Importance of h5-HT(1B) receptor selectivity for 5-HT terminal autoreceptor activity: An in vivo microdialysis study in the freely-moving guinea-pig

Neuropharmacology

Volumn 36, Issue 4-5, 1997, Pages 549-557

  Roberts, C ^a   Price, G W ^a   Gaster, L ^a   Jones, B J ^a   Middlemiss, D N ^a   Routledge, C ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

5 HT; 5 HT(1B 1D) receptors; Guinea pig; Microdialysis

Indexed keywords

2,3,6,7 TETRAHYDRO 1' METHYL 5 [[2' METHYL 4' (5 METHYL 1,2,4 OXADIAZOL 3 YL) 4 BIPHENYLYL]CARBONYL]SPIRO[FURO[2,3 F]INDOLE 3,4' PIPERIDINE]; AUTORECEPTOR; BUSPIRONE; DEXFENFLURAMINE; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); KETANSERIN; MESULERGINE; METITEPINE; MIANSERIN; PARTIAL AGONIST; RADIOISOTOPE; SB 216641; SB 219085; SB 220272; SEROTONIN; SEROTONIN 1B RECEPTOR; SEROTONIN 1D RECEPTOR; SEROTONIN AGONIST; SEROTONIN ANTAGONIST; SEROTONIN RECEPTOR AFFECTING AGENT; UNCLASSIFIED DRUG; LIGAND; SEROTONIN RECEPTOR;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BRAIN SLICE; CELL LINE; CHO CELL; CONTROLLED STUDY; DRUG EFFICACY; DRUG SELECTIVITY; FRONTAL CORTEX; GUINEA PIG; HUMAN; HUMAN CELL; INTRAPERITONEAL DRUG ADMINISTRATION; MICRODIALYSIS; NERVE ENDING; NONHUMAN; PRIORITY JOURNAL; RAPHE NUCLEUS; RECEPTOR AFFINITY; RECEPTOR BINDING; SEROTONIN RELEASE; SEROTONINERGIC NERVE; ANIMAL; BRAIN CORTEX; BRAIN LEVEL; DRUG EFFECT; ELECTROCHEMISTRY; HAMSTER; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; MALE; METABOLISM; PHYSIOLOGY;

ANIMALS; AUTORECEPTORS; BRAIN CHEMISTRY; CEREBRAL CORTEX; CHO CELLS; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; CRICETINAE; ELECTROCHEMISTRY; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); GUINEA PIGS; LIGANDS; MALE; MICRODIALYSIS; RAPHE NUCLEI; RECEPTORS, SEROTONIN; SEROTONIN;

EID: 0030610866     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0028-3908(97)00026-9     Document Type: Article

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