메뉴 건너뛰기




Volumn 6, Issue 4, 1997, Pages 250-258

Brimonidine: A new alpha2-adrenoreceptor agonist for glaucoma treatment

Author keywords

Alpha2 adrenoreceptor agonist; Brimonidine

Indexed keywords

BETAXOLOL; BRIMONIDINE; TIMOLOL; ALPHA ADRENERGIC RECEPTOR STIMULATING AGENT; BETA ADRENERGIC RECEPTOR BLOCKING AGENT; EYE DROPS; QUINOXALINE DERIVATIVE;

EID: 0030611851     PISSN: 10570829     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review
Times cited : (93)

References (52)
  • 1
    • 0026409550 scopus 로고
    • Relationship between intraocular pressure and primary open-angle glaucoma among white and black Americans
    • Sommer A, Tielsch JM, Katz J, et al. Relationship between intraocular pressure and primary open-angle glaucoma among white and black Americans. Arch Ophthalmol 1991;109:1090-5.
    • (1991) Arch Ophthalmol , vol.109 , pp. 1090-1095
    • Sommer, A.1    Tielsch, J.M.2    Katz, J.3
  • 2
    • 0028048319 scopus 로고
    • The global impact of glaucoma
    • Thylefors B, Négrel AD. The global impact of glaucoma. Bull WHO 1994;72:323-6.
    • (1994) Bull WHO , vol.72 , pp. 323-326
    • Thylefors, B.1    Négrel, A.D.2
  • 4
    • 0029752042 scopus 로고    scopus 로고
    • Preclinical evaluation of brimonidine
    • Burke J, Schwartz M. Preclinical evaluation of brimonidine. Surv Ophthalmol 1996;41(suppl 1):9-18.
    • (1996) Surv Ophthalmol , vol.41 , Issue.1 SUPPL. , pp. 9-18
    • Burke, J.1    Schwartz, M.2
  • 5
    • 0014026037 scopus 로고
    • Ophthalmological studies with dichlorophenyl-aminoimidazoline
    • Makabe R. Ophthalmological studies with dichlorophenyl-aminoimidazoline. Dtsch Med Wochenschr 1966;91:1686.
    • (1966) Dtsch Med Wochenschr , vol.91 , pp. 1686
    • Makabe, R.1
  • 6
    • 0000217817 scopus 로고    scopus 로고
    • Catecholamines, sympathomimetic drugs, and adrenergic receptor antagonists
    • Hardman JG, Gilman AG, Limbird LE, eds. New York: McGraw-Hill
    • Hoffman BB, Lefkowitz RJ. Catecholamines, sympathomimetic drugs, and adrenergic receptor antagonists. In: Hardman JG, Gilman AG, Limbird LE, eds. Goodman and Gilman's The Pharmacological Basis of Therapeutics. 9th ed. New York: McGraw-Hill, 1996:199-248.
    • (1996) Goodman and Gilman's the Pharmacological Basis of Therapeutics. 9th Ed. , pp. 199-248
    • Hoffman, B.B.1    Lefkowitz, R.J.2
  • 7
    • 0017895549 scopus 로고
    • The response of ophthalmic arterial pressure to topically applied clonidine
    • Krieglstein GK, Gramer E. The response of ophthalmic arterial pressure to topically applied clonidine. Graefes Arch Clin Exp Ophthalmol 1978;207:1-5.
    • (1978) Graefes Arch Clin Exp Ophthalmol , vol.207 , pp. 1-5
    • Krieglstein, G.K.1    Gramer, E.2
  • 8
    • 0019419041 scopus 로고
    • The effect of topical clonidine on intraocular pressure
    • Hodapp E, Kolker, AE, Kass MA, al. The effect of topical clonidine on intraocular pressure. Arch Ophthalmol 1981;99:1208.
