Short synthesis of (3S,6S,9S)-2-oxo-3-(N-Boc-amino)-1-azabicyclo[4.3.0]nonane-9-carboxylic acid methyl ester: Tandem cyclization protocol

Tetrahedron Letters

Volumn 38, Issue 37, 1997, Pages 6483-6484

  Kim, Hwa Ok ^a   Kahn, Michael ^a,b  

^a Molecumetics Ltd   (United States)

^b UNIVERSITY OF WASHINGTON   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CARBOXYLIC ACID DERIVATIVE; GLUTAMIC ACID;

ARTICLE; CYCLIZATION; STEREOSPECIFICITY; SYNTHESIS;

EID: 0030767555     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(97)01492-5     Document Type: Article

References (9)

1. a) Peptide Secondary Structure Mimetics. Tetrahedron Symposia-in-print no. 50, Kahn, M. Ed., 1993, 49, 3444.
2. b) Kahn, M. Synlett. 1993, 821.
3. a) Lombart, H.-G.; Lubell, W. J. Org. Chem. 1994, 59, 6147 and references cited therein.
4. b) Li, W.; Hanau, C. E.; d'Avignon, A.; Moeller, K. D. J. Org. Chem. 1995, 60, 8155.
5. c) Kim, H. -O.; Lum, C.; Lee, M. S. Terahedron Lett. in print.
6. Olsen, R. K.; Ramasamy, K. J. Org. Chem. 1985, 50, 2264.
7. a) Kim, H. -O.; Olsen, R. K.; Choi, O. -S. J. Org. Chem. 1987, 52, 4531.
8. b) Harris, B. D.; Bhat, K. L.; Joullie, M. M. Tetrahedron Lett. 1987, 25, 2837.
9. +). All spectral data were in good agreement with literature; ref. 2a.