-
2
-
-
0011476882
-
-
Niedle, S. and Waring, M. J. Eds.; Verlag Chemie: Weinheim
-
b) Denny, W. A.; Baguley, B. C.; Cain, B. F.; Waring, M. J. Molecular Aspects of Anticacer Drug Action; Niedle, S. and Waring, M. J. Eds.; Verlag Chemie: Weinheim, 1983; pp. 1-34.
-
(1983)
Molecular Aspects of Anticacer Drug Action
, pp. 1-34
-
-
Denny, W.A.1
Baguley, B.C.2
Cain, B.F.3
Waring, M.J.4
-
3
-
-
0025274372
-
-
2. a) Deny, W. A.; Atwell, G. J.; Anderson, R. F; Wilson, W. R. J. Med. Chem. 1990, 33, 1288.
-
(1990)
J. Med. Chem.
, vol.33
, pp. 1288
-
-
Deny, W.A.1
Atwell, G.J.2
Anderson, R.F.3
Wilson, W.R.4
-
4
-
-
0023222336
-
-
b) Wakelin, L. P. G.; Atwell, G. J.; Rewcastle, G. W.; Denny, W. A. J. Med. Chem. 1987, 30, 855.
-
(1987)
J. Med. Chem.
, vol.30
, pp. 855
-
-
Wakelin, L.P.G.1
Atwell, G.J.2
Rewcastle, G.W.3
Denny, W.A.4
-
5
-
-
0021678126
-
-
c) Atwell, G. J.; Cain, B. F.; Baguley, B. C.; Finlay, G. F.; Denny, W. A. J. Med. Chem. 1984, 27, 1481.
-
(1984)
J. Med. Chem.
, vol.27
, pp. 1481
-
-
Atwell, G.J.1
Cain, B.F.2
Baguley, B.C.3
Finlay, G.F.4
Denny, W.A.5
-
7
-
-
0012049299
-
-
d) Capps, D. B. European Patent Appl. EP 145,226, 1985. (Chem. Abstr. 1985, 103, 2151825.
-
(1985)
Chem. Abstr.
, vol.103
, pp. 2151825
-
-
-
8
-
-
0028917629
-
-
e) Kimura, M.; Okabayashi, I.; Inone, H. J. Heterocycl. Chem. 1995, 32, 265.
-
(1995)
J. Heterocycl. Chem.
, vol.32
, pp. 265
-
-
Kimura, M.1
Okabayashi, I.2
Inone, H.3
-
10
-
-
0020033516
-
-
b) Deny, W. A.; Cain, B. F.; Atwell, G. J.; Hansch, C.; Panthanamickal, A.; Leo, A. J. Med. Chem. 1982, 25, 276.
-
(1982)
J. Med. Chem.
, vol.25
, pp. 276
-
-
Deny, W.A.1
Cain, B.F.2
Atwell, G.J.3
Hansch, C.4
Panthanamickal, A.5
Leo, A.6
-
11
-
-
0021165002
-
-
c) Baguley, B. C.; Denny, W. A.; Atwell, G. J.; Finlay, G. F.; Rewcastle, G. W.; Twidgen, S. J.; Wilson W. R. Cancer Res. 1984, 44, 3245.
-
(1984)
Cancer Res.
, vol.44
, pp. 3245
-
-
Baguley, B.C.1
Denny, W.A.2
Atwell, G.J.3
Finlay, G.F.4
Rewcastle, G.W.5
Twidgen, S.J.6
Wilson, W.R.7
-
12
-
-
0013910108
-
-
d) Goldin, A.; Serpick, A. A.; Mantel, N. Cancer Chemother. Rep. 1966, 50, 173.
-
(1966)
Cancer Chemother. Rep.
, vol.50
, pp. 173
-
-
Goldin, A.1
Serpick, A.A.2
Mantel, N.3
-
13
-
-
0015350296
-
-
e) Atwell, G. J.; Cain, B. F.; Seeley, R. N. J. Med. Chem. 1972, 15, 611.