    • (1981) Arch Ophthalmol , vol.99 , pp. 1208
    • Hodapp, E.1    Kolker, A.E.2    Kass, M.A.3
  • 9
    • 0018273075 scopus 로고
    • Pharmacological study of para-aminoclonidine, an alpha sympathomimetic
    • Rouot B, Leclerc G, Bieth N, et al. Pharmacological study of para-aminoclonidine, an alpha sympathomimetic. Coll R Acad Sci 1978;286:909-12.
    • (1978) Coll R Acad Sci , vol.286 , pp. 909-912
    • Rouot, B.1    Leclerc, G.2    Bieth, N.3
  • 10
    • 0004982046 scopus 로고
    • Studies of p-aminoclonidine as a potential antiglaucoma agent
    • Chandler ML, DeSantis L. Studies of p-aminoclonidine as a potential antiglaucoma agent. Invest Ophthalmol Vis Sci 1985;26 (suppl):227.
    • (1985) Invest Ophthalmol Vis Sci , vol.26 , Issue.SUPPL. , pp. 227
    • Chandler, M.L.1    DeSantis, L.2
  • 11
  • 12
    • 0023848670 scopus 로고
    • ALO 2145 reduces the IOP elevation after anterior segment laser surgery
    • Brown RH, Stewart RH, Lynch MG, et al. ALO 2145 reduces the IOP elevation after anterior segment laser surgery. Ophthalmology 1988;95:378-84.
    • (1988) Ophthalmology , vol.95 , pp. 378-384
    • Brown, R.H.1    Stewart, R.H.2    Lynch, M.G.3
  • 13
    • 0026637132 scopus 로고
    • Apraclonidine and argon laser trabeculoplasty
    • Holmwood PC, Chase RD, Krupin T, et al. Apraclonidine and argon laser trabeculoplasty. Am J Ophthalmol 1992;114:19-22.
    • (1992) Am J Ophthalmol , vol.114 , pp. 19-22
    • Holmwood, P.C.1    Chase, R.D.2    Krupin, T.3
  • 14
    • 0023222745 scopus 로고
    • Effect of ALO-2145 on intraocular pressure following argon laser trabeculoplasty
    • Robin AL, Pollack IP, House B, Enger C. Effect of ALO-2145 on intraocular pressure following argon laser trabeculoplasty. Arch Ophthalmol 1987;105:646-50.
    • (1987) Arch Ophthalmol , vol.105 , pp. 646-650
    • Robin, A.L.1    Pollack, I.P.2    House, B.3    Enger, C.4
  • 15
    • 0023220944 scopus 로고
    • Effects of topical ALO 2145 (p-aminoclonidine hydrochloride,) on intraocular pressure rise following argon laser iridotomy
    • Robin AL, Pollack IP, DeFaller JM. Effects of topical ALO 2145 (p-aminoclonidine hydrochloride,) on intraocular pressure rise following argon laser iridotomy. Arch Ophthalmol 1987;105:1208-11.
    • (1987) Arch Ophthalmol , vol.105 , pp. 1208-1211
    • Robin, A.L.1    Pollack, I.P.2    DeFaller, J.M.3
  • 16
    • 0026589778 scopus 로고
    • Prophylactic use of apraclonidine for intraocular pressure increase after Nd:YAG capsulotomies
    • Silverstone DE, Brint SF, Olander KW, et al. Prophylactic use of apraclonidine for intraocular pressure increase after Nd:YAG capsulotomies. Am J Ophthalmol 1992;113:401-5.
    • (1992) Am J Ophthalmol , vol.113 , pp. 401-405
    • Silverstone, D.E.1    Brint, S.F.2    Olander, K.W.3
  • 17
    • 0028883384 scopus 로고
    • Short-term efficacy of apraclonidine hydrochloride added to maximum-tolerated medical therapy for glaucoma
    • Robin AL, Ritch R, Shin DH, et al. Short-term efficacy of apraclonidine hydrochloride added to maximum-tolerated medical therapy for glaucoma. Am J Ophthalmol 1995;120:423-32.
