Thioperamide, a histamine H3 receptor antagonist, increases GABA release from the rat hypothalamus

Methods and Findings in Experimental and Clinical Pharmacology

Volumn 19, Issue 5, 1997, Pages 289-298

  Yamamoto, Yumiko ^a   Mochizuki, Takatoshi ^b   Okakura Mochizuki, Kaori ^a   Uno, Atsuhiko ^a   Yamatodani, Atsushi ^a,c  

^a OSAKA UNIVERSITY MEDICAL SCHOOL   (Japan)

^b EHIME UNIVERSITY SCHOOL OF MEDICINE   (Japan)

^c OSAKA UNIVERSITY   (Japan)

Author keywords

Clobenpropit; GABA; Histamine; Immepip; In vivo microdialysis; Rat; Thioperamide

Indexed keywords

ALPHA FLUOROMETHYLHISTIDINE; CLOBENPROPIT; EGTAZIC ACID; HISTAMINE H3 RECEPTOR ANTAGONIST; IMMEPIP; PHTHALALDEHYDE; THIOPERAMIDE; UNCLASSIFIED DRUG; 4 (1H IMIDAZOL 4 YLMETHYL)PIPERIDINE; 4 AMINOBUTYRIC ACID; 4-(1H-IMIDAZOL-4-YLMETHYL)PIPERIDINE; ALPHA-FLUOROMETHYLHISTIDINE; ANTIHISTAMINIC AGENT; CALCIUM; DRUG DERIVATIVE; ENZYME INHIBITOR; HISTAMINE AGONIST; HISTAMINE H3 RECEPTOR; HISTIDINE DECARBOXYLASE; HISTIDINE DERIVATIVE; IMIDAZOLE DERIVATIVE; PIPERIDINE DERIVATIVE; THIOUREA;

4 AMINOBUTYRIC ACID RELEASE; ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; CONTROLLED STUDY; DRUG EFFECT; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HISTAMINE RELEASE; HYPOTHALAMUS; MICRODIALYSIS; NEUROTRANSMITTER RELEASE; NONHUMAN; RAT; ANIMAL; DRUG ANTAGONISM; MALE; METABOLISM; NERVE CELL; WISTAR RAT;

ANIMALS; CALCIUM; ENZYME INHIBITORS; GAMMA-AMINOBUTYRIC ACID; HISTAMINE AGONISTS; HISTAMINE ANTAGONISTS; HISTIDINE DECARBOXYLASE; HYPOTHALAMUS; IMIDAZOLES; MALE; METHYLHISTIDINES; MICRODIALYSIS; NEURONS; PIPERIDINES; RATS; RATS, WISTAR; RECEPTORS, HISTAMINE H3; THIOUREA;

EID: 0030612872     PISSN: 03790355     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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