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Volumn 19, Issue 4, 1997, Pages 245-251

Effects of NIK-247 on cholinesterase and scopolamine-induced amnesia

Author keywords

Acetylcholinesterase; E 2020; NIK 247; Passive avoidance task; Scopolamine; Tacrine

Indexed keywords

AMIRIDINE; CHOLINESTERASE; CHOLINESTERASE INHIBITOR; DONEPEZIL; SCOPOLAMINE; TACRINE;

EID: 0030748352     PISSN: 03790355     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (12)

References (28)
  • 1
    • 0018675642 scopus 로고
    • Neurotransmitter-related enzymes in senile dementia of the Alzheimer type
    • Davies, P. Neurotransmitter-related enzymes in senile dementia of the Alzheimer type. Brain Res 1979, 171: 319-27.
    • (1979) Brain Res , vol.171 , pp. 319-327
    • Davies, P.1
  • 2
    • 0020072221 scopus 로고
    • Alzheimer's disease and senile dementia: Loss of neurons in the basal forebrain
    • Whitehouse, P.J., Price, D.L., Struble, R.G. et al. Alzheimer's disease and senile dementia: Loss of neurons in the basal forebrain. Science 1982, 215: 1237-9.
    • (1982) Science , vol.215 , pp. 1237-1239
    • Whitehouse, P.J.1    Price, D.L.2    Struble, R.G.3
  • 3
    • 0015965912 scopus 로고
    • Human memory and the cholinergic system
    • Drachman, D. A., Leavitt, J. Human memory and the cholinergic system. Arch Neurol 1974, 30: 113-21.
    • (1974) Arch Neurol , vol.30 , pp. 113-121
    • Drachman, D.A.1    Leavitt, J.2
  • 4
    • 0028575329 scopus 로고
    • Effect of NIK-247 on basal concentrations of extracellular acetylcholine in the cerebral cortex of conscious, freely moving rats
    • Ishii, Y., Kojima, J., Ikeda, N., Kawashima, K. Effect of NIK-247 on basal concentrations of extracellular acetylcholine in the cerebral cortex of conscious, freely moving rats. Jpn J Pharmacol 1994. 66: 289-93.
    • (1994) Jpn J Pharmacol , vol.66 , pp. 289-293
    • Ishii, Y.1    Kojima, J.2    Ikeda, N.3    Kawashima, K.4
  • 5
    • 0026322494 scopus 로고
    • NIK-247 blocks voltage-dependent ionic currents in crayfish axon
    • Kojima, J., Sugawara, Y., Obara, S. NIK-247 blocks voltage-dependent ionic currents in crayfish axon. Jpn J Pharmacol 1991, 57: 545-52.
    • (1991) Jpn J Pharmacol , vol.57 , pp. 545-552
    • Kojima, J.1    Sugawara, Y.2    Obara, S.3
  • 6
    • 0012690547 scopus 로고
    • Kinetics of inhibition of cholinesterases by l,2,3,4-tetrahydro-9-aminoacridine in vitro
    • Patocka, J., Bajagar, J., Bielavsky, J., Fusek, J. Kinetics of inhibition of cholinesterases by l,2,3,4-tetrahydro-9-aminoacridine in vitro. Coll Czech Chem Commun 1976, 41: 816-24.
    • (1976) Coll Czech Chem Commun , vol.41 , pp. 816-824
    • Patocka, J.1    Bajagar, J.2    Bielavsky, J.3    Fusek, J.4
  • 7
    • 0024818025 scopus 로고
    • Correlation of brain levels of 9-amino-l,2,3,4-tetrahydroacridine (THA) with neurochemical and behavioral changes
    • Nielsen, J.A., Mena, E.E., Williams, I.H. et al. Correlation of brain levels of 9-amino-l,2,3,4-tetrahydroacridine (THA) with neurochemical and behavioral changes. Eur J Pharmacol 1989, 173: 53-64.
    • (1989) Eur J Pharmacol , vol.173 , pp. 53-64
    • Nielsen, J.A.1    Mena, E.E.2    Williams, I.H.3
  • 8
    • 0025074669 scopus 로고
    • Multiple effects of tetrahydroaminoacridine on the cholinergic system: Biochemical and behavioural aspects
    • Adem, A., Mohammed, A.K., Winblad, B. Multiple effects of tetrahydroaminoacridine on the cholinergic system: Biochemical and behavioural aspects. J Neural Transm 1990, 2: 113-28.
    • (1990) J Neural Transm , vol.2 , pp. 113-128
    • Adem, A.1    Mohammed, A.K.2    Winblad, B.3
  • 9
    • 0000557157 scopus 로고
    • E-2020 - The pharmacology of a piperidine cholinesterase inhibitor
    • Becker, R., Giacobini, E. (Eds.). Birkhaeuser: Boston
    • Rogers, S.L., Yamanishi, Y., Yamatsu, K. E-2020 - The pharmacology of a piperidine cholinesterase inhibitor. In: Cholinergic Basis for Alzheimer Therapy. Becker, R., Giacobini, E. (Eds.). Birkhaeuser: Boston 1991, 314-20.