    • (1995) Am J Ophthalmol , vol.120 , pp. 423-432
    • Robin, A.L.1    Ritch, R.2    Shin, D.H.3
  • 18
    • 0028967586 scopus 로고
    • Clinical experience with the long-term use of 1% apraclonidine. Incidence of allergic reactions
    • Butler P, Mannschreck M, Lin S, et al. Clinical experience with the long-term use of 1% apraclonidine. Incidence of allergic reactions. Arch Ophthalmol 1995;113:293-6.
    • (1995) Arch Ophthalmol , vol.113 , pp. 293-296
    • Butler, P.1    Mannschreck, M.2    Lin, S.3
  • 19
    • 0027272396 scopus 로고
    • Comparison of apraclonidine and timolol in chronic open-angle glaucoma
    • Nagasubramanian S, Hitchings RA, Demailly P, et al. Comparison of apraclonidine and timolol in chronic open-angle glaucoma. Ophthalmology 1993;100:1318-23.
    • (1993) Ophthalmology , vol.100 , pp. 1318-1323
    • Nagasubramanian, S.1    Hitchings, R.A.2    Demailly, P.3
  • 20
    • 0028959409 scopus 로고
    • The efficacy of apraclonidine as an adjunct to timolol therapy
    • Stewart WC, Ritch R, Shin DH, et al. The efficacy of apraclonidine as an adjunct to timolol therapy. Arch Ophthalmol 1995;113:287-92.
    • (1995) Arch Ophthalmol , vol.113 , pp. 287-292
    • Stewart, W.C.1    Ritch, R.2    Shin, D.H.3
  • 22
    • 0342595900 scopus 로고
    • AGN 190342 (UK-14304-18) stimulates an imidazoline receptor to lower intraocular pressure (IOP) in conscious monkeys
    • Burke J, Padillo E, Shan T, et al. AGN 190342 (UK-14304-18) stimulates an imidazoline receptor to lower intraocular pressure (IOP) in conscious monkeys. Invest Ophthalmol Vis Sci 1991;32 (suppl):867.
    • (1991) Invest Ophthalmol Vis Sci , vol.32 , Issue.SUPPL. , pp. 867
    • Burke, J.1    Padillo, E.2    Shan, T.3
  • 24
    • 4244057996 scopus 로고
    • Use of recombinant human alpha adrenergic receptors for the pharmacological evaluation of alpha adrenergic ocular hypertensive agents
    • Gluchowski C, Jeon YT, Wetzel JM, et al. Use of recombinant human alpha adrenergic receptors for the pharmacological evaluation of alpha adrenergic ocular hypertensive agents. Invest Ophthalmol Vis Sci 1994;35(suppl):1399.
    • (1994) Invest Ophthalmol Vis Sci , vol.35 , Issue.SUPPL. , pp. 1399
    • Gluchowski, C.1    Jeon, Y.T.2    Wetzel, J.M.3
  • 25
    • 0017750402 scopus 로고
    • Presynaptic receptors and the regulation of transmitter release in the peripheral and central nervous system
    • Sixth Gaddum Memorial Lecture
    • Langer SZ. Presynaptic receptors and the regulation of transmitter release in the peripheral and central nervous system. Sixth Gaddum Memorial Lecture. Br J Ophthalmol 1977;60:481-97.
    • (1977) Br J Ophthalmol , vol.60 , pp. 481-497
    • Langer, S.Z.1
  • 26
    • 0023889603 scopus 로고
    • 2-adrenergic receptors: Delineation of domains involved in effector coupling and ligand binding specificity
    • 2-adrenergic receptors: delineation of domains involved in effector coupling and ligand binding specificity. Science 1989;240:1310-6.
