메뉴 건너뛰기




Volumn 331, Issue 2-3, 1997, Pages 285-293

Properties of a new radioiodinated antagonist for human vasopressin V2 and V(1a) receptors

Author keywords

Autoradiography; Vasopressin receptor antagonist, iodinated; Vasopressin V2 receptor, human

Indexed keywords

1 (BETA MERCAPTO BETA,BETA PENTAMETHYLENEPROPIONIC ACID) 2 O ETHYL TYROSINE 4 VALINE 9 TYROSYLAMIDE; OXYTOCIN RECEPTOR; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG; VASOPRESSIN ANTAGONIST; VASOPRESSIN V1 RECEPTOR; VASOPRESSIN V2 RECEPTOR;

EID: 0030814154     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(97)01021-2     Document Type: Article
Times cited : (18)

References (39)
  • 3
    • 0020465411 scopus 로고
    • Lithium amplifies agonist-dependent phosphatidylinositol responses in brain and salivary glands
    • Berridge, M.J., Downes, C.P., Hanley, M.R., 1982. Lithium amplifies agonist-dependent phosphatidylinositol responses in brain and salivary glands. Biochem. J. 206, 587.
    • (1982) Biochem. J. , vol.206 , pp. 587
    • Berridge, M.J.1    Downes, C.P.2    Hanley, M.R.3
  • 5
    • 0015694586 scopus 로고
    • 3H]lysine vasopressin to pig kidney plasma membranes. Relationship of receptor occupancy to adenylate cyclase activation
    • 3H]lysine vasopressin to pig kidney plasma membranes. Relationship of receptor occupancy to adenylate cyclase activation. J. Biol. Chem. 248, 5922.
    • (1973) J. Biol. Chem. , vol.248 , pp. 5922
    • Bockaert, J.1    Roy, C.2    Rajerison, R.3    Jard, S.4
  • 6
    • 0003359140 scopus 로고
    • Active esters and resins in peptide synthesis
    • Bodanszky, M., Sheehan, J.T., 1964. Active esters and resins in peptide synthesis, Chem. Ind., 1423.
    • (1964) Chem. Ind. , pp. 1423
    • Bodanszky, M.1    Sheehan, J.T.2
  • 8
    • 0001641316 scopus 로고
    • The quantitative assay of vasopressin
    • Dekanski, J., 1952. The quantitative assay of vasopressin. Br. J. Pharmacol. 7, 567.
    • (1952) Br. J. Pharmacol. , vol.7 , pp. 567
    • Dekanski, J.1
  • 10
    • 0020406390 scopus 로고
    • Kinetic and pharmacological characterisation of vasopressin membrane receptors from human kidney medulla: Relation to adenylate cyclase activation
    • Guillon, G., Butlen, D., Cantau, B., Barth, T., Jard, S., 1982. Kinetic and pharmacological characterisation of vasopressin membrane receptors from human kidney medulla: Relation to adenylate cyclase activation. Eur. J. Pharmacol. 85, 291.
    • (1982) Eur. J. Pharmacol. , vol.85 , pp. 291
    • Guillon, G.1    Butlen, D.2    Cantau, B.3    Barth, T.4    Jard, S.5
  • 11
    • 0029786715 scopus 로고    scopus 로고
    • A fully active nonglycosylated V2 vasopressin receptor
    • Innamorati, G., Sadeghi, H., Birnbaumer, M., 1996. A fully active nonglycosylated V2 vasopressin receptor. Mol. Pharmacol. 50, 467.
    • (1996) Mol. Pharmacol. , vol.50 , pp. 467
    • Innamorati, G.1    Sadeghi, H.2    Birnbaumer, M.3
  • 12
    • 0023521253 scopus 로고
    • Iodination of vasopressin analogues with agonistic and antagonistic properties: Effects on biological properties and affinity for vascular and renal vasopressin receptors
    • Jard, S., Lombard, C., Seyer, R., Aumelas, A., Manning, M., Sawyer, W.H., 1987. Iodination of vasopressin analogues with agonistic and antagonistic properties: Effects on biological properties and affinity for vascular and renal vasopressin receptors. Mol. Pharmacol. 32, 369.
    • (1987) Mol. Pharmacol. , vol.32 , pp. 369
