SAR of 2-benzyl-4-aminopiperidines NK1 antagonists. Part 2. Synthesis of CGP 49823

Bioorganic and Medicinal Chemistry Letters

Volumn 6, Issue 24, 1996, Pages 3029-3034

  Veenstra, Siem J ^a   Hauser, Kathleen ^a   Schilling, Walter ^a   Betschart, Claudia ^a   Ofner, Silvio ^a  

^a F HOFFMANN LA ROCHE LTD   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

2 BENZYL 1 (3,5 DIMETHYLBENZOYL) 4 (4 QUINOLINYLMETHYLAMINO)PIPERIDINE; NEUROKININ 1 RECEPTOR; NEUROKININ 1 RECEPTOR ANTAGONIST; PIPERIDINE DERIVATIVE; SUBSTANCE P; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CATTLE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; NONHUMAN; QUANTITATIVE STRUCTURE ACTIVITY RELATION; REACTION ANALYSIS; RETINA; STEREOCHEMISTRY; TECHNIQUE;

EID: 0030591843     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(96)00563-X     Document Type: Article

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