    • (1989) Science , vol.240 , pp. 1310-1316
    • Kobilka, B.K.1    Kobilka, T.S.2    Daniel, K.3
  • 28
    • 0027231501 scopus 로고
    • The efficacy of brimonidine in decreasing elevation in intraocular pressure after laser trabeculoplasty
    • Barnebey HS, Robin AL, Zimmerman TJ, et al. The efficacy of brimonidine in decreasing elevation in intraocular pressure after laser trabeculoplasty. Ophthalmology 1993;100:1083-8.
    • (1993) Ophthalmology , vol.100 , pp. 1083-1088
    • Barnebey, H.S.1    Robin, A.L.2    Zimmerman, T.J.3
  • 29
    • 0022998446 scopus 로고
    • 2 agonist (UK-14304-18) in cats, rabbits, and monkeys
    • 2 agonist (UK-14304-18) in cats, rabbits, and monkeys. Curr Eye Res 1986;5:665-76.
    • (1986) Curr Eye Res , vol.5 , pp. 665-676
    • Burke, J.A.1    Potter, D.E.2
  • 30
    • 0024372244 scopus 로고
    • Can UK-14304-18 lower IOP in rabbits by a peripheral mechanism?
    • Burke J, Crosson C, Potter DE. Can UK-14304-18 lower IOP in rabbits by a peripheral mechanism? Curr Eye Res 1989;8:547-52.
    • (1989) Curr Eye Res , vol.8 , pp. 547-552
    • Burke, J.1    Crosson, C.2    Potter, D.E.3
  • 31
  • 32
    • 0028588575 scopus 로고
    • Apraclonidine and brimonidine effects on anterior ocular and cardiovascular physiology on normal and sympathectomized monkeys
    • Gabelt BT, Robinson JC, Hubbard WC, et al. Apraclonidine and brimonidine effects on anterior ocular and cardiovascular physiology on normal and sympathectomized monkeys. Exp Eye Res 1994;59:633-44.
    • (1994) Exp Eye Res , vol.59 , pp. 633-644
    • Gabelt, B.T.1    Robinson, J.C.2    Hubbard, W.C.3
  • 33
    • 0029082601 scopus 로고
    • Adrenergic and imidazoline receptor-mediated responses to UK-14302-18 (brimonidine) in rabbits and monkeys: A species difference
    • Reis D, Bousquet P, Parini A, eds. New York: New York Academy of Science
    • Burke J, Kharlamb A, Shan T, et al. Adrenergic and imidazoline receptor-mediated responses to UK-14302-18 (brimonidine) in rabbits and monkeys: a species difference. In: Reis D, Bousquet P, Parini A, eds. The Imidazoline Receptor: Pharmacology, Functions, Ligands, and Relevance to Biology and Medicine. New York: New York Academy of Science, 1995:78-95.
    • (1995) The Imidazoline Receptor: Pharmacology, Functions, Ligands, and Relevance to Biology and Medicine , pp. 78-95
    • Burke, J.1    Kharlamb, A.2    Shan, T.3
  • 34
    • 0343465789 scopus 로고
    • The cynomolgus monkey has a CNS imidazoline receptor which mediates IOP and cardiovascular responses to UK-14304 (AGN 190342)
    • Kharlamb A, Shan T, Runde E, et al. The cynomolgus monkey has a CNS imidazoline receptor which mediates IOP and cardiovascular responses to UK-14304 (AGN 190342). Invest Ophthalmol Vis Sci 1992;33(suppl):1115.
    • (1992) Invest Ophthalmol Vis Sci , vol.33 , Issue.SUPPL. , pp. 1115
    • Kharlamb, A.1    Shan, T.2    Runde, E.3
  • 35
    • 0029731764 scopus 로고    scopus 로고
    • Clinical experience with brimonidine 0.2% and timolol 0.5% in glaucoma and ocular hypertension
    • Schuman JS. Clinical experience with brimonidine 0.2% and timolol 0.5% in glaucoma and ocular hypertension. Surv Ophthalmol 1996;41(suppl 1):27-37.
