New heteroaryl-spaced phosphono α-amino acids are competitive NMDA antagonists with analgesic activity

Bioorganic and Medicinal Chemistry Letters

Volumn 6, Issue 14, 1996, Pages 1635-1640

  Swahn, Britt Marie ^a   Claesson, Alf ^a   Pelcman, Benjamin ^a   Besidski, Yevgeni ^a   Molin, Håkan ^a   Sandberg, Mats P ^a   Berge, Odd Geir ^a  

^a ASTRAZENECA R AND D   (Sweden)

Author keywords

[No Author keywords available]

Indexed keywords

LAS 333; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; N METHYL DEXTRO ASPARTIC ACID RECEPTOR BLOCKING AGENT; PHOSPHONOAMINO ACID; UNCLASSIFIED DRUG;

ANALGESIA; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; MOUSE; NONHUMAN; ORAL DRUG ADMINISTRATION; QUANTITATIVE STRUCTURE ACTIVITY RELATION; RAT; SWINE;

ANIMALIA; SUS SCROFA;

EID: 0030598670     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0960-894X(96)00288-0     Document Type: Article

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