    • Jard, S.1    Lombard, C.2    Seyer, R.3    Aumelas, A.4    Manning, M.5    Sawyer, W.H.6
  • 15
    • 0029117328 scopus 로고
    • A new tritiated oxytocin receptor radioligand-synthesis and application for localization of central oxytocin receptors
    • Klein, U., Jurzak, M., Gerstberger, R., Fahrenholz, F., 1995. A new tritiated oxytocin receptor radioligand-synthesis and application for localization of central oxytocin receptors. Peptides 16, 851.
    • (1995) Peptides , vol.16 , pp. 851
    • Klein, U.1    Jurzak, M.2    Gerstberger, R.3    Fahrenholz, F.4
  • 16
    • 0026740975 scopus 로고
    • Cloning and characterization of a vasopressin V2 receptor and possible link to nephrogenic diabetes insipidus
    • Lolait, S.J., O'Carroll, A.M., McBride, O.W., Konig, M., Morel, A., Brownstein, M.J., 1992. Cloning and characterization of a vasopressin V2 receptor and possible link to nephrogenic diabetes insipidus. Nature 357, 336.
    • (1992) Nature , vol.357 , pp. 336
    • Lolait, S.J.1    O'Carroll, A.M.2    McBride, O.W.3    Konig, M.4    Morel, A.5    Brownstein, M.J.6
  • 17
    • 0014432614 scopus 로고
    • Synthesis by the Merrifield method of a protected nonapeptide amide with the amino acid sequence of oxytocin
    • Manning, M., 1968. Synthesis by the Merrifield method of a protected nonapeptide amide with the amino acid sequence of oxytocin. J. Am. Chem. Soc. 90, 1348.
    • (1968) J. Am. Chem. Soc. , vol.90 , pp. 1348
    • Manning, M.1
  • 20
    • 0021271889 scopus 로고
    • Potent and selective antagonists of the antidiuretic reponses to arginine vasopressin based on modifications of [1-(β-mercapto-β,β-cyclopentamethylene propionic acid), 2-D-isoleucine, 4-valine] arginine-vasopressin at position 4
    • Manning, M., Nawrocka, E., Misicka, A., Olma, A., Klis, W.A., 1984. Potent and selective antagonists of the antidiuretic reponses to arginine vasopressin based on modifications of [1-(β-mercapto-β,β-cyclopentamethylene propionic acid), 2-D-isoleucine, 4-valine] arginine-vasopressin at position 4. J. Med. Chem. 27, 423.
    • (1984) J. Med. Chem. , vol.27 , pp. 423
    • Manning, M.1    Nawrocka, E.2    Misicka, A.3    Olma, A.4    Klis, W.A.5
  • 21
    • 0020026845 scopus 로고
    • Design of more potent antagonists of the antidiuretic response to arginine-vasopressin
    • Manning, M., Olma, A., Klis, W.A., Kolodziejczyk, A., Seto, J., Sawyer, W.H., 1982. Design of more potent antagonists of the antidiuretic response to arginine-vasopressin. J. Med. Chem. 25, 45.
    • (1982) J. Med. Chem. , vol.25 , pp. 45
    • Manning, M.1    Olma, A.2    Klis, W.A.3    Kolodziejczyk, A.4    Seto, J.5    Sawyer, W.H.6
  • 22
    • 0027532677 scopus 로고
    • Design, synthesis and some uses of receptor-specific agonists and antagonists of vasopressin and oxytocin
    • Manning, M., Sawyer, W.H., 1993. Design, synthesis and some uses of receptor-specific agonists and antagonists of vasopressin and oxytocin. J. Recept. Res. 13, 195.
    • (1993) J. Recept. Res. , vol.13 , pp. 195
    • Manning, M.1    Sawyer, W.H.2
  • 24
    • 0001611730 scopus 로고
    • Solid phase peptide synthesis. III. An improved synthesis of bradykinin
    • Merrifield, R.B., 1964. Solid phase peptide synthesis. III. An improved synthesis of bradykinin. Biochemistry 2, 1385.
    • (1964) Biochemistry , vol.2 , pp. 1385
    • Merrifield, R.B.1
  • 26
    • 0026604171 scopus 로고
    • Molecular cloning and expression of a rat Via arginine vasopressin receptor
