[Cys(O2NH2)2]enkephalin analogues and dalargin: Selectivity for δ-opioid receptors

European Journal of Pharmacology

Volumn 304, Issue 1-3, 1996, Pages 99-108

  Pencheva, Nevena ^a   Bocheva, Adriana ^a   Dimitrov, Emil ^a   Ivancheva, Christina ^a   Radomirov, Radomir ^a  

^a INSTITUTE OF PHYSIOLOGY   (Bulgaria)

Author keywords

adrenergic component; cysteine sulfonamide enkephalin analog; dalargin; electrical field stimulation; purinergic component; vas deferens, mouse; opioid receptor

Indexed keywords

ADENOSINE TRIPHOSPHATE; ALPHA,BETA METHYLENEADENOSINE TRIPHOSPHATE; BACITRACIN; DELTA OPIATE RECEPTOR; ENKEPHALIN DERIVATIVE; KAPPA OPIATE RECEPTOR; LEUCINE ENKEPHALIN; LEUCINE ENKEPHALIN[2 DEXTRO ALANINE 6 ARGININE]; METENKEPHALIN; MU OPIATE RECEPTOR; NALOXONE; NORADRENALIN; OPIATE AGONIST; POSTSYNAPTIC RECEPTOR; PRAZOSIN; RECEPTOR SUBTYPE; TETRODOTOXIN; DRUG DERIVATIVE; ENKEPHALIN; ENKEPHALIN LEU, ALA(2) ARG(6); ENKEPHALIN LEU, CYS(O2NH2)(2); ENKEPHALIN MET, CYS(O2NH2)(2); ENKEPHALIN-LEU, ALA(2)-ARG(6)-; ENKEPHALIN-LEU, CYS(O2NH2)(2)-; ENKEPHALIN-MET, CYS(O2NH2)(2)-; ENKEPHALIN[2 ALANINE 5 LEUCINE];

ADRENERGIC NERVE; ANIMAL TISSUE; ARTICLE; AUTONOMIC NERVE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG POTENCY; DRUG SELECTIVITY; ELECTROSTIMULATION; GUINEA PIG; ILEUM; MALE; MOUSE; NONHUMAN; PRIORITY JOURNAL; SMOOTH MUSCLE CONTRACTILITY; STRUCTURE ACTIVITY RELATION; VAS DEFERENS; ANIMAL; COMPARATIVE STUDY; DOSE RESPONSE; DRUG EFFECT; IN VITRO STUDY; MUSCLE CONTRACTION; SMOOTH MUSCLE;

ADENOSINE TRIPHOSPHATE; ANIMALS; DOSE-RESPONSE RELATIONSHIP, DRUG; ELECTRIC STIMULATION; ENKEPHALIN, LEUCINE; ENKEPHALIN, LEUCINE-2-ALANINE; ENKEPHALIN, METHIONINE; ENKEPHALINS; GUINEA PIGS; ILEUM; MALE; MICE; MUSCLE CONTRACTION; MUSCLE, SMOOTH; NOREPINEPHRINE; RECEPTORS, OPIOID, DELTA; RECEPTORS, OPIOID, KAPPA; STRUCTURE-ACTIVITY RELATIONSHIP; VAS DEFERENS;

EID: 0030598577     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/0014-2999(96)00083-0     Document Type: Article

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