Synthesis of 14C-labelled CGS 16949A (fadrozole HCI), a potent aromatase inhibitor

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 39, Issue 11, 1997, Pages 885-890

  Markus, Bohdan ^a   Allentoff, Alban J ^a   Desai, Mahesh ^a   Chaudhuri, Naba K ^a   Duelfer, Timothy ^a  

^a NOVARTIS PHARMA AG   (Switzerland)

Author keywords

Aromatase Inhibitor; Potassium 14C cyanide; 14C CGS 16949A

Indexed keywords

CYANIDES; POTASH;

AROMATASE INHIBITORS; IMIDAZOL; OESTROGENS; PHARMACOKINETIC STUDIES; POTASSIUM [14C]CYANIDE; SYNTHESIS PATHWAYS; SYNTHESISED; THIONYL CHLORIDES; TOLUNITRILE; [14C]CGS 16949A;

CHLORINE COMPOUNDS;

AROMATASE INHIBITOR; CARBON 14; FADROZOLE;

ANTINEOPLASTIC ACTIVITY; ARTICLE; BREAST CANCER; DRUG SYNTHESIS; ISOTOPE LABELING; JAPAN;

EID: 0030701561     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(199711)39:11<885::AID-JLCR33>3.0.CO;2-I     Document Type: Article

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