Selectivity of [PHE-I7], [Ala6], and [D-Ala4, Gln5, Tyr6] substituted ACTH (4-10) analogues for the melanocortin receptors

Peptides

Volumn 18, Issue 5, 1997, Pages 761-763

  Schiöth, Helgi B ^a,b   Muceniece, Ruta ^a   Wikberg, Jarl E S ^a  

^a UPPSALA UNIVERSITY   (Sweden)

^b UPPSALA UNIVERSITY   (Sweden)

Author keywords

ACTH; BIM 22015; Ligand binding; Melanocortin receptor subtypes; MSH

Indexed keywords

BIM 22015; CORTICOTROPIN[4-10]; CORTICOTROPIN[4-10] DERIVATIVE; HORMONE RECEPTOR; INTERMEDIN; UNCLASSIFIED DRUG; ACTH (4 10); CORTICOTROPIN; CORTICOTROPIN RECEPTOR; DRUG DERIVATIVE; MELANOCORTIN 3 RECEPTOR; MELANOCORTIN 4 RECEPTOR; MELANOCORTIN 5 RECEPTOR; MELANOCORTIN RECEPTOR; PEPTIDE FRAGMENT; RECEPTOR;

ANIMAL CELL; ARTICLE; BINDING COMPETITION; CELL STRAIN COS1; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG COMPETITION; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG SPECIFICITY; HORMONE RECEPTOR INTERACTION; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY; ANIMAL; DRUG ANTAGONISM; GENETICS; HUMAN; METABOLISM; MOLECULAR CLONING; PROTEIN BINDING; RADIOASSAY;

ADRENOCORTICOTROPIC HORMONE; ANIMALS; CLONING, MOLECULAR; COS CELLS; HUMANS; PEPTIDE FRAGMENTS; PROTEIN BINDING; RADIOLIGAND ASSAY; RECEPTOR, MELANOCORTIN, TYPE 3; RECEPTOR, MELANOCORTIN, TYPE 4; RECEPTORS, CORTICOTROPIN; RECEPTORS, MELANOCORTIN; RECEPTORS, PEPTIDE;

EID: 0030612436     PISSN: 01969781     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0196-9781(97)00126-5     Document Type: Article

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