Transdermal iontophoresis of sodium nonivamide acetate I. Consideration of electrical and chemical factors

International Journal of Pharmaceutics

Volumn 143, Issue 1, 1996, Pages 47-58

  Fang, Jia You ^a   Huang, Yaw Bin ^a   Wu, Pao Chu ^a   Tsai, Yi Hung ^a  

^a KAOHSIUNG MEDICAL UNIVERSITY   (Taiwan)

Author keywords

Iontophoresis; Sodium nonivamide acetate; Transdermal absorption

Indexed keywords

NONIVAMIDE;

ANIMAL TISSUE; ARTICLE; DIFFUSION; ELECTRIC FIELD; IONIC STRENGTH; IONTOPHORESIS; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; SKIN PENETRATION;

EID: 0030601839     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-5173(96)04681-9     Document Type: Article

References (43)

1. Bannon, Y.B., Corish, J., Corrigan O.I. and Masterson, J.G., Iontophoretically induced transdermal delivery of salbutamol. Drug Dev. Ind. Pharm., 14 (1988) 2151-2166.
2. Behl, C.R., Kumar, S., Malick, A.W., Del Terzo, S., Higuchi, W.I. and Nash, R.A., Iontophoretic drug delivery: effects of physicochemical factors on the skin uptake of nonpeptide drugs. J. Pharm. Sci., 78 (1989) 355-360.
3. Bellantone, N.H., Rim, S., Francoeur, M.L. and Rasadi, B., Enhanced percutaneous absorption via iontophoresis I. Evaluation of an in vitro system and transport of model compounds. Int. J. Pharm., 30 (1986) 63-72.
4. Bronaugh, R.L., Stewart, R.F. and Congdon, E.R., Methods for in vitro percutaneous absorption studies I. Animal models for human skin. Toxicol. Appl. Pharmacol., 62 (1982) 481-488.
5. Burnette, R.R. and Bagniefski, T.M., Influence of constant current iontophoresis on the impedence and passive Napermeability of excised nude mouse skin. J. Pharm. Sci., 11 (1988) 492-497.
6. Burnette, R.R. and Marrero, D., Comparison between the iontophoretic and passive transport of thyrotropin releasing hormone across excised nude mouse skin. J. Pharm. Sci., 75 (1986) 738-743.
7. Burnette, R.R. and Ongpipattanakul, B., Characterization of the permselective properties of excised human skin during iontophoresis. J. Pharm. Sci., 76 (1987) 765-773.
8. Chen, I.J., Yang, J.M., Yeh, J.L., Wu, B.N., Lo, Y.C. and Chen, S.J., Hypotensive and antinociceptive effects of ether-linked and relatively non-pungent analogues of N-nonanoyl vanillylamide. Eur. J. Med. Chem., 27 (1992) 187-192.
9. Chien, Y.W. and Banga, A.K., Iontophoretic (Transdermal) delivery of drugs: overview of historical development. J. Pharm. Sci., 78 (1989) 353-354.
10. Chien, Y.W., Siddiqui, O., Shi, W.M., Lelawongs, P. and Liu, J.C., Direct current iontophoretic transdermal delivery of peptide and protein drugs. J. Pharm. Sci., 78 (1989) 376-383.
11. Donnerer, J., Amann, R., Schuligoi, R. and Lembeck, F., Absorption and metabolism of capsaicinoids following intragastric administration in rats. Arch. Pharmacol., 342 (1990) 357-361.
12. Fang, J.Y., Wu, P.C., Huang Y.B. and Tsai, Y.H., In vitro permeation study of capsaicin and its synthetic derivatives from ointment bases using various skin types. Int. J. Pharm., 126 (1995) 119-128.
13. Fang, J.Y., Wu, P.C., Huang Y.B. and Tsai, Y.H., Percutaneous absorption of capsaicin, nonivamide and sodium nonivamide acetate from gel and ointment bases: in vitro formulation evaluations in pigs and in vivo bioengineering methods in humans. Int. J. Pharm. 130 (1996) 121-135.
14. Gangarosa, L.P., Park, N.H., Wiggins, C.A. and Hill, J.M., Increased penetration of nonelectrolytes into mouse skin during iontophoretic water transport (iontohydrokinesis). J. Pharmacol Exp. Ther., 212 (1980) 377-381.
15. Green, P.G., Hinz, R.S., Cullander, C., Yamane, G. and Guy, R.H., Iontophoretic delivery of amino acids and amino acid derivatives across the skin in vitro. Pharm. Res., 8 (1991) 1113-1120.
16. Higuchi, W.I., Diffusional models useful in biopharmaceutics. J. Pharm. Sci., 51 (1962) 802-804.
17. Illel, B., Schaefer, H., Wepierre. J. and Doucet, O., Follicles play an important role in percutaneous absorption. J. Pharm. Sci., 80 (1991) 424-427.
18. Kasting, G.B. and Bowman, L.A., DC electrical properties of frozen, excised human skin. Pharm. Res., 1 (1990) 134-143.
19. Kasting, G.B., Merrit, E.W. and Keister, J.C., An in vitro method for studying the iontophoretic enhancement of drug transport through the skin. J. Membr. Sci., 35 (1988) 137-159.
