Analysis of α1-adrenoceptors in rabbit lower urinary tract and mesenteric artery

European Journal of Pharmacology

Volumn 327, Issue 1, 1997, Pages 25-32

  Van Der Graaf, Pieter H ^a   Deplanne, Valérie ^a   Duquenne, Chantal ^a   Angel, Itzchak ^a  

^a SANOFI   (France)

Author keywords

Mesenteric artery; Prostate; Rabbit; Trigone; Urethra; 1 Adrenoceptor

Indexed keywords

2 [[2 (2,6 DIMETHOXYPHENOXY)ETHYL]AMINOMETHYL] 1,4 BENZODIOXAN; 5 CHLORO N [2 (2 CYCLOPROPYLMETHOXYPHENOXY)ETHYL] ALPHA,ALPHA DIMETHYL 1H INDOLE 3 ETHANAMINE; 5 METHYLURAPIDIL; 8 [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] 8 AZASPIRO[4.5]DECANE 7,9 DIONE; ALFUZOSIN; ALPHA 1 ADRENERGIC RECEPTOR; ALPHA 1 ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA ETHYL 3,4,5 TRIMETHOXY ALPHA [3 [[2 (2 METHOXYPHENOXY)ETHYL]AMINO]PROPYL]BENZENEACETONITRILE FUMARATE; COCAINE; CORTICOSTERONE; INDORAMIN; PHENTOLAMINE; PHENYLEPHRINE; PRAZOSIN; RECEPTOR SUBTYPE; TAMSULOSIN; TERAZOSIN; ALPHA ADRENERGIC RECEPTOR BLOCKING AGENT; PIPERAZINE DERIVATIVE;

ANIMAL TISSUE; ARTICLE; CATECHOLAMINE UPTAKE; CONTROLLED STUDY; MALE; MESENTERIC ARTERY; NONHUMAN; PRIORITY JOURNAL; PROSTATE; RABBIT; SMOOTH MUSCLE RELAXATION; URETHRA; ANIMAL; CLASSIFICATION; DRUG EFFECT; IN VITRO STUDY; PHYSIOLOGY; URINARY TRACT; URINARY TRACT FUNCTION;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMALS; MALE; MESENTERIC ARTERIES; PHENYLEPHRINE; PIPERAZINES; PROSTATE; RABBITS; RECEPTORS, ADRENERGIC, ALPHA-1; URETHRA; URINARY TRACT; URINARY TRACT PHYSIOLOGY;

EID: 0030610262     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(97)89674-4     Document Type: Article

References (39)

