메뉴 건너뛰기




Volumn 24, Issue 3, 1997, Pages 269-273

Application of a novel phenylpiperazine formation reaction to the radiosynthesis of a model fluorine-18-labeled radiopharmaceutical (18FTFMPP)

Author keywords

18F Fluoride; Phenylpiperazine; Serotonin; TFMPP

Indexed keywords

3 FLUORO N (1,1,1 TRIFLUORO 3 TOLYL)PIPERAZINE F 18; PIPERAZINE DERIVATIVE; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG;

EID: 0030738287     PISSN: 09698051     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0969-8051(97)00063-2     Document Type: Article
Times cited : (11)

References (23)
  • 1
    • 0027955904 scopus 로고
    • Growth inhibition of human prostatic carcinoma cell lines by serotonin antagonist
    • Abdul M., Anezinis P. E., Logothetis C. J. and Hoosein N. M. (1994) Growth inhibition of human prostatic carcinoma cell lines by serotonin antagonist. Anticancer Res. 14, 1215-1220.
    • (1994) Anticancer Res. , vol.14 , pp. 1215-1220
    • Abdul, M.1    Anezinis, P.E.2    Logothetis, C.J.3    Hoosein, N.M.4
  • 2
    • 0022853146 scopus 로고
    • Peptide-hormone and serotonin immunoreactive cells in normal and hyperplastic prostate glands
    • Abrahamsson P. A., Wadstrom L. B., Alumets J., Falkmer S. and Grimelius L. (1986) Peptide-hormone and serotonin immunoreactive cells in normal and hyperplastic prostate glands. Pathol. Res. Pract. 181, 675-681
    • (1986) Pathol. Res. Pract. , vol.181 , pp. 675-681
    • Abrahamsson, P.A.1    Wadstrom, L.B.2    Alumets, J.3    Falkmer, S.4    Grimelius, L.5
  • 7
    • 0018890855 scopus 로고
    • Structural relationships in the inhibition of [3H]serotonin binding to rat brain membranes in vitro by 1-phenyl-piperazines
    • Fuller R. W., Mason N. R. and Molloy B. B. (1980) Structural relationships in the inhibition of [3H]serotonin binding to rat brain membranes in vitro by 1-phenyl-piperazines. Biochem. Pharmacol. 29, 833-855.
    • (1980) Biochem. Pharmacol. , vol.29 , pp. 833-855
    • Fuller, R.W.1    Mason, N.R.2    Molloy, B.B.3
  • 8
    • 0023078613 scopus 로고
    • Central serotonin receptors as target for drug research
    • S. Glennon R. A. (1987) Central serotonin receptors as target for drug research. J. Med. Chem. 30, 1-12.
    • (1987) J. Med. Chem. , vol.30 , pp. 1-12
    • Glennon, R.A.1
  • 9
    • 0025232511 scopus 로고
    • Serotonin receptors: Clinical implications
    • Glennon R. A. (1990) Serotonin receptors: Clinical implications. Neurosci. Biobehav. Rev. 14, 35-47.
    • (1990) Neurosci. Biobehav. Rev. , vol.14 , pp. 35-47
    • Glennon, R.A.1
  • 10
    • 0343736674 scopus 로고
    • Functional/clinical significance of 5-hydroxytryptamine binding sites
    • Edited by Paoletti R. Kluwer Academic Publishers, New York
    • Glennon R. A. (1990) Functional/clinical significance of 5-hydroxytryptamine binding sites. In: Serotonin: From Cell Biology to Pharmacology and Therapeutics (Edited by Paoletti R), p. 259. Kluwer Academic Publishers, New York.
    • (1990) Serotonin: From Cell Biology to Pharmacology and Therapeutics , pp. 259
    • Glennon, R.A.1
  • 11
    • 0029071971 scopus 로고
    • Substance P receptors in human primary neoplasms: Tumoural and vascular localisation
    • Hennig I. M., Laissue J. A., Horisberger U. and Reubi J. C. (1995) Substance P receptors in human primary neoplasms: Tumoural and vascular localisation. Int. J. Cancer 61, 786-792.
    • (1995) Int. J. Cancer , vol.61 , pp. 786-792
