메뉴 건너뛰기




Volumn 65, Issue 1, 1996, Pages 61-70

Structure-affinity studies of C-terminally modified analogs of neuropeptide Y led to a novel class of peptidic Y1 receptor antagonist

Author keywords

[No Author keywords available]

Indexed keywords

NEUROPEPTIDE Y; NEUROPEPTIDE Y DERIVATIVE; NEUROPEPTIDE Y RECEPTOR ANTAGONIST;

EID: 0030603862     PISSN: 01670115     EISSN: None     Source Type: Journal    
DOI: 10.1016/0167-0115(96)00073-0     Document Type: Article
Times cited : (21)

References (35)
  • 2
    • 0011918368 scopus 로고
    • Molecular structure of mammalian neuropeptide Y: Analysis by molecular cloning and computer-aided comparison with crystal structure of avian homologue
    • [2] Allen, J., Novotny, J., Martin, J. and Heinrich, G., Molecular structure of mammalian neuropeptide Y: analysis by molecular cloning and computer-aided comparison with crystal structure of avian homologue, Proc. Natl. Acad. Sci. USA, 84 (1987) 2532-2536.
    • (1987) Proc. Natl. Acad. Sci. USA , vol.84 , pp. 2532-2536
    • Allen, J.1    Novotny, J.2    Martin, J.3    Heinrich, G.4
  • 3
    • 0019944850 scopus 로고
    • Neuropeptide Y - A novel brain peptide with structural similarities to peptide YY and pancreatic polypeptide
    • [3] Tatemoto, K., Carlquist, M. and Mutt, V. Neuropeptide Y - A novel brain peptide with structural similarities to peptide YY and pancreatic polypeptide, Nature (Lond.), 296 (1982) 659-660.
    • (1982) Nature (Lond.) , vol.296 , pp. 659-660
    • Tatemoto, K.1    Carlquist, M.2    Mutt, V.3
  • 4
    • 0020419772 scopus 로고
    • Complete amino acid sequence of the brain peptide
    • [4] Tatemoto, K., Complete amino acid sequence of the brain peptide, Proc. Natl. Acad. Sci. USA. 79, (1982) 5485-5489.
    • (1982) Proc. Natl. Acad. Sci. USA , vol.79 , pp. 5485-5489
    • Tatemoto, K.1
  • 5
    • 0003080075 scopus 로고
    • Origin and actions of neuropeptide Y in the cardiovascular system
    • In W.F. Colmers and C. Wahlestedt (Eds.). Humana Press, Totowa, NJ
    • [5] Zukowska-Grojec, Z. and Wahlestedt C., Origin and actions of neuropeptide Y in the cardiovascular system. In W.F. Colmers and C. Wahlestedt (Eds.). The Biology of Neuropeptide Y and Related Peptides, Humana Press, Totowa, NJ, 1993, pp. 315-388.
    • (1993) The Biology of Neuropeptide Y and Related Peptides , pp. 315-388
    • Zukowska-Grojec, Z.1    Wahlestedt, C.2
  • 6
    • 0002168533 scopus 로고
    • Characterization of receptor types for neuropeptide Y and related peptides
    • In W.F. Colmers and C. Wahlestedt (Eds.), Humana Press, Totowa, NJ
    • [6] Grundemar, L., Sheikh, S.P. and Wahlestedt C., Characterization of receptor types for neuropeptide Y and related peptides. In W.F. Colmers and C. Wahlestedt (Eds.), The Biology of Neuropeptide Y and Related Peptides, Humana Press, Totowa, NJ, 1993, pp. 197-239.
    • (1993) The Biology of Neuropeptide Y and Related Peptides , pp. 197-239
    • Grundemar, L.1    Sheikh, S.P.2    Wahlestedt, C.3
  • 7
    • 0027512327 scopus 로고
    • Neuropeptide Y-related peptides and their receptors - Are the receptors potential therapeutic drug targets?
    • [7] Wahlestedt, C. and Reis, D.J., Neuropeptide Y-related peptides and their receptors - Are the receptors potential therapeutic drug targets? Annu. Rev. Pharmacol. Toxicol., 32 (1993) 309-318.
    • (1993) Annu. Rev. Pharmacol. Toxicol. , vol.32 , pp. 309-318
    • Wahlestedt, C.1    Reis, D.J.2
  • 8
    • 0028030717 scopus 로고
    • Effects of neuropeptide Y on the electrical properties of neurons
