Radiosynthesis and PET imaging of [N-methyl-11C]LY257327 as a tracer for 5-HT transporters

Nuclear Medicine and Biology

Volumn 24, Issue 3, 1997, Pages 251-254

  Zea Ponce, Yolanda ^a,c   Baldwin, Ronald M ^a   Stratton, Morgan D ^a   Al Tikriti, Mohammed ^a   Soufer, Robert ^a   Schaus, John M ^b   Innis, Robert B ^a  

^a YALE UNIVERSITY SCHOOL OF MEDICINE   (United States)

^b ELI LILLY AND COMPANY   (United States)

^c NEW YORK STATE PSYCHIATRIC INSTITUTE   (United States)

Author keywords

N methyl 11C LY257327; PET; Serotonin reuptake sites; Serotonin transporter radiotracer

Indexed keywords

CARBON 11; CITALOPRAM; LY 214281; LY 257327; PIPERAZINE DERIVATIVE; SEROTONIN; SEROTONIN UPTAKE INHIBITOR; TETRALIN DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; BABOON; BRAIN REGION; DRUG PURITY; DRUG SYNTHESIS; DRUG UPTAKE; FEMALE; INTRAVENOUS DRUG ADMINISTRATION; NONHUMAN; POSITRON EMISSION TOMOGRAPHY;

ANIMALS; BRAIN; CARRIER PROTEINS; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; CITALOPRAM; FEMALE; ISOTOPE LABELING; MALE; MEMBRANE GLYCOPROTEINS; MEMBRANE TRANSPORT PROTEINS; NERVE TISSUE PROTEINS; OVARIECTOMY; PAPIO; PAROXETINE; PIPERAZINES; RADIOPHARMACEUTICALS; RATS; RATS, SPRAGUE-DAWLEY; SEROTONIN PLASMA MEMBRANE TRANSPORT PROTEINS; SEROTONIN UPTAKE INHIBITORS; SPECTROPHOTOMETRY, ULTRAVIOLET; TETRAHYDRONAPHTHALENES; TOMOGRAPHY, EMISSION-COMPUTED;

EID: 0030737592     PISSN: 09698051     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0969-8051(97)00062-0     Document Type: Article

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