-
(1972)
J. Med. Chem.
, vol.15
, pp. 611
-
-
Atwell, G.J.1
Cain, B.F.2
Seeley, R.N.3
-
15
-
-
0021333644
-
-
g) Nelson, E. M.; Tewey, K. M.; Lin, L. F. Proc. Natl. Acad. Sci. U.S.A. 1984, 81, 1361.
-
(1984)
Proc. Natl. Acad. Sci. U.S.A.
, vol.81
, pp. 1361
-
-
Nelson, E.M.1
Tewey, K.M.2
Lin, L.F.3
-
21
-
-
0001234289
-
-
c) Schmitz, F. J.; Agarwal, S. K.; Gunasekera, S. P.; Schmidt, P. G.; Shoolery, J. N. J. Am. Chem. Soc. 1983, 105, 4835.
-
(1983)
J. Am. Chem. Soc.
, vol.105
, pp. 4835
-
-
Schmitz, F.J.1
Agarwal, S.K.2
Gunasekera, S.P.3
Schmidt, P.G.4
Shoolery, J.N.5
-
22
-
-
0024428281
-
-
d) Charyulu, G. A.; McKee, T. Z.; Ireland, C. M. Tetrahedron Lett. 1989, 30, 4201.
-
(1989)
Tetrahedron Lett.
, vol.30
, pp. 4201
-
-
Charyulu, G.A.1
McKee, T.Z.2
Ireland, C.M.3
-
23
-
-
0023937279
-
-
e) Kobayashi, J.; Cheng, J.-F.; Wälchi, M. R.; Nakamura, H.; Hirata, Y.; Sasaki, T.; Ohizumi, Y. J. Org. Chem. 1988, 53, 1800.
-
(1988)
J. Org. Chem.
, vol.53
, pp. 1800
-
-
Kobayashi, J.1
Cheng, J.-F.2
Wälchi, M.R.3
Nakamura, H.4
Hirata, Y.5
Sasaki, T.6
Ohizumi, Y.7
-
25
-
-
0000152808
-
-
g) Carroll, A. R.; Cooray, N. M.; Poiner, A.; Schener, J. P. J. Org. Chem. 1989, 54, 4231.
-
(1989)
J. Org. Chem.
, vol.54
, pp. 4231
-
-
Carroll, A.R.1
Cooray, N.M.2
Poiner, A.3
Schener, J.P.4
-
27
-
-
0025971350
-
-
i) Schmitz, F. J.; DeGuzman, F. S.; Hossain, M. B.; Van der Helm, D. J. Org. Chem. 1991, 56, 804.
-
(1991)
J. Org. Chem.
, vol.56
, pp. 804
-
-
Schmitz, F.J.1
DeGuzman, F.S.2
Hossain, M.B.3
Van Der Helm, D.4
-
28
-
-
0023905863
-
-
j) Kobayashi, J.; Cheng, J.-F.; Nakamura, H.; Ohimizu, Y.; Hirata, Y.; Sasaki, T.; Otha, T.; Nozoe, S. Tetrahedron Lett. 1988, 29, 1177.
-
(1988)
Tetrahedron Lett.
, vol.29
, pp. 1177
-
-
Kobayashi, J.1
Cheng, J.-F.2
Nakamura, H.3
Ohimizu, Y.4
Hirata, Y.5
Sasaki, T.6
Otha, T.7
Nozoe, S.8
-
29
-
-
0001625491
-
-
k) Cimino, G.; Crispino, A.; de Rosa, S.; de Stefano, S.; Gavagnin, M.; Sodano, G. Tetrahedron 1987, 43, 4023.
