Characterisation of the binding of [3H]MDL 105,519, a radiolabelled antagonist for the N-methyl-D-aspartate-associated glycine site, to pig cortical brain membranes

Neuroscience Letters

Volumn 226, Issue 2, 1997, Pages 79-82

  Hofner G ^a   Wanner, K Th ^a  

^a Inst Pharm und Lebensmittelchemie   (Germany)

Author keywords

3H MDL 105,519; Agonist; Antagonist; Glycine site; N Methyl D aspartate receptor complex; Pharmacological profile; Pig cortical brain membranes

Indexed keywords

GLYCINE RECEPTOR; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; N METHYL DEXTRO ASPARTIC ACID RECEPTOR BLOCKING AGENT; N METHYL DEXTRO ASPARTIC ACID RECEPTOR STIMULATING AGENT; RADIOLIGAND; 3 (2 CARBOXY 2 PHENYLETHENYL) 4,6 DICHLORO 1H INDOLE 2 CARBOXYLIC ACID; AMINO ACID RECEPTOR BLOCKING AGENT; AMINO ACID RECEPTOR STIMULATING AGENT; DIZOCILPINE MALEATE; GLYCINE; INDOLE DERIVATIVE; TRITIUM;

ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; BRAIN MEMBRANE; CONTROLLED STUDY; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING; SWINE; ANIMAL; BINDING COMPETITION; BINDING SITE; CELL MEMBRANE; KINETICS; METABOLISM; RADIOASSAY;

ANIMALS; BINDING SITES; BINDING, COMPETITIVE; CELL MEMBRANE; CEREBRAL CORTEX; DIZOCILPINE MALEATE; EXCITATORY AMINO ACID AGONISTS; EXCITATORY AMINO ACID ANTAGONISTS; GLYCINE; INDOLES; KINETICS; RADIOLIGAND ASSAY; RECEPTORS, N-METHYL-D-ASPARTATE; SWINE; TRITIUM;

EID: 0030611299     PISSN: 03043940     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0304-3940(97)00238-3     Document Type: Article

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