8-Amino-6-(arylsulphonyl)-5-nitroquinolines: Novel nonpeptide neuropeptide Y1 receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 6, Issue 15, 1996, Pages 1809-1814

  Wright, Jon ^a   Bolton, Gary ^a   Creswell, Mark ^a   Downing, Dennis ^a   Georgic, Lynn ^a   Heffner, Thomas ^a   Hodges, John ^a   MacKenzie, Robert ^a   Wise, Lawrence ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

NEUROPEPTIDE Y RECEPTOR; NEUROPEPTIDE Y1 RECEPTOR ANTAGONIST; PD 160170; PD 9262; QUINOLINE DERIVATIVE; RECEPTOR BLOCKING AGENT; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; HIPPOCAMPUS; NONHUMAN; RAT; STRUCTURE ACTIVITY RELATION;

ANIMALIA;

EID: 0030572489     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0960-894X(96)00319-8     Document Type: Article

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19. +, 100%).