Synergy between anions and farnesyldiphosphate competitive inhibitors of farnesyl:protein transferase

Journal of Biological Chemistry

Volumn 272, Issue 29, 1997, Pages 18077-18081

  Scholten, Jeffrey D ^a   Zimmerman, Karen K ^a   Oxender, Maritza G ^a   Leonard, Daniele ^a   Sebolt Leopold, Judith ^a   Gowan, Richard ^a   Hupe, Donald J ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANION; ENZYME INHIBITOR; PROTEIN FARNESYLTRANSFERASE;

ANIMAL CELL; ARTICLE; CATALYSIS; COMPETITIVE INHIBITION; CONTROLLED STUDY; ENZYME ACTIVE SITE; ENZYME INHIBITOR INTERACTION; MOLECULAR DYNAMICS; MOLECULAR INTERACTION; NONHUMAN; PRIORITY JOURNAL; REACTION ANALYSIS;

ALKYL AND ARYL TRANSFERASES; ANIMALS; ANIONS; BINDING, COMPETITIVE; CELL LINE; DRUG SYNERGISM; KINETICS; MODELS, CHEMICAL; OLIGOPEPTIDES; POLYISOPRENYL PHOSPHATES; PROTEIN ISOPRENYLATION; RECOMBINANT PROTEINS; SPODOPTERA; TRANSFECTION; TRANSFERASES;

ANIMALIA;

EID: 0030741535     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.272.29.18077     Document Type: Article

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