20. Koizumi, T., Kakemi, M., Katayama, K., Inada, H., Sudeji, K. and Kawasaki, M., Transfer of diclofenac sodium across excised guinea pig skin on high-frequency pulse iontophoresis. I. equivalent circuit model., Chem. Pharm. Bull., 38 (1990) 1019-1021.
21. Lashmar, U.T. and Manger, J., Investigation into the potential for iontophoresis facilitated transdermal delivery of acyclovir. Int. J. Pharm., 111 (1994) 73-82.
22. Lelawongs, P., Liu, J.C. and Chien, Y.W., Transdermal iontophoretic delivery (II): Evaluation of electrical and operational factors. Int. J. Pharm., 61 (1990) 179-188.
23. Lelawongs, P., Liu, J.C., Siddiqui, O. and Chien, Y.W., Transdermal iontophoretic delivery of arginine-vasopressin (I): Physicochemical considerations. Int. J. Pharm., 56 (1989) 13-22.
24. Li, L.C., Vu, N.T. and Allen, L.V., Iontophoretic permeation of sodium cromoglycate through synthetic membrane and excised hairless mouse skin. J. Pharm. Pharmacol., 44 (1992) 444-446.
25. Masada, T., Higuchi, W.I., Srinivasan, V., Rohr, U., Fox, J., Behl, C. and Pons, S., Examination of iontophoretic transport of ionic drugs across skin: baseline studies with the four-electrode system. Int. J. Pharm., 49 (1989) 57-62.
26. Miller, L.L. and Smith, G.A., Iontophoretic transport of acetate and carboxylate ions through hairless mouse skin. A cation exchange membrane model. Int. J. Pharm., 49 (1989) 15-22.
27. Nakhare, S., Jain, N.K. and Verma, H.V., Iontophoretic cellophane membrane delivery of diclofenac sodium. Pharmazie., 49 (1994) 672-675.
28. Padmanabhan, R.V., Phipps, J.B. and Lattin, G.A., In vitro and in vivo evaluation of transdermal iontophoretic delivery of hydromorphone. J. Controlled Release, 11 (1990) 123-135.
29. Phipps, J.B., Padmanabhan, R.V. and Lattin, G.A., Iontophoretic delivery of model inorganic and drug ions. J. Pharm. Sci., 78 (1989) 365-369.
30. Santi, P., Catellani, P.L., Massimo, G., Zanardi, G. and Colombo, P., Iontophoretic transport of verapamil and melatonin I. cellophane membrane as a barrier. Int. J. Pharm., 92 (1993) 23-28.
31. Schade, H. and Marchionini, A., Uber die azidose aut der normalen haut und ihre bedeutung zur abwehr der bakterien. Munchen. Med. Wchnschr., 74 (1927) 1435-1436.
32. Siddiqui, O., Roberts, M.S. and Polack, A., The effect of iontophoresis and vehicle pH on the in-vitro permeation of lignocaine through human stratum corneum. J. Pharm. Pharmacol., 37 (1985) 732-735.
33. Sietsema, K., Berman, F., Farmer, W. and Maddin, S., The antinociceptive effect and pharmacokinetics of olvanil following oral and subcutaneous dosing in the mouse. Life Sci., 43 (1988) 1385-1391.
34. Sims, S.M., Higuchi, W.I. and Srinivasan, V., Interaction of electric field and electro-osmotic effects in determining iontophoretic enhancement of anions and cations. Int. J. Pharm., 69 (1991) 109-121.
35. Singh, P., Anliker, M., Smith, G.A., Zavortink, D. and Maibach, H.I., Transdermal iontophoresis and solute penetration across excised human skin. J. Pharm. Sci., 84 (1995) 1342-1346.
36. Singh, P. and Maibach, H.I., Transdermal iontophoresis. Pharmacokinetic considerations. Clin. Pharmacokinet., 26 (1994) 327-334.
37. Thysman, S., Tasset, C. and Preat, V., Transdermal iontophoresis of fentanyl: delivery and mechanistic analysis. Int. J. Pharm., 101 (1994) 105-113.
38. Tsai, Y.H., Huang, Y.B., Fang, J.Y. and Wu, P.C., Percutaneous absorption of capsaicin and its derivatives. Drug Dev. Ind. Pharm., 20 (1994) 719-730.
39. Tyle, P., Iontophoretic devices for drug delivery. Pharm. Res., 3 (1986) 318-326.
40. Wearley, L. and Chien, Y.W., Enhancement of the in vitro skin permeability of azidothymidine (AZT) via iontophoresis and chemical enhancer. Pharm. Res., 7 (1990) 34-40.
41. Wearley, L., Liu, J.C. and Chien, Y.W., Iontophoresis facilitated transdermal delivery of verapamil I. In vitro evaluation and mechanistic studies. J. Controlled Release, 8 (1989) 237-250.
42. Williams, A.C. and Barry, B.W., Skin absorption enhancers. Crit. Rev. Ther. Drug Carrier Syst., 9 (1992) 305-353.
43. Yang, J.M., Wu, B.N. and Chen, I.J., Depressor response of sodium nonivamide acetate: a newly synthesized nonpungent analogue of capsaicin. Asia Pac. J. Pharmacol., 7 (1992) 95-102.