1. Agrawal D.K., Triggle C.R., Daniel E.E. Pharmacological characterization of the postsynaptic alpha adrenoceptors in vascular smooth muscle from canine and rat mesenteric beds. J. Pharmacol. Exp. Ther. 229:1984;831-838.
2. Andersson K.-E. Current concepts in the treatment of disorders of micturition. Drugs. 35:1988;477-494.
3. Andersson K.-E. Pharmacology of lower urinary tract smooth muscles and penile erectile tissues. Pharmacol. Rev. 45:1993;253-308.
4. Arunlakshana O., Schild H.O. Some quantitative uses of drug antagonists. Br. J. Pharmacol. 14:1959;48-58.
5. 1-adrenoceptor subtypes mediate contraction in rabbit aorta and urethra. Eur. J. Pharmacol. 287:1995;153-161.
6. 1A-Adrenoceptor subtype mediates contraction of the rat urethra. J. Auton. Pharmacol. 14:1994;375-381.
7. De Lean A.P., Munson P.J., Rodbard D. Simultaneous analysis of families of sigmoidal curves: application to bioassay, radioligand assay and physiological dose-response curves. Am. J. Physiol. 235:1978;E97-E102.
8. Deplanne V., Galzin A.M. Functional characterization of alpha-1-adrenoceptor subtypes in the prostatic urethra and trigone of male rabbit. J. Pharmacol. Exp. Ther. 278:1996;527-534.
9. Digges K.G., Summers R.J. Characterization of postsynaptic α-adrenoceptors in rat aortic strips and portal veins. Br. J. Pharmacol. 79:1983;655-665.
10. Drew G.M. What do antagonists tell us about α-adrenoceptors? Clin. Sci. 68:1985;15s-16s.
11. 1-Adrenoceptor subclassification in vascular smooth muscle. Trends Pharmacol. Sci. 7:1986;347-349.
12. 1-Adrenoceptor classification: sharpening Occam's razor. Trends Pharmacol. Sci. 15:1994;167-170.
13. 1-adrenoceptors in human prostate: implications for adrenoceptor classification. Mol. Pharmacol. 49:1996;209-215.
14. 1-adrenoceptors. Eur. J. Pharmacol. 272:1995;R5-R6.
15. Hieble J.P., Bondinell W.E., Ruffolo R.R. Jr. α- and α-adrenoceptors: from gene to the clinic. 1. Molecular biology and adrenoceptor subclassification J. Med. Chem. 38:1995;3415-3444.
16. 1-adrenoceptors: consensus update. Pharmacol. Rev. 47:1995;267-270.
17. 1-adrenoceptor subtypes in the rabbit prostate. J. Auton. Pharmacol. 15:1995;271-278.
18. Holck M.I., Jones C.H.M., Haeusler G. Differential interactions of clonidine and methoxamine with the postsynaptic α-adrenoceptor of rabbit main pulmonary artery. J. Cardiovasc. Pharmacol. 5:1983;240-248.
19. Honda K., Nakagawa C. Alpha-1 adrenoceptor antagonist effects of the optical isomers of YM-12617 in rabbit lower urinary tract and prostate. J. Pharmacol. Exp. Ther. 239:1986;512-516.
20. 1-Adrenoceptor subtype mediating contraction of the smooth muscle in the lower urinary tract and prostate of rabbits. Naunyn-Schmiedeberg's Arch. Pharmacol. 330:1985;16-21.
21. Jenkinson D.H. How we describe competitive antagonists: three questions of usage. Trends Pharmacol. Sci. 12:1991;53-54.
22. Jenkinson D.H., Barnard E.A., Hoyer D., Humphrey P.P.A., Leff P., Shankley N.P. Recommendations on terms and symbols in quantitative pharmacology. Pharmacol. Rev. 47:1995;255-266.
23. Kenakin, T.P., 1993. Pharmacological Analysis of Drug-Receptor Interaction. Raven Press, New York, NY, p. 176.
24. 1D-adrenoceptor mediating the contractile response of rat aorta to noradrenaline. Br. J. Pharmacol. 115:1995;981-986.
25. 1-adrenoceptor subtypes involved in adrenergic contractions of dog blood vessels. Br. J. Pharmacol. 112:1994;1167-1173.
26. Langer S.Z., Trendelenburg U. The effect of a saturable uptake mechanism on the slopes of dose-response curves for sympathomimetic amines and on the shifts of dose-response curves produced by a competitive antagonist. J. Pharmacol. Exp. Ther. 167:1969;117-142.
27. 1-adrenoceptor antagonist in the lower urinary tract. Br. J. Pharmacol. 109:1993;1282-1289.
28. McGrath J., Wilson V. α-Adrenoceptor subclassification by classical and response-related methods: same question, different answers. Trends Pharmacol. Sci. 9:1988;162-165.
29. Medgett I.C., Langer S.Z. Heterogeneity of smooth muscle alpha adrenoceptors in rat tail artery in vitro. J. Pharmacol. Exp. Ther. 229:1984;823-830.
30. 1-adrenoceptor subtypes. Naunyn-Schmiedeberg's Arch. Pharmacol. 352:1995;1-10.
31. 1-adrenoceptor subtypes in dog mesenteric and carotid arteries and rabbit carotid arteries. Br. J. Pharmacol. 102:1991;210-214.
32. 1-adrenoceptors in vascular smooth muscle. Br. J. Pharmacol. 99:1990;197-201.
33. 1-adrenoceptors involved in noradrenaline-induced contractions of rat thoracic aorta and dog carotid artery. Jpn. J. Pharmacol. 57:1991;535-544.
34. 1-adrenoceptor subtypes in the dog prostate. Urol. Res. 21:1993;211-215.
35. Piascik M.T., Guarino R.D., Smith M.S., Soltis E.E., Saussy D.L. Jr., Perez D.M. The specific contribution of the novel alpha-1D adrenoceptor to the contraction of vascular smooth muscle. J. Pharmacol. Exp. Ther. 275:1995;1583-1589.
36. 1-adrenoceptor subtypes and noradrenaline-induced contraction in rat portal vein smooth muscle. Br. J. Pharmacol. 110:1993;207-212.
37. 1-adrenoceptor subtypes in prostate and prostatic urethra of rat, rabbit, dog and man. Eur. J. Pharmacol. 249:1993;307-315.
38. Wein A.J. Practical uropharmacology. Urol. Clin. North Am. 18:1991;269-281.
39. Yoshida M., Latifpour J., Nishimoto T., Weiss R.M. Pharmacological characterization of alpha adrenergic receptors in the young and old female rabbit urethra. J. Pharmacol. Exp. Ther. 257:1991;1100-1108.