D-Stereospecificity in the inhibition of thermolysin by N-acyl-N-hydroxy-α-amino acid esters

Tetrahedron Asymmetry

Volumn 8, Issue 22, 1997, Pages 3699-3702

  Jin, Yonghao ^a   Kim, Dong H ^a  

^a Pohang University of Science and Technology (POSTECH)   (South Korea)

Author keywords

[No Author keywords available]

Indexed keywords

AMINO ACID DERIVATIVE; HYDROXAMIC ACID DERIVATIVE; THERMOLYSIN;

ARTICLE; CHIRALITY; DRUG DESIGN; DRUG SYNTHESIS; ENZYME INHIBITION; IN VITRO STUDY; PRIORITY JOURNAL; STEREOSPECIFICITY; STRUCTURE ACTIVITY RELATION;

EID: 0030782502     PISSN: 09574166     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0957-4166(97)00535-1     Document Type: Article

References (9)

1. Kurzak, B.; Kozolowski, H.; Farkas, E. Coord. Chem. Rev. 1992, 114, 169-200.
2. Powers, J. C.; Harper, J. W. In Proteinase Inhibitors, Barrett, A. J.; Salvesen, G. Eds.; Elsevier; Amsterdam, 1986; pp. 244-253.
3. Matthews, B. W. Acc. Chem. Res. 1988, 21, 333-340.
4. Grundke, G.; Keese, W.; Rimpler, M. Synthesis 1987, 1115-1116.
5. 23 =+49.0 (c= 1.0, MeOH).
6. Ando, N.; Tsumaki, H. Synth. Commun. 1983, 13, 1053-1056.
7. Feder, J. Biochem. Biophys. Res. Commun. 1968, 32, 326-332.
8. Holmes, M. A.; Matthews, B. W. Biochemistry 1981, 20, 6912-6920.
9. Holmes, M. A.; Tronrud, D. E.; Matthews, B. W. Biochemistry 1983, 22, 236-240.