; Nash, J. J. J. Org. Chem. 1989, 54, 389-93.