    • [8] Colmers, W.F. and Bleakman, D., Effects of neuropeptide Y on the electrical properties of neurons (review). Trends Neurosci., 17 (1994) 373-379.
    • (1994) Trends Neurosci. , vol.17 , pp. 373-379
    • Colmers, W.F.1    Bleakman, D.2
  • 9
    • 0022588106 scopus 로고
    • Evidence for different pre-and post-junctional receptors for neuropeptide Y and related peptides
    • [9] Wahlestedt, C., Yanaihara, N. and Håkanson, R., Evidence for different pre-and post-junctional receptors for neuropeptide Y and related peptides, Regul. Pept., 13 (1986) 307-318.
    • (1986) Regul. Pept. , vol.13 , pp. 307-318
    • Wahlestedt, C.1    Yanaihara, N.2    Håkanson, R.3
  • 11
    • 0025132297 scopus 로고
    • Molecular cloning of a novel G protein-coupled receptor that may belong to the neuropeptide receptor family
    • [11] Eva, C., Kemanen, K., Monyer, H., Seeburg, P. and Sprengel, R., Molecular cloning of a novel G protein-coupled receptor that may belong to the neuropeptide receptor family, FEBS Lett., 271 (1990) 80-84.
    • (1990) FEBS Lett. , vol.271 , pp. 80-84
    • Eva, C.1    Kemanen, K.2    Monyer, H.3    Seeburg, P.4    Sprengel, R.5
  • 12
  • 13
    • 0026711234 scopus 로고
    • Cloned human neuropeptide Y receptor couples to two different second messenger systems
    • [13] Herzog, H., Hort, Y., Ball, H.J., Hayes, G., Shine, J. and Selbie, L.A., Cloned human neuropeptide Y receptor couples to two different second messenger systems, Proc. Natl. Acad. Sci. USA, 89 (1992) 5794-5798.
    • (1992) Proc. Natl. Acad. Sci. USA , vol.89 , pp. 5794-5798
    • Herzog, H.1    Hort, Y.2    Ball, H.J.3    Hayes, G.4    Shine, J.5    Selbie, L.A.6
  • 15
    • 0025908658 scopus 로고
    • Receptors for neuropeptide Y: Multiple subtypes and multiple second messengers
    • [15] Michel, M.C., Receptors for neuropeptide Y: multiple subtypes and multiple second messengers, Trends Pharmacol. Sci., 12 (1991) 392-394.
    • (1991) Trends Pharmacol. Sci. , vol.12 , pp. 392-394
    • Michel, M.C.1
  • 16
    • 0000734566 scopus 로고
    • Peptidmimetika für Rezeptorliganden -Entdeckung, Entwicklung und medizinische Aspekte
    • [16] Giannis, A. and Kolter, T., Peptidmimetika für Rezeptorliganden -Entdeckung, Entwicklung und medizinische Aspekte, Angew. Chem., 105 (1993) 1303-1326.
    • (1993) Angew. Chem. , vol.105 , pp. 1303-1326
    • Giannis, A.1    Kolter, T.2
  • 19
    • 0026592837 scopus 로고
    • Characterisation of the binidng site of neuropeptide Y to the rabbit kidney receptor using multiple peptide synthesis
    • [19] Beck-Sickinger, A.G., Dürr. H., Hoffmann, E., Gaida, W. and Jung, G., Characterisation of the binidng site of neuropeptide Y to the rabbit kidney receptor using multiple peptide synthesis. Biochem. Soc. Trans., 20, (1993) 847-850.
    • (1993) Biochem. Soc. Trans., 20 , pp. 847-850
    • Beck-Sickinger, A.G.1    Dürr, H.2    Hoffmann, E.3    Gaida, W.4    Jung, G.5
  • 21
    • 0022996556 scopus 로고    scopus 로고
    • Phenylethylamide derivatives of the C-terminal tetrapeptide of gastrin. Potent inhibitors of gastrin-stimulated acid secretion
    • [21] Martinez, J., Rodriguez, M., Bali, J.-P. and Laur, J., Phenylethylamide derivatives of the C-terminal tetrapeptide of gastrin. Potent inhibitors of gastrin-stimulated acid secretion. Int. J. Pept. Protein Res., 28 (1996) 529-535.
    • (1996) Int. J. Pept. Protein Res. , vol.28 , pp. 529-535
    • Martinez, J.1    Rodriguez, M.2    Bali, J.-P.3    Laur, J.4
  • 23
    • 0020644532 scopus 로고
    • Cholecystokinin-27-32-amide. A member of a new class of cholecystokinin receptor antagonists