    • (1996) Surv Ophthalmol , vol.41 , Issue.1 SUPPL. , pp. 27-37
    • Schuman, J.S.1
  • 36
    • 0029731441 scopus 로고    scopus 로고
    • A comparison of the safety and efficacy of twice daily brimonidine 0.2% versus betaxolol 0.25% in subjects with elevated intraocular pressure
    • Serle JB, The brimonidine Study Group III. A comparison of the safety and efficacy of twice daily brimonidine 0.2% versus betaxolol 0.25% in subjects with elevated intraocular pressure. Surv Ophthalmol 1996;41(suppl 1):39-47.
    • (1996) Surv Ophthalmol , vol.41 , Issue.1 SUPPL. , pp. 39-47
    • Serle, J.B.1
  • 37
    • 0001535125 scopus 로고
    • Comparative effects of brimonidine, p-aminoclonidine and clonidine on arteriolar caliber in human retinal tissue
    • Spada CS, Nieves AL, Burke JA, et al. Comparative effects of brimonidine, p-aminoclonidine and clonidine on arteriolar caliber in human retinal tissue. Invest Ophthalmol Vis Sci 1995;36(suppl): 1041.
    • (1995) Invest Ophthalmol Vis Sci , vol.36 , Issue.SUPPL. , pp. 1041
    • Spada, C.S.1    Nieves, A.L.2    Burke, J.A.3
  • 39
    • 0004660888 scopus 로고
    • Human ocular microcirculation: Intravital microscopy of retinal and choroid circulations grafted into the cheek pouch of the hamster
    • Weinreb RN, Joyner WL, Wheeler LA, eds. Elsevier Scientific: Amsterdam
    • Joyner WL, Tang T, Macek BA, et al. Human ocular microcirculation: intravital microscopy of retinal and choroid circulations grafted into the cheek pouch of the hamster. In: Weinreb RN, Joyner WL, Wheeler LA, eds. Biology of the Ocular Microcirculation. Elsevier Scientific: Amsterdam, 1992:61-70.
    • (1992) Biology of the Ocular Microcirculation , pp. 61-70
    • Joyner, W.L.1    Tang, T.2    Macek, B.A.3
  • 40
    • 0008441359 scopus 로고
    • Drug distribution of brimonidine in albino and pigmented rabbit eyes
    • Chien DS, Richman J, Zolezio H, et al. Drug distribution of brimonidine in albino and pigmented rabbit eyes. Pharm Res 1992; 9:336.
    • (1992) Pharm Res , vol.9 , pp. 336
    • Chien, D.S.1    Richman, J.2    Zolezio, H.3
  • 41
    • 0029072535 scopus 로고
    • Comparative ocular pharmacokinetics of brimonidine after a single dose application to the eyes of albino and pigmented rabbits
    • Acheampong AA, Shackleton M, Tang-Liu DDS. Comparative ocular pharmacokinetics of brimonidine after a single dose application to the eyes of albino and pigmented rabbits. Drug Metab Disposition 1995;27:708-12.
    • (1995) Drug Metab Disposition , vol.27 , pp. 708-712
    • Acheampong, A.A.1    Shackleton, M.2    Tang-Liu, D.D.S.3
  • 42
    • 34547392774 scopus 로고
    • One year oral and one year ocular toxicity studies of AGN-190342-LF (brimonidine tartrate) in cynomolgus monkeys
    • Angelov O, Wiese A, Tang-Liu D, et al. One year oral and one year ocular toxicity studies of AGN-190342-LF (brimonidine tartrate) in cynomolgus monkeys. Toxicologist 1994;14:255.
    • (1994) Toxicologist , vol.14 , pp. 255
    • Angelov, O.1    Wiese, A.2    Tang-Liu, D.3
  • 43
    • 0000893624 scopus 로고
    • Brimonidine tartrate: A one-month dose response study
    • Derick RJ, Walters TR, Robin AL, et al. Brimonidine tartrate: a one-month dose response study. Invest Ophthalmol Vis Sci 1993; 34(suppl):929.
