Correlation of 'in vitro' release and 'in vivo' absorption characteristics of four salbutamol sulphate formulations

International Journal of Pharmaceutics

Volumn 139, Issue 1-2, 1996, Pages 45-52

  Hernandez R M ^a   Gascon A R ^a   Calvo, M B ^a   Caramella, C ^b   Conte, U ^b   Dominguez Gil A ^c   Pedraz, J L ^a  

^a UNIVERSITY OF THE BASQUE COUNTRY UPV EHU   (Spain)

^b UNIVERSITY OF PAVIA   (Italy)

^c UNIVERSITY OF SALAMANCA   (Spain)

Author keywords

'In vitro in vivo' correlation; Absorption, 'in vivo'; Release, 'in vitro'; Salbutamol

Indexed keywords

SALBUTAMOL; SALBUTAMOL SULFATE;

ANIMAL EXPERIMENT; AREA UNDER THE CURVE; ARTICLE; CONTROLLED STUDY; DISSOLUTION; DOG; DRUG ABSORPTION; DRUG BLOOD LEVEL; DRUG DOSAGE FORM; DRUG FORMULATION; DRUG RELEASE; INTRAVENOUS DRUG ADMINISTRATION; NONHUMAN; ORAL DRUG ADMINISTRATION; PHARMACOKINETICS; PRIORITY JOURNAL;

EID: 0030576620     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/0378-5173(96)04571-1     Document Type: Article

References (12)

1. Baveja, S.K., Ranga Rao, K.V. and Padmalatha Devi, K., Zero-order release hydrophilic matrix tablets of β-adrenergic blockers. Int. J. Pharm., 39 (1987) 39-45.
2. Bonferoni, M.C., Caramella, C., Sangalli, M.E., Conte, U., Hernández, R.M. and Pedraz, J.L., Rheological behaviour of hydrophilic polymers and drug release from erodible matrices. J. Control. Rel., 18 (1992) 205-212.
3. Blume, H.H., McGilveray, J.J. and Midha, K.K., Bio-International '94, Bioavailability, Bioequivalence and Pharmacokinetic Studies and Pre-Conference Satellite on 'In vitro In vivo Correlation. Eur. J. Drug Metabol. Pharmacokin., 20 (1995) 3-13.
4. ® program. Eur. J. Metab., 18 (1993) 5242-5246.
5. Gibaldi. M. and Perrier D., Noncompartmental analysis based on statistical moment theory. In Pharmacokinetics, M, Dekker, (Ed), New York. (1982), pp. 409-417.
6. Hernández, R.M., Gascón, A.R., Calvo. M.B., Bonferoni, M.C., Caramella, C., Sangalli, M.E., Conte, U. and Domínguez-Gil, A., Evaluatión biofarmacéutica de comprimidos de sulfato de salbutamol elaborados con hidroxipropilmetilcelulosa. Ind. Farm., 2 (1994) 39-44.
7. Hutchings, M.J., Paul. J.D. and Morgan, D.J., Determination of salbutamol in plasma by high performance liquid chromatography. J. Chromatogr. Biomed. Appl., 227 (1983) 423-426.
8. R. Geavanceerde berekening van biologische beschibaarheid en geneesmiddel absorptiesnelheis, Mediware, Groningen, 1991.
9. Mulholland, M. and Waterhouse. J., Investigation of the limitations of satured fractional factorial experimental designs, with confounding effects for an HPLC ruggedness test. Chromatographia. 25 (1988) 769-774.
10. Schumaker, B., PKCALC: A basis interactive computer program for statistical and pharmacokinetic analysis of data. Drug Metab. Rev., 17 (1986) 331-336.
11. Skelley, J.P., Amidon, G.L., Barr, W.J., Benet, L.Z., Carter, J.E., Robinson, J.R., Shah, V.P. and Yacobi, A., Report of the workshop on in-vitro and in-vivo testing and correlation for oral controlled/modified-release dosage forms. J. Pharm. Sci., 79 (1990) 849-854.
12. USP 23, US Pharmacopeial Convention. Inc, Rockville, 1995, pp. 1924-1929.