Characterization of des-Arg9-bradykinin-induced contraction in guinea-pig gallbladder in vitro

European Journal of Pharmacology

Volumn 331, Issue 1, 1997, Pages 31-38

  Cabrini, Daniela A ^a   Calixto, João B ^a  

^a FEDERAL UNIVERSITY OF SANTA CATARINA   (Brazil)

Author keywords

Bradykinin B1 receptor selective antagonist; Bradykinin B2 receptor selective antagonist; Ca2+; Des Arg9 bradykinin; Gallbladder, guinea pig; Prostanoid

Indexed keywords

3 [1 (4 CHLOROBENZYL) 5 FLUORO 3 METHYL 2 INDOLYL] 2,2 DIMETHYLPROPIONIC ACID; BRADYKININ DERIVATIVE; BRADYKININ RECEPTOR; BRADYKININ[1-8]; CYCLOHEXIMIDE; DAZOXIBEN; EGTAZIC ACID; ESCHERICHIA COLI ENDOTOXIN; IBUPROFEN; ICATIBANT; INDOMETACIN; NICARDIPINE; NPC 17731; NPC 17761; PHENIDONE; RECEPTOR SUBTYPE; STAUROSPORINE; UNCLASSIFIED DRUG; VERLUKAST; BRADYKININ; BRADYKININ B1 RECEPTOR; BRADYKININ B2 RECEPTOR; BRADYKININ, DES ARG(9); BRADYKININ, DES-ARG(9)-; CALCIUM; DRUG DERIVATIVE; OLIGOPEPTIDE; PROSTAGLANDIN; PROTEIN KINASE C;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BLADDER CONTRACTION; CONTROLLED STUDY; FEMALE; GALLBLADDER; GUINEA PIG; IN VITRO STUDY; MALE; NONHUMAN; PRIORITY JOURNAL; ANIMAL; DOSE RESPONSE; DRUG ANTAGONISM; DRUG EFFECT; METABOLISM; MUSCLE CONTRACTION; PHYSIOLOGY; SMOOTH MUSCLE;

ANIMALS; BRADYKININ; CALCIUM; DOSE-RESPONSE RELATIONSHIP, DRUG; GALLBLADDER; GUINEA PIGS; MUSCLE CONTRACTION; MUSCLE, SMOOTH; OLIGOPEPTIDES; PROSTAGLANDINS; PROTEIN KINASE C; RECEPTOR, BRADYKININ B1; RECEPTOR, BRADYKININ B2; RECEPTORS, BRADYKININ;

EID: 0030610175     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(97)01010-8     Document Type: Article

References (24)

1. Altinkurt, O., Ozturk, Y., 1990. Bradykinin receptors in isolated rat duodenum. Peptides 11, 39-44.
2. 1 receptors in isolated rabbit aorta by using metabolic inhibitors. Eur. J. Pharmacol. 271, 551-555.
3. 9-bradykinin with isolated pig coronary arteries: Mechanical and electrophysiological events. Regul. Pept. 17, 181-190.
4. Bhoola, K.D., Figueroa, C.D., Worthy, K., 1992. Bioregulation of kinins, kallikreins, kininogens and kininases. Pharmacol. Rev. 44, 1-80.
5. 9-bradykinin in vitro and in vivo. Br. J. Pharmacol. 92, 257-264.
6. Burch, R.M., Kyle, D.J., Stormenn, T.M., 1993. Transduction of bradykinin signals. In: Burch, R.M., Austin, R.G. (Eds.), Molecular Biology and Pharmacology of Bradykinin Receptors. Landes, Austin, TX, pp. 33-52.
7. Cabrini, D.A., Silva, A.M., Calixto, J.B., 1995. Mechanisms of bradykinin-induced contraction of the guinea-pig gallbladder in vitro. Br. J. Pharmacol. 114, 1549-1556.
8. Cabrini, D.A., Kyle, D.J., Calixto, J.B., 1996. A pharmacological analysis of receptor subtypes and the mechanisms mediating the biphasic response induced by kinins in the rat stomach fundus in vitro. J. Pharmacol. Exp. Ther. 277, 299-307.
9. 2 receptors. J. Pharmacol. Exp. Ther. 268, 902-909.
10. 2 receptors in bradykinin-induced rat paw oedema. Br. J. Pharmacol. 113, 1005-1013.
11. 9-bradykinin-induced rat paw oedema by systemic treatment with bacterial endotoxin. Br. J. Pharmacol. 117, 793-798.
12. Hall, J.M., 1992. Bradykinin receptors: Pharmacological properties and biological roles. Pharmacol. Ther. 56, 131-190.
13. Hess, J.F., Borkowski, J.A., Young, G.S., Strader, C.D., Ransom, R.W., 1992. Cloning and pharmacological characterization of a human bradykinin (BK-2) receptor. Biochem. Biophys. Res. Commun. 184, 260-268.
14. Hess, J.F., Borkowiski, J.A., Macneil, T., Stonesifer, G.Y., Fraher, J., Strader, C.D., 1994. Differential pharmacology of cloned human and mouse b, bradykinin receptors. Mol. Pharmacol. 45, 1-8.
15. 2 receptor agonists synergistically potentiate interleukin-1 -induced prostaglandin biosynthesis in human gingivalfibroblasts. Inflammation 15, 427-436.
16. 1 receptors: A review. Immunopharmacology 30, 1-26.
17. 2 receptor. Proc. Natl. Acad. Sci. USA 88, 7724-7728.
18. 2 pharmacological sensitivity. Mol. Pharmacol. 44, 346-355.
19. 1 receptor gene. Biochem. Biophys. Res. Commun. 220, 219-223.
20. Regoli, D., Barabé, J., 1980. Pharmacology of bradykinin and related kinins. Pharmacol. Rev. 32, 1-12.
21. Regoli, D., Marceau, F., Barabé, J., 1978. De novo formation of vascular receptors for bradykinin. Can. J. Physiol. Pharmacol. 56, 674-677.
22. 9-bradykinin and bradykinin. J. Pharmacol. Exp. Ther. 264, 930-937.
23. Van Rossum, J.M., 1963. Cumulative dose-response curves. II. Techniques for making dose-response curves in isolated organs and the evaluation of drug parameters. Arch. Int. Pharmacodyn. Ther. 143, 299-330.
24. 2 kinin receptors in cultured bovine aortic endothelial cells. J. Pharmacol. Exp. Ther. 262, 729-733.