Discovery and development of non-peptide antagonists of peptide hormone receptors

Biochemical Society Transactions

Volumn 25, Issue 3, 1997, Pages 1051-1057

  Pettibone, D J ^a   Freidinger, R M ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1 (2,3 DIHYDRO 1 METHYL 2 OXO 5 PHENYL 1H 1,4 BENZODIAZEPIN 3 YL) 3 (3 METHYLPHENYL)UREA; 1 [1 [4 (3 ACETAMIDOPROPOXY)BENZOYL] 4 PIPERIDYL] 1,2,3,4 TETRAHYDRO 2 QUINOLINONE; ANTIHYPERTENSIVE AGENT; ARGIPRESSIN RECEPTOR; ASPERLICIN; BOSENTAN; CHOLECYSTOKININ RECEPTOR BLOCKING AGENT; DEVAZEPIDE; ENDOTHELIN RECEPTOR ANTAGONIST; GUANINE NUCLEOTIDE BINDING PROTEIN; HORMONE ANTAGONIST; HORMONE RECEPTOR; HORMONE RECEPTOR STIMULATING AGENT; LOSARTAN POTASSIUM; MOZAVAPTAN; N [[4' [(2 ETHYL 5,7 DIMETHYL 3H IMIDAZO[4,5 B]PYRIDIN 3 YL)METHYL] 2 BIPHENYLYL]SULFONYL]BENZAMIDE; NEUROKININ 1 RECEPTOR ANTAGONIST; OXYTOCIN ANTAGONIST; PEPTIDE HORMONE ANTAGONIST; RELCOVAPTAN; SUBSTANCE P ANTAGONIST;

ANIMAL EXPERIMENT; ANIMAL MODEL; CLINICAL TRIAL; CONFERENCE PAPER; CONGESTIVE HEART FAILURE; CONTROLLED CLINICAL TRIAL; CONTROLLED STUDY; DRUG IDENTIFICATION; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG RESEARCH; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; GASTROINTESTINAL SYMPTOM; HUMAN; HYPERTENSION; INTRADUODENAL DRUG ADMINISTRATION; INTRAVENOUS DRUG ADMINISTRATION; MOLECULAR MODEL; NONHUMAN; ORAL DRUG ADMINISTRATION; PREMATURE LABOR; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

ANIMALIA;

EID: 0030822663     PISSN: 03005127     EISSN: None     Source Type: Journal    
DOI: 10.1042/bst0251051     Document Type: Conference Paper

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