Stereochemical influence on the stability of radio-metal complexes in vivo. Synthesis and evaluation of the four stereoisomers of 2-(p- nitrobenzyl)-trans-CyDTPA

Bioorganic and Medicinal Chemistry

Volumn 5, Issue 10, 1997, Pages 1925-1934

  Wu, C ^b   Kobayashi, H ^b   Sun, B ^b   Yoo, T M ^b   Paik, C H ^b   Gansow, O A ^b   Carrasquillo, J A ^b   Pastan, I ^a   Brechbiel, M W ^a  

^a NATIONAL CANCER INSTITUTE   (United States)

^b NCI ^*

Author keywords

[No Author keywords available]

Indexed keywords

CYCLOHEXANE; PENTETIC ACID; YTTRIUM;

ARTICLE; BINDING AFFINITY; DRUG SYNTHESIS; ISOTOPE LABELING; METAL BINDING; MOLECULAR STABILITY; STEREOISOMERISM; STRUCTURE ACTIVITY RELATION;

ANIMALS; CHELATING AGENTS; DRUG STABILITY; HUMANS; ISOTHIOCYANATES; LIGANDS; MICE; PENTETIC ACID; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; TISSUE DISTRIBUTION; YTTRIUM;

EID: 0030785406     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(97)00130-2     Document Type: Article

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