    • (1991) Cholinergic Basis for Alzheimer Therapy , pp. 314-320
    • Rogers, S.L.1    Yamanishi, Y.2    Yamatsu, K.3
  • 10
    • 0024538288 scopus 로고
    • Effects of cholinergic drugs on learning impairment in ventral globus pallidus-lexioned rats
    • Ueki, A., Miyoshi, K. Effects of cholinergic drugs on learning impairment in ventral globus pallidus-lexioned rats. J Neurol Sci 1989,90: 1-21.
    • (1989) J Neurol Sci , vol.90 , pp. 1-21
    • Ueki, A.1    Miyoshi, K.2
  • 11
    • 0023721555 scopus 로고
    • Effects of the novel compound NIK-247 on impairment of passive avoidance response in mice
    • Nabeshima, T., Yoshida, S., Kameyama, T. Effects of the novel compound NIK-247 on impairment of passive avoidance response in mice. Eur J Pharmacol 1988, 154: 263-70.
    • (1988) Eur J Pharmacol , vol.154 , pp. 263-270
    • Nabeshima, T.1    Yoshida, S.2    Kameyama, T.3
  • 12
    • 0026600776 scopus 로고
    • Effects of NIK-247 on CO-induced impairment of passive avoidance in mice
    • Yoshida, S., Nabeshima, T., Kinbara, K., Kameyama, T. Effects of NIK-247 on CO-induced impairment of passive avoidance in mice. Eur J Pharmacol 1992, 214: 247-52.
    • (1992) Eur J Pharmacol , vol.214 , pp. 247-252
    • Yoshida, S.1    Nabeshima, T.2    Kinbara, K.3    Kameyama, T.4
  • 13
    • 0027492370 scopus 로고
    • Ameliorative effects of the centrally active cholinesterase inhibitor, NIK-247, on impairment of working memory in rats
    • Yamamoto, T., Ohno, M., Kitajima. I. et al. Ameliorative effects of the centrally active cholinesterase inhibitor, NIK-247, on impairment of working memory in rats. Physiol Behav 1993, 53: 5-10.
    • (1993) Physiol Behav , vol.53 , pp. 5-10
    • Yamamoto, T.1    Ohno, M.2    Kitajima, I.3
  • 14
    • 0027386197 scopus 로고
    • Antiamnesic and cholinomimetic side-effects of the cholinesterase inhibitors, physostigmine, tcrine and NIK-247 in rats
    • Yoshida, S., Suzuki, N. Antiamnesic and cholinomimetic side-effects of the cholinesterase inhibitors, physostigmine, tcrine and NIK-247 in rats. Eur J Pharmacol 1993, 250: 117-24.
    • (1993) Eur J Pharmacol , vol.250 , pp. 117-124
    • Yoshida, S.1    Suzuki, N.2
  • 16
    • 0023701604 scopus 로고
    • 50 values and the type of inhibition for enzyme-catalyzed reactions
    • 50 values and the type of inhibition for enzyme-catalyzed reactions. Biochem Med Metab Biol 1988, 40: 204-12.
    • (1988) Biochem Med Metab Biol , vol.40 , pp. 204-212
    • Duggleby, R.G.1
  • 17
    • 0028492689 scopus 로고
    • PD-142676 (CI-1002), a novel anticholinesterase and muscarinic antagonist
    • Emmerling, M.R., Gregor, V.E., Schwarz, R.D. et al. PD-142676 (CI-1002), a novel anticholinesterase and muscarinic antagonist. Mol Neurobiol 1994, 9: 93-106.
    • (1994) Mol Neurobiol , vol.9 , pp. 93-106
    • Emmerling, M.R.1    Gregor, V.E.2    Schwarz, R.D.3
  • 18
    • 0026504115 scopus 로고
    • Interaction of tetrahydroaminoacridine with acetylcholinesterase and butyrylcholinestenise
    • Berman, H.A., Leonard, K. Interaction of tetrahydroaminoacridine with acetylcholinesterase and butyrylcholinestenise. Mol Pharmacol 1991, 41: 412-8.
    • (1991) Mol Pharmacol , vol.41 , pp. 412-418
    • Berman, H.A.1    Leonard, K.2
  • 19
    • 0027092277 scopus 로고
    • Ambenonium is a rapidly reversible noncovalent inhibitor of acetylcholinesterase, with one of the highest known affinities
    • Hodge, A.S., Humphrey, D.R., Rosenberry, T.L. Ambenonium is a rapidly reversible noncovalent inhibitor of acetylcholinesterase, with one of the highest known affinities. Mol Pharmacol 1992, 41: 937-42.
    • (1992) Mol Pharmacol , vol.41 , pp. 937-942
    • Hodge, A.S.1    Humphrey, D.R.2    Rosenberry, T.L.3
  • 20
    • 0029127347 scopus 로고
    • Kinetic study on the inhibition of acetylcholinesterase by 1-benzyl-4-[(5,6-dimethoxy-1-indanon)-2-yl ]methylpiperidine hydrochloride (E2020)
