112. Novel heterospirocyclic 3-amino-2H-azirines as synthons for heterocyclic α-amino acids)

Helvetica Chimica Acta

Volumn 80, Issue 5, 1997, Pages 1528-1554

  Strässler, Christoph ^a   Linden, Anthony ^a   Heimgartner, Heinz ^a  

^a UNIVERSITY OF ZURICH   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

AZIRINE DERIVATIVE;

AMINO ACID SUBSTITUTION; ARTICLE; COUPLING FACTOR; DRUG SYNTHESIS; NONHUMAN; PEPTIDE SYNTHESIS; PROTEIN SECONDARY STRUCTURE; PROTON NUCLEAR MAGNETIC RESONANCE; X RAY CRYSTALLOGRAPHY;

EID: 0030806311     PISSN: 0018019X     EISSN: None     Source Type: Journal    
DOI: 10.1002/hlca.19970800515     Document Type: Article

References (20)

1. E. Benedetti, C. Toniolo, in 'Polymeric Materials', Ed. J. C. Salamone, CRC Press, New York, 1996, Vol. 8, p. 6472;
2. C. Toniolo, E. Benedetti, Macromoleculcs 1991, 24, 4004.
3. C. Toniolo, M. Crisma, F. Formaggio, G. Valle, G. Cavicchioni, G. Précigoux, A. Aubry, J. Kamphuis, Biopolymers 1993, 33, 1061.
4. C. Toniolo, M. Crisma, G. Valle, G. M. Bonora, S. Polinelli, E. L. Becker, R. J. Freer, R. Sudhanand, R. Balaji Rao, P. Balaram, M. Sukumar, Pept. Res. 1989, 2, 275.
5. a) P. Wipf, H. Heimgartner, Helv Chim. Acta 1988, 71, 258;
6. b) P. Wipf, R. W. Kunz, H. Heimgartner, ibid. 1988, 71, 268.
7. M. Sahebi, P. Wipf, H. Heimgartner, Tetrahedron 1989, 45, 2999.
8. H. Heimgartner, Angew. Chem. Int. Ed. 1991, 30, 238.
9. A. W. Coulter, J. B. Lombardini, J. R. Sufrin, P. Talalay, Mol. Pharm. 1974, 10, 319.
10. N. J. Lewis, R. L. Inloes, J. Hes, R. H. Matthews, G. Milo, J. Med. Chem. 1978, 21, 1070.
11. M. Sukumar, P. A. Raj, P. Balaram, E. L. Becker, Biochem. Biophys. Res. Commun. 1985, 128, 339.
12. C. A. Fink, Y. Qiao, C. J. Berry, Y. Sakane, R. D. Ghai, A. J. Trapani, J. Med. Chem. 1995, 38, 5023.
13. P. Wipf, H. Heimgartner, Helv. Chim. Acta 1990, 73, 13.
14. J. M. Villalgordo, H. Heimgartner, Tetrahedron 1993, 49, 7215.
15. W. Altherr, Dissertation, Universität Zürich, 1994
16. ; W. Altherr, H. Heimgartner, in 'Peptides 1990', Eds. E. Giralt and D. Andreu, Escom, Leiden, 1991, p. 107;
17. in 'Peptides 1992', Eds. C. H. Schneider and A. N. Eberle, Escom, Leiden, 1993, p. 387.
18. C. B. Bucher, A. Linden, H. Heimgartner, Helv. Chim. Acta 1995, 78, 935.
19. R. Luykx, C. B. Bucher, A. Linden, H. Heimgartner, Helv. Chim. Acta 1996, 79, 527;
20. C. B. Bucher, H. Heimgartner, ibid. 1996, 79, 1903.