-
(1987)
Tetrahedron
, vol.43
, pp. 4023
-
-
Cimino, G.1
Crispino, A.2
De Rosa, S.3
De Stefano, S.4
Gavagnin, M.5
Sodano, G.6
-
34
-
-
0012015957
-
-
9. O'Callaghan, C. N.; Brian, T.; McMurry, H.; O'Brien, J. E. J. Chem. Soc. Perkin Trans 1 1995, 417.
-
(1995)
J. Chem. Soc. Perkin Trans 1
, pp. 417
-
-
O'Callaghan, C.N.1
Brian, T.2
McMurry, H.3
O'Brien, J.E.4
-
35
-
-
85084771057
-
-
10. Bengelmans, R.; Bois-Chonssy, M.; Chastanet, J.; Le Glenher, M.; Zhu, J. Heterocycles 1993, 36, 2723.
-
(1993)
Heterocycles
, vol.36
, pp. 2723
-
-
Bengelmans, R.1
Bois-Chonssy, M.2
Chastanet, J.3
Le Glenher, M.4
Zhu, J.5
-
36
-
-
0025816845
-
-
11. a) Alo, B. I.; Kandil, A.; Patil, P. A.; Sharp, M. J.; Siddiqui, M. A.; Smieckus, V.; Josephy, P. D. J. Org. Chem. 1991, 56, 3763.
-
(1991)
J. Org. Chem.
, vol.56
, pp. 3763
-
-
Alo, B.I.1
Kandil, A.2
Patil, P.A.3
Sharp, M.J.4
Siddiqui, M.A.5
Smieckus, V.6
Josephy, P.D.7
-
38
-
-
0026072682
-
-
Petrillo, G.; Novi, M.; Dell'Erba, C.; Tavani, C. Tetrahedron 1991, 47, 9297.
-
(1991)
Tetrahedron
, vol.47
, pp. 9297
-
-
Petrillo, G.1
Novi, M.2
Dell'Erba, C.3
Tavani, C.4
-
39
-
-
0012045739
-
-
d) Manthey, M. K.; Pyne, S. G.; Truscott, R. J. W. J. Org. Chem. 1990, 55, 4581.
-
(1990)
J. Org. Chem.
, vol.55
, pp. 4581
-
-
Manthey, M.K.1
Pyne, S.G.2
Truscott, R.J.W.3
-
41
-
-
0042717277
-
-
and references therein
-
12. a) Elnadgi, M. H.; Sherif, S. M.; Mohareb, R. M. Heterocycles 1987, 26, 497 and references therein,
-
(1987)
Heterocycles
, vol.26
, pp. 497
-
-
Elnadgi, M.H.1
Sherif, S.M.2
Mohareb, R.M.3
-
43
-
-
0001819012
-
Addition to the Cyano group to form heterocycles
-
Rappoport, Z. J. Ed.; Wiley and Sons: New York
-
c) Mayers, A. I.; Sircar, J. C. Addition to the Cyano Group to Form Heterocycles. In The Chemistry of the Cyano Group; Rappoport, Z. J. Ed.; Wiley and Sons: New York, 1970; p. 341.
-
(1970)
The Chemistry of the Cyano Group
, pp. 341
-
-
Mayers, A.I.1
Sircar, J.C.2
-
44
-
-
0004063060
-
Synthesis of fused heterocycles
-
Taylor E. C. Ed.; Jhon Wiley: New York
-
d) Ellis G. P. Synthesis of Fused Heterocycles. In The Chemistry of Heterocyclic Compounds; Vol 47, Taylor E. C. Ed.; Jhon Wiley: New York, 1992; p. 739.
-
(1992)
The Chemistry of Heterocyclic Compounds
, vol.47
, pp. 739
-
-
Ellis, G.P.1
-
48
-
-
0002740319
-
-
Taylor, E. C. Ed.; Wiley, Interscience: New York
-
14. Böhme, H.; Viehe, H. G. Advances in Organic Chemistry; Vol 9, Taylor, E. C. Ed.; Wiley, Interscience: New York, 1976; p.1.
-
(1976)
Advances in Organic Chemistry
, vol.9
, pp. 1
-
-
Böhme, H.1
Viehe, H.G.2
-
50
-
-
0012045741
-
Chemistry of Dichloromethyleniminium salts (Phosgeniminium salts)
-
Böhme, H.; Viehe, H. G., Eds.; John Wiley and Sons, Inc.: New York
-
16. a) Janousek, Z.; Viehe, H. G. Chemistry of Dichloromethyleniminium salts (Phosgeniminium salts). In Iminium Salts in Organic Chemistry Advances in Organic Chemistry, Vol 9, Part I, Böhme, H.; Viehe, H. G., Eds.; John Wiley and Sons, Inc.: New York, 1976; p. 343.