    • [23] Spanarkel, M., Martinez, J., Briet, C., Jensen, R.T. and Gardner, J.D., Cholecystokinin-27-32-amide. A member of a new class of cholecystokinin receptor antagonists, J. Biol. Chem., 258, (1983) 6746-6749.
    • (1983) J. Biol. Chem. , vol.258 , pp. 6746-6749
    • Spanarkel, M.1    Martinez, J.2    Briet, C.3    Jensen, R.T.4    Gardner, J.D.5
  • 25
    • 0017816363 scopus 로고
    • Studies on organophosphorus compounds XXI. The dimer of p-methoxyphenylthionophosphine sulfide as a thiation reagent. A new route to thiocarboxamides
    • [25] Scheibye, S., Petersen, B.S. and Lawesson, S.O., Studies on organophosphorus compounds XXI. The dimer of p-methoxyphenylthionophosphine sulfide as a thiation reagent. A new route to thiocarboxamides. Bull. Soc. Chim. Belg., 87 (1978) 229-238.
    • (1978) Bull. Soc. Chim. Belg. , vol.87 , pp. 229-238
    • Scheibye, S.1    Petersen, B.S.2    Lawesson, S.O.3
  • 26
    • 0021895138 scopus 로고
    • A new generation of calcium indicators with greatly improved fluorecence properties
    • [26] Grynkiewicz, G., Poenie, M. and Tsien, R.Y., A new generation of calcium indicators with greatly improved fluorecence properties, J. Biol. Chem., 260 (1985) 3440-3450.
    • (1985) J. Biol. Chem. , vol.260 , pp. 3440-3450
    • Grynkiewicz, G.1    Poenie, M.2    Tsien, R.Y.3
  • 28
    • 0025148350 scopus 로고
    • Neuropeptide Y (18-36) is a competitive antagonist of neuropeptide Y in rat cardiac ventricular membranes
    • [28] Balasubramaniam, A. and Sheriff, S., Neuropeptide Y (18-36) is a competitive antagonist of neuropeptide Y in rat cardiac ventricular membranes, J. Biol. Chem., 265 (1990) 14724-14727.
    • (1990) J. Biol. Chem. , vol.265 , pp. 14724-14727
    • Balasubramaniam, A.1    Sheriff, S.2
  • 29
    • 0027217002 scopus 로고
    • Molecular cloning, characterisation and localization of the human homolog to the reported bovine NPY Y3 receptor: Lack of NPY binding and activation
    • [29] Herzog, H., Hort, Y., Shine, J. and Selbie, L.A., Molecular cloning, characterisation and localization of the human homolog to the reported bovine NPY Y3 receptor: lack of NPY binding and activation. DNA Cell. Biol., 12 (1993) 465-471.
    • (1993) DNA Cell. Biol. , vol.12 , pp. 465-471
    • Herzog, H.1    Hort, Y.2    Shine, J.3    Selbie, L.A.4
  • 30
    • 0026557170 scopus 로고
    • Synthesis of receptor antagonists of neuropeptide Y
    • [30] Tatemoto, K., Mann, M.J. and Shimizu, M., Synthesis of receptor antagonists of neuropeptide Y. Proc. Natl. Acad. Sci. USA, 89 (1992) 1174-1178.
    • (1992) Proc. Natl. Acad. Sci. USA , vol.89 , pp. 1174-1178
    • Tatemoto, K.1    Mann, M.J.2    Shimizu, M.3
  • 32
    • 0025845031 scopus 로고
    • Blockade of neuropeptide Y -induced potentiation of noradrenaline-evoked vasoconstriction by D-myo-inositol 1,2,6-triphosphate (PP56) in rabbit femoral arteries
    • [32] Adamsson, M. and Edvinsson, L., Blockade of neuropeptide Y -induced potentiation of noradrenaline-evoked vasoconstriction by D-myo-inositol 1,2,6-triphosphate (PP56) in rabbit femoral arteries, Neuropeptides, 19 (1991) 13-16.
    • (1991) Neuropeptides , vol.19 , pp. 13-16
    • Adamsson, M.1    Edvinsson, L.2
  • 34
    • 0026508363 scopus 로고
    • Neuropeptide Y and its antagonists
    • [34] Michel, M.C. and Buschauer, A., Neuropeptide Y and its antagonists, Drugs Future, 17 (1992) 39-45.
    • (1992) Drugs Future , vol.17 , pp. 39-45
    • Michel, M.C.1    Buschauer, A.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.