    • Hennig, I.M.1    Laissue, J.A.2    Horisberger, U.3    Reubi, J.C.4
  • 12
    • 0027189659 scopus 로고
    • Differential effects of peptide hormones bombesin, vascoactive intestinal polypeptide and somatostatin analog RC-160 on the invasive capacity of human prostatic carcinoma cells
    • Hoosein N. M., Logothetis C. J. and Chung L. W. (1993) Differential effects of peptide hormones bombesin, vascoactive intestinal polypeptide and somatostatin analog RC-160 on the invasive capacity of human prostatic carcinoma cells. J. Urol. 149, 1209-1213.
    • (1993) J. Urol. , vol.149 , pp. 1209-1213
    • Hoosein, N.M.1    Logothetis, C.J.2    Chung, L.W.3
  • 14
    • 0012409009 scopus 로고    scopus 로고
    • 3-((4-C4-chlorophenylpiperazine-1-yl)-methyl)-1H-pyrolo-2,3β- pyridine: An antagonist with high affinity and selectivity for human dopamine D4 receptor
    • Kulagowski J. J., Broughton H. B., Curtis N. R., Mawer I. M., Ridgill M. P., Baker R. and Emms F. (1996) 3-((4-C4-chlorophenylpiperazine-1-yl)-methyl)-1H-pyrolo-2,3β-pyridine: An antagonist with high affinity and selectivity for human dopamine D4 receptor. J. Med. Chem. 39, 1941-1942.
    • (1996) J. Med. Chem. , vol.39 , pp. 1941-1942
    • Kulagowski, J.J.1    Broughton, H.B.2    Curtis, N.R.3    Mawer, I.M.4    Ridgill, M.P.5    Baker, R.6    Emms, F.7
  • 17
    • 0000959883 scopus 로고
    • 18F]fluoro-for-nitro exchange: A useful intermediate in the synthesis of highly fluorinated radiopharmaceuticals
    • 18F]fluoro-for-nitro exchange: A useful intermediate in the synthesis of highly fluorinated radiopharmaceuticals. J. Label. Compd. Radiopharm. 37, 575-578.
    • (1995) J. Label. Compd. Radiopharm. , vol.37 , pp. 575-578
    • Mishani, E.1    Dence, C.S.2    McCarthy, T.J.3    Welch, M.J.4
  • 18
    • 0030040462 scopus 로고    scopus 로고
    • Formation of phenylpiperazine by a novel alumina supported bisalkylation
    • Mishani E., Dence C. S., McCarthy T. J. and Welch M. J. (1996) Formation of phenylpiperazine by a novel alumina supported bisalkylation. Tetrahedron Lett 37, 319-322.
    • (1996) Tetrahedron Lett , vol.37 , pp. 319-322
    • Mishani, E.1    Dence, C.S.2    McCarthy, T.J.3    Welch, M.J.4
  • 19
    • 0022892343 scopus 로고
    • Further studies of the putative serotonin agonist m-chlorophenylpiperazine: Evidence for a serotonin receptor mediated mechanism of action in humans
    • Mueller E. A., Murphy D. L, and Sunderland T. (1986) Further studies of the putative serotonin agonist m-chlorophenylpiperazine: Evidence for a serotonin receptor mediated mechanism of action in humans. Psychopharmacology 89, 388-391.
    • (1986) Psychopharmacology , vol.89 , pp. 388-391
    • Mueller, E.A.1    Murphy, D.L.2    Sunderland, T.3
  • 20
    • 0000927978 scopus 로고
    • New synthetic methods: 24. Organic reactions on aluminum oxide surfaces
    • Posner G. H. (1978) New synthetic methods: 24. Organic reactions on aluminum oxide surfaces. Angew. Chem. 90, 527-536.
    • (1978) Angew. Chem. , vol.90 , pp. 527-536
    • Posner, G.H.1
  • 21
    • 0028825878 scopus 로고
    • Neuropeptide receptors in health and disease: The molecular basis for in vivo imaging
    • Reubi J. C. (1995) Neuropeptide receptors in health and disease: The molecular basis for in vivo imaging. J. Nucl. Med. 36, 1825-1835.
    • (1995) J. Nucl. Med. , vol.36 , pp. 1825-1835
    • Reubi, J.C.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.