Relative efficacies of 6-opioid receptor agonists at the cloned human δ-opioid receptor

European Journal of Pharmacology

Volumn 326, Issue 1, 1997, Pages 101-104

  Quock, Raymond M ^a,e   Hosohata, Yoshiaki ^a   Knapp, Richard J ^a,f   Burkey, Thomas H ^a   Hosohata, Keiko ^a   Zhang, Xiaoyan ^b   Rice, Kenner C ^b   Nagase, Hiroshi ^c   Hruby, Victor J ^a   Porreca, Frank ^a   Roeske, William R ^a   Yamamura, Henry I ^a,d  

^a UNIVERSITY OF ARIZONA   (United States)

^b NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

^c TORAY INDUSTRIES INC   (Japan)

^d UNIVERSITY OF ARIZONA   (United States)

^e UNIVERSITY OF ILLINOIS   (United States)

^f Cortex Pharmaceuticals ^*  (United States)

Author keywords

Efficacy; Radioligand binding; 35S GTP S binding; Opioid receptor agonist; Opioid receptor, human

Indexed keywords

1,2,3,4,4A,5,12,12AALPHA OCTAHYDRO 4AALPHA (3 HYDROXYPHENYL) 2 METHYLQUINOLINO[2,3 G]ISOQUINOLINE; 4 [ALPHA (4 ALLYL 2,5 DIMETHYL 1 PIPERAZINYL) 3 METHOXYBENZYL] N,N DIETHYLBENZAMIDE; DELTA OPIATE RECEPTOR; ENKEPHALIN DERIVATIVE; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); NALTRINDOLE; OPIATE AGONIST; UNCLASSIFIED DRUG; 4 (ALPHA (4 ALLYL 2,5 DIMETHYL 1 PIPERAZINYL) 3 METHOXYBENZYL) N,N DIETHYLBENZAMIDE; 4-(ALPHA-(4-ALLYL-2,5-DIMETHYL-1-PIPERAZINYL)-3-METHOXYBENZYL)-N,N-DIETHYLBENZAMIDE; BENZAMIDE DERIVATIVE; DIAGNOSTIC AGENT; DRUG DERIVATIVE; ENKEPHALIN; ENKEPHALIN[2,5 DEXTRO PENICILLAMINE]; NALTREXONE; NARCOTIC ANTAGONIST; PIPERAZINE DERIVATIVE; QUINOLINE DERIVATIVE; SULFUR;

ANIMAL CELL; ARTICLE; CHO CELL; CONTROLLED STUDY; DRUG RECEPTOR BINDING; GENE EXPRESSION; HUMAN; IN VITRO STUDY; MOLECULAR CLONING; PRIORITY JOURNAL; ANIMAL; DRUG POTENTIATION; HAMSTER; METABOLISM;

ANIMALS; BENZAMIDES; CHO CELLS; CLONING, MOLECULAR; CRICETINAE; ENKEPHALIN, D-PENICILLAMINE (2,5)-; ENKEPHALINS; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); HUMANS; NALTREXONE; NARCOTIC ANTAGONISTS; PIPERAZINES; QUINOLINES; RECEPTORS, OPIOID, DELTA; SULFUR RADIOISOTOPES;

EID: 0030610216     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(97)83488-7     Document Type: Article

References (13)

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