Conformationally restricted 1,5-diarylpyrazoles are selective COX-2 inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 6, Issue 23, 1996, Pages 2827-2830

  Bertenshaw, Stephen R ^a   Talley, John J ^a   Rogier, D J ^a   Graneto, Matthew J ^a   Koboldt, Carol M ^a   Zhang, Yan ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ISOENZYME; NONSTEROID ANTIINFLAMMATORY AGENT; PROSTAGLANDIN SYNTHASE; PROSTAGLANDIN SYNTHASE INHIBITOR; PYRAZOLE DERIVATIVE; SULFONAMIDE; SULFONE;

ANIMAL MODEL; ANTIINFLAMMATORY ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; ENZYME INHIBITION; IN VITRO STUDY; NONHUMAN;

ANIMALIA;

EID: 0030568116     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(96)00530-6     Document Type: Article

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