    • Nochi, S., Asakawa, N., Sato, T. Kinetic study on the inhibition of acetylcholinesterase by 1-benzyl-4-[(5,6-dimethoxy-1-indanon)-2-yl ]methylpiperidine hydrochloride (E2020). Biol Pharm Bull 1995, 18: 1145-7.
    • (1995) Biol Pharm Bull , vol.18 , pp. 1145-1147
    • Nochi, S.1    Asakawa, N.2    Sato, T.3
  • 21
    • 0028062912 scopus 로고
    • Characterization of a novel muscarinic receptor agonist, YM796: Comparison with cholinesterase inhibitors in in vivo pharmacological studies
    • Wanibuchi, F., Nishida, T., Yamashita, H. et al. Characterization of a novel muscarinic receptor agonist, YM796: Comparison with cholinesterase inhibitors in in vivo pharmacological studies. Eur J Pharmacol 1994, 265: 151-8.
    • (1994) Eur J Pharmacol , vol.265 , pp. 151-158
    • Wanibuchi, F.1    Nishida, T.2    Yamashita, H.3
  • 22
    • 4243977170 scopus 로고    scopus 로고
    • Brain pharmacokinetics and pharmacological properties of a novel cognitive enhancer. NIK-247 (1)
    • Yano, M., Kawai, H., Ishiguro, M. et al. Brain pharmacokinetics and pharmacological properties of a novel cognitive enhancer. NIK-247 (1). Jpn J Pharmacol 1996, 71(Suppl.): 101P.
    • (1996) Jpn J Pharmacol , vol.71 , Issue.SUPPL.
    • Yano, M.1    Kawai, H.2    Ishiguro, M.3
  • 23
    • 0025030077 scopus 로고
    • High-performance liquid chromatography for the determination of tacrine and its metabolites in plasma
    • Hsu, R.S., DiLeo, E.M., Chesson, S.M. High-performance liquid chromatography for the determination of tacrine and its metabolites in plasma. J Chromatogr 1990, 530: 170-6.
    • (1990) J Chromatogr , vol.530 , pp. 170-176
    • Hsu, R.S.1    DiLeo, E.M.2    Chesson, S.M.3
  • 24
    • 0027402636 scopus 로고
    • Distribution of tacrine across the blood-brain barrier in awake, freely moving rats using in vivo microdialysis sampling
    • Telting-Diaz, M., Lunte, C.E. Distribution of tacrine across the blood-brain barrier in awake, freely moving rats using in vivo microdialysis .sampling. Pharm Res 1993, 10: 44-8.
    • (1993) Pharm Res , vol.10 , pp. 44-48
    • Telting-Diaz, M.1    Lunte, C.E.2
  • 25
    • 0024457285 scopus 로고
    • Multiple in vitro interactions with and differential in vivo regulation on muscarinic receptor subtypes by tetrahydroaminoacridine
    • Flynn, D.D., Mash, D.C. Multiple in vitro interactions with and differential in vivo regulation on muscarinic receptor subtypes by tetrahydroaminoacridine. J Pharmacol Exp Ther 1989, 250: 573-81.
    • (1989) J Pharmacol Exp Ther , vol.250 , pp. 573-581
    • Flynn, D.D.1    Mash, D.C.2
  • 26
    • 0023684301 scopus 로고
    • Tetrahydroaminoacridine selectively attenuates NMDA receptor-mediated neurotoxicity
    • Davenport. C.J., Monyer, H., Choi, D.W. Tetrahydroaminoacridine selectively attenuates NMDA receptor-mediated neurotoxicity. Eur J Pharmacol 1988, 154: 73-8.
    • (1988) Eur J Pharmacol , vol.154 , pp. 73-78
    • Davenport, C.J.1    Monyer, H.2    Choi, D.W.3
  • 27
    • 0025226511 scopus 로고
    • A comparison of the effects of cholinergic and dopaminergic agents on scopolamine-induced hyperreactivity in mice
    • Shannon, H.E., Peters, S.C. A comparison of the effects of cholinergic and dopaminergic agents on scopolamine-induced hyperreactivity in mice. J Pharmacol Exp Ther 1990, 255: 549-53.
    • (1990) J Pharmacol Exp Ther , vol.255 , pp. 549-553
    • Shannon, H.E.1    Peters, S.C.2
  • 28
    • 0025743417 scopus 로고
    • Biochemical and behavioral characterization of a novel cholinergic agonist, SR-95639
    • Boast, C.A., Leventer, S., Sabb, A. et al. Biochemical and behavioral characterization of a novel cholinergic agonist, SR-95639. Pharmacol Biochem Behav 1991, 39: 287-92.
    • (1991) Pharmacol Biochem Behav , vol.39 , pp. 287-292
    • Boast, C.A.1    Leventer, S.2    Sabb, A.3


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