    • Morel, A., O'Carroll, A.M., Brownstein, M.J., Lolait, S.J., 1992. Molecular cloning and expression of a rat Via arginine vasopressin receptor. Nature 356, 523.
    • (1992) Nature , vol.356 , pp. 523
    • Morel, A.1    O'Carroll, A.M.2    Brownstein, M.J.3    Lolait, S.J.4
  • 27
    • 72849154573 scopus 로고
    • Effect of magnesium ion on the response of the rat uterus to neurohypophysial hormones and analogues
    • Munsick, R.A., 1960. Effect of magnesium ion on the response of the rat uterus to neurohypophysial hormones and analogues. Endocrinology 66, 451.
    • (1960) Endocrinology , vol.66 , pp. 451
    • Munsick, R.A.1
  • 28
    • 0017861160 scopus 로고
    • Solid-phase synthesis of somatostatin and glucagon-selective analogs in gram quantities
    • Rivier, J., Kaiser, R., Galyean, R., 1978. Solid-phase synthesis of somatostatin and glucagon-selective analogs in gram quantities. Biopolymers 17, 1927.
    • (1978) Biopolymers , vol.17 , pp. 1927
    • Rivier, J.1    Kaiser, R.2    Galyean, R.3
  • 29
    • 0016374975 scopus 로고
    • A highly sensitive adenylate cyclase assay
    • Salomon, Y., Londos, C., Rodbell, M., 1974. A highly sensitive adenylate cyclase assay. Anal. Biochem. 58, 541.
    • (1974) Anal. Biochem. , vol.58 , pp. 541
    • Salomon, Y.1    Londos, C.2    Rodbell, M.3
  • 30
    • 0001201002 scopus 로고
    • Differences in antidiuretic responses of rats to the intravenous administration of lysine and arginine vasopressins
    • Sawyer, W.H., 1958. Differences in antidiuretic responses of rats to the intravenous administration of lysine and arginine vasopressins. Endocrinology 63, 694.
    • (1958) Endocrinology , vol.63 , pp. 694
    • Sawyer, W.H.1
  • 31
    • 84982328496 scopus 로고
    • p A, a new scale of the measurement of drug antagonism
    • Schild, H.O., 1947. p A, a new scale of the measurement of drug antagonism. Br. J. Pharmacol. 2, 189.
    • (1947) Br. J. Pharmacol. , vol.2 , pp. 189
    • Schild, H.O.1
  • 36
    • 0027959744 scopus 로고
    • Molecular cloning and functional expression of a cDNA encoding the human V1b vasopressin receptor
    • Sugimoto, T., Saito, M., Mochizuchi, S., Watanabe, Y., Hashimoto, S., Kawashima, H., 1994. Molecular cloning and functional expression of a cDNA encoding the human V1b vasopressin receptor. J. Biol. Chem. 269, 27088.
    • (1994) J. Biol. Chem. , vol.269 , pp. 27088
    • Sugimoto, T.1    Saito, M.2    Mochizuchi, S.3    Watanabe, Y.4    Hashimoto, S.5    Kawashima, H.6
  • 37
    • 0028017952 scopus 로고
    • Molecular cloning, sequencing and functional expression of a cDNA encoding the human Via vasopressin receptor
    • Thibonnier, M., Auzan, C., Madhun, Z., Wilkins, P., Berti-Mattera, L., Clauser, E., 1994. Molecular cloning, sequencing and functional expression of a cDNA encoding the human Via vasopressin receptor. J. Biol. Chem. 269, 3304.
    • (1994) J. Biol. Chem. , vol.269 , pp. 3304
    • Thibonnier, M.1    Auzan, C.2    Madhun, Z.3    Wilkins, P.4    Berti-Mattera, L.5    Clauser, E.6
  • 38
    • 0023912848 scopus 로고
    • Autoradiographic localization of vasopressin and oxytocin binding sites in rat kidney
    • Tribollet, E., Barberis, C., Dreifuss, J.J., Jard, S., 1988. Autoradiographic localization of vasopressin and oxytocin binding sites in rat kidney. Kidney Int. 33, 959.
    • (1988) Kidney Int. , vol.33 , pp. 959
    • Tribollet, E.1    Barberis, C.2    Dreifuss, J.J.3    Jard, S.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.