-
(1976)
Iminium Salts in Organic Chemistry Advances in Organic Chemistry
, vol.9
, Issue.PART I
, pp. 343
-
-
Janousek, Z.1
Viehe, H.G.2
-
51
-
-
0012017606
-
-
b) Guillot, N.; Viehe, H. G.; Tinault, B.; DeClerq, J. P. Tetrahedron 1990, 46, 3897.
-
(1990)
Tetrahedron
, vol.46
, pp. 3897
-
-
Guillot, N.1
Viehe, H.G.2
Tinault, B.3
DeClerq, J.P.4
-
57
-
-
84984195846
-
-
h) Kokel, B.; Lespagnol, C.; Viehe, H. G. Bull. Soc. Chim. Belg. 1980, 89, 651.
-
(1980)
Bull. Soc. Chim. Belg.
, vol.89
, pp. 651
-
-
Kokel, B.1
Lespagnol, C.2
Viehe, H.G.3
-
58
-
-
0012017464
-
-
i) Bitter, I.; Pete, B.; Hermecz, I.; Tóth, G.; Simon, K.; Czugler, M.; Mészáros, Z. Tetrahedron Lett. 1982, 23, 2891.
-
(1982)
Tetrahedron Lett.
, vol.23
, pp. 2891
-
-
Bitter, I.1
Pete, B.2
Hermecz, I.3
Tóth, G.4
Simon, K.5
Czugler, M.6
Mészáros, Z.7
-
62
-
-
0028997820
-
-
18. a) Quintela, J. M.; Peinador, C.; Moreira, M. J. Tetrahedron 1995, 51, 5901.
-
(1995)
Tetrahedron
, vol.51
, pp. 5901
-
-
Quintela, J.M.1
Peinador, C.2
Moreira, M.J.3
-
63
-
-
0012015822
-
-
b) Peinador, C.; Veiga, M. C.; Ojea, V.; Quintela, J. M. Heterocycles 1994, 38, 2065.
-
(1994)
Heterocycles
, vol.38
, pp. 2065
-
-
Peinador, C.1
Veiga, M.C.2
Ojea, V.3
Quintela, J.M.4
-
64
-
-
0030046594
-
-
c) Quintela, J. M.; Moreira, M. J.; Peinador, C. Tetrahedron 1996, 52, 3037.
-
(1996)
Tetrahedron
, vol.52
, pp. 3037
-
-
Quintela, J.M.1
Moreira, M.J.2
Peinador, C.3
-
65
-
-
0027055396
-
-
19. a) Peinador, C.; Ojea, V.; Quintela, J.M. J. Heterocycl. Chem. 1992, 29, 1693.
-
(1992)
J. Heterocycl. Chem.
, vol.29
, pp. 1693
-
-
Peinador, C.1
Ojea, V.2
Quintela, J.M.3
-
66
-
-
0028352223
-
-
b) Peinador, C.; Moreira, M. J.; Quintela, J. M. Tetrahedron 1994, 50, 6705.
-
(1994)
Quintela, J. M. Tetrahedron
, vol.50
, pp. 6705
-
-
Peinador, C.1
Moreira, M.J.2
-
67
-
-
0012078144
-
-
c) Peinador, C.; Veiga, M. C.; Ojea, V.; Quintela, J. M. Heterocycles 1995, 41, 37.
-
(1995)
Heterocycles
, vol.41
, pp. 37
-
-
Peinador, C.1
Veiga, M.C.2
Ojea, V.3
Quintela, J.M.4
-
68
-
-
0000893306
-
-
20. Alvarez-Insua, A. S.; Lora-Tamayo, M. ;Soto, J. L. J. Heterocycl. Chem. 1970, 7, 1305.
-
(1970)
J. Heterocycl. Chem.
, vol.7
, pp. 1305
-
-
Alvarez-Insua, A.S.1
Lora-Tamayo, M.2
Soto, J.L.3
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