Selective deprotection of phthalyl protected amines

Tetrahedron Letters

Volumn 37, Issue 42, 1996, Pages 7469-7472

  Costello, Colleen A ^a   Kreuzman, Adam J ^a   Zmijewski, Milton J ^a  

^a ELI LILLY AND COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMINE;

ARTICLE; CHIRALITY; DRUG SYNTHESIS; ENZYME ACTIVITY; REACTION ANALYSIS; TECHNIQUE;

EID: 0030583466     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/0040-4039(96)01752-2     Document Type: Article

References (11)

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3. 3. Kukolja, S.; Lammert, S. R.; Ellis, A. I.; Croatica Chemica Acta 1977, 49, 779-795.
4. 4. Vu, H.; Joyce, N.; Rieger, M.; Walker, D.; Goldknopf, I.; Schmaltz-Hill, T.; Jayaraman, K.; Mulvey, D. Bioconjugate Chemistry 1995, 6, 599-607.
5. 5. Briggs, B. S.; Kreuzman, A. J.; Whitesitt, C.; Yeh, W-K; Zmijewski, M. J. J. Mol. Catalysis B: Enzymes 1996, 34, in press.
6. 6. Zock, J.; Kreuzman, A. J.; Queener, S. Gene 1996, manuscript in preparation.
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8. 7. Rudinger, J.; Krupica, J.; Zaoral, M.; Cernik, V. Collection Czechoslov. Chem. Commun. 1960, 25, 3338-3343. Yang, Y-S; Ramaswamy, S.; Jakoby, W. B. J. Biol. Chem. 1993, 268, 10870-10875.
9. 3CN.
10. 2: methylene chloride. Assays were monitored at spectrophotometrically at 380nm using 200μM 5 at 30°C.
11. 10. Bender, M. J.; Chow, Y-L; Chloupek, F. J. Amer. Chem. Soc. 1958, 80, 5380-5387.