    • (1993) Invest Ophthalmol Vis Sci , vol.34 , Issue.SUPPL. , pp. 929
    • Derick, R.J.1    Walters, T.R.2    Robin, A.L.3
  • 44
    • 34547392959 scopus 로고
    • Brimonidine tartrate dose-response study in glaucoma and ocular hypertension
    • Robin AL, Barnebey HS, Choplin N, et al. Brimonidine tartrate dose-response study in glaucoma and ocular hypertension. Eur J Ophthalmol 1995;5(suppl):156.
    • (1995) Eur J Ophthalmol , vol.5 , Issue.SUPPL. , pp. 156
    • Robin, A.L.1    Barnebey, H.S.2    Choplin, N.3
  • 45
    • 0008788278 scopus 로고    scopus 로고
    • A comparison of the safety and efficacy of brimonidine 0.2%, bid verses tid, in subjects with elevated intraocular pressure
    • Rosenthal AL, Walters T, Berg E, et al. A comparison of the safety and efficacy of brimonidine 0.2%, bid verses tid, in subjects with elevated intraocular pressure. Invest Ophthalmol Vis Sci 1996;37 (suppl):1102.
    • (1996) Invest Ophthalmol Vis Sci , vol.37 , Issue.SUPPL. , pp. 1102
    • Rosenthal, A.L.1    Walters, T.2    Berg, E.3
  • 46
    • 0028814882 scopus 로고
    • The cardiovascular, pulmonary, and ocular hypotensive effects of 0.2% brimonidine
    • Nordlund JR, Pasquale LR, Robin AL, et al. The cardiovascular, pulmonary, and ocular hypotensive effects of 0.2% brimonidine. Arch Ophthalmol 1995;113:77-83.
    • (1995) Arch Ophthalmol , vol.113 , pp. 77-83
    • Nordlund, J.R.1    Pasquale, L.R.2    Robin, A.L.3
  • 47
    • 0027517943 scopus 로고
    • Brimonidine in the prevention of intraocular pressure elevation following argon laser trabeculoplasty
    • David R, Spaeth GL, Clevenger CE, et al. Brimonidine in the prevention of intraocular pressure elevation following argon laser trabeculoplasty. Arch Ophthalmol 1993;111:1387-90.
    • (1993) Arch Ophthalmol , vol.111 , pp. 1387-1390
    • David, R.1    Spaeth, G.L.2    Clevenger, C.E.3
  • 48
    • 0028805185 scopus 로고
    • Effect of brimonidine 0.5% on intraocular pressure spikes following 360° argon laser trabeculoplasty
    • Brimonidine-ALT Study Group. Effect of brimonidine 0.5% on intraocular pressure spikes following 360° argon laser trabeculoplasty. Ophthalmic Surg Lasers 1995;26:404-9.
    • (1995) Ophthalmic Surg Lasers , vol.26 , pp. 404-409
  • 50
    • 0017805415 scopus 로고
    • Central nervous system depressant actions of clonidine and UK-14,304: Partial dissociation of EEG and behavioral effects
    • Ashton H, Rawlins MD. Central nervous system depressant actions of clonidine and UK-14,304: partial dissociation of EEG and behavioral effects. Br J Clin Pharmacol 1978;5:135-40.
    • (1978) Br J Clin Pharmacol , vol.5 , pp. 135-140
    • Ashton, H.1    Rawlins, M.D.2
  • 51
    • 0027248053 scopus 로고
    • Neuroprotection by the alpha-2 adrenoceptor agonist dexmedetomidine in a focal model of cerebral ischemia
    • Maier C, Steinberg GK, Sun GH, et al. Neuroprotection by the alpha-2 adrenoceptor agonist dexmedetomidine in a focal model of cerebral ischemia. Anesthesiology 1993;79:306-12.
    • (1993) Anesthesiology , vol.79 , pp. 306-312
    • Maier, C.1    Steinberg, G.K.2    Sun, G.H.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.