Lipophilic bioisosteres of nucleoside triphosphates

Bioorganic and Medicinal Chemistry Letters

Volumn 6, Issue 20, 1996, Pages 2411-2416

  Goldring, Alastair O ^a   Gilbert, Ian H ^a   Mahmood, Naheed ^b   Balzarini, Jan ^c  

^a CARDIFF UNIVERSITY   (United Kingdom)

^b MEDICAL RESEARCH COUNCIL   (United Kingdom)

^c REGA INSTITUTE FOR MEDICAL RESEARCH   (Belgium)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIVIRUS AGENT; NUCLEOSIDE DERIVATIVE; RNA DIRECTED DNA POLYMERASE; STAVUDINE; ZIDOVUDINE;

ANTIVIRAL ACTIVITY; ARTICLE; CELL LINE; CONTROLLED STUDY; DRUG DESIGN; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS 1; HUMAN IMMUNODEFICIENCY VIRUS 2; STEREOCHEMISTRY;

HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 1; HUMAN IMMUNODEFICIENCY VIRUS 2;

EID: 0030598171     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0960-894X(96)00443-X     Document Type: Article

References (11)

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2. 1. Balzarini, J.; Herdewijn, P.; De Clercq, E., J. Biol. Chem., 1989, 264, 6127. Gao, W.-Y.; Agbaria, R.; Driscoll, J. S.; Mitsuya, H., J. Biol. Chem., 1994, 269, 12633.
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6. 5. Otoski, R. M.; Wilcox, C. S., Tetrahedron Letts., 1988, 29, 2615.
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8. 7. Acknowledgement to C. S. Wilcox for supplying experimental details.
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11. 10. Weaver, R.; Gilbert, I. H.; Mahmood, N., manuscript in preparation.