Peptidic prodrugs of novel aminomethyl-THF 1β-methylcarbapenems

Bioorganic and Medicinal Chemistry Letters

Volumn 7, Issue 13, 1997, Pages 1665-1670

  Lin, Yang I ^a   Bitha, Panayota ^a   Sakya, Subas M ^a   Li, Zhong ^a   Lang Jr , Stanley A ^a   Yang, Youjun ^a   Bhachech, Niraja ^a   Weiss, William J ^a   Petersen, Peter J ^a   Jacobus, Nilda V ^a   Bush, Karen ^a   Testa, Raymond T ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ALANINE DERIVATIVE; AMINO ACID DERIVATIVE; CARBAPENEM DERIVATIVE; CILASTATIN PLUS IMIPENEM; DIPEPTIDE; GLYCINE DERIVATIVE; PEPTIDASE; PEPTIDE DERIVATIVE; PHENYLALANINE DERIVATIVE; PRODRUG; TETRAHYDROFURAN DERIVATIVE; TRIPEPTIDE; VALINE;

ACTIVE TRANSPORT; ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIMICROBIAL ACTIVITY; ARTICLE; BACTERIAL INFECTION; CONTROLLED STUDY; DRUG HYDROLYSIS; DRUG SYNTHESIS; DRUG TRANSPORT; ESCHERICHIA COLI; MOUSE; NONHUMAN; ORAL DRUG ADMINISTRATION; PARTITION COEFFICIENT; STAPHYLOCOCCUS AUREUS; SUBCUTANEOUS DRUG ADMINISTRATION;

EID: 0030812297     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(97)00281-3     Document Type: Article

References (11)

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2. (b) Lin, Y.-I; Bitha, P.; Sakya, S. M.; Strohmeyer, T. W.; Feigelson, G. B.; Ziegler, C. B., Jr.; Lee, V. J.; Tally, F. P. 34th Interscience Conference on Antimicrobial Agents and Chemotherapy. Orlando 1994. Abstract F70.
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