N-peptidyl, O-acyl hydroxamates: Comparison of the selective inhibition of serine and cysteine proteinases

Biochimica et Biophysica Acta - Protein Structure and Molecular Enzymology

Volumn 1295, Issue 2, 1996, Pages 179-186

  Demuth, Hans Ulrich ^a   Schierhorn, Angelika ^a   Bryan, Philip ^b   Höfke, Ralph ^a   Kirschke, Heidrun ^a   Brömme, Dieter ^a  

^a MARTIN LUTHER UNIVERSITY HALLE WITTENBERG   (Germany)

^b UNIVERSITY OF MARYLAND BIOTECHNOLOGY INSTITUTE   (United States)

Author keywords

Cysteine proteinase; Hydroxamate; Inhibitor; Mechanism; Serine proteinase

Indexed keywords

CYSTEINE PROTEINASE; CYSTEINE PROTEINASE INHIBITOR; ENZYME INHIBITOR; HYDROXAMIC ACID DERIVATIVE; SERINE PROTEINASE; SERINE PROTEINASE INHIBITOR;

ARTICLE; CHEMICAL MODIFICATION; DRUG DECOMPOSITION; DRUG STABILITY; DRUG SYNTHESIS; ENZYME INHIBITION; ENZYME KINETICS; PRIORITY JOURNAL;

EID: 0030592186     PISSN: 01674838     EISSN: None     Source Type: Journal    
DOI: 10.1016/0167-4838(96)00038-6     Document Type: Article

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