Syntheses of stable bacteriochlorophyll-a derivatives as potential photosensitizers for photodynamic therapy

Tetrahedron Letters

Volumn 37, Issue 36, 1996, Pages 6431-6434

  Kozyrev, Andrei N ^a   Zheng, Gang ^a   Zhu, Chunfeng ^b   Dougherty, Thomas J ^a   Smith, Kevin M ^b   Pandey, Ravindra K ^a  

^a ROSWELL PARK CANCER INSTITUTE   (United States)

^b UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BACTERIOCHLORIN; BACTERIOCHLOROPHYLL; PHOTOSENSITIZING AGENT;

ANIMAL MODEL; ARTICLE; CANCER; CONTROLLED STUDY; DRUG SYNTHESIS; MASS SPECTROMETRY; MOUSE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; PHOTODYNAMIC THERAPY; PHOTOSENSITIZATION; SPECTROMETRY;

ANIMALIA;

EID: 0030565603     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/0040-4039(96)01346-9     Document Type: Article

References (17)

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5. (a) Pandey, R. K.; Shiau, F. Y.; Sumlin, A. B.; Dougherty, T. J. and Smith, K. M., Bioorg & Med. Chem. Lett., 1994, 4, 1263.
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7. (c) Kozyrev, A. N.; Pandey, R. K.; Medforth, C. J., Zheng, G.; Dougherty, T. J. and Smith, K. M., Tetrahedron Lett., 1996, 6, 747.
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9. Lee, S. H.; Jagerovic, N. and Smith, K. M., J. Chem. Soc. Perkin Trans 1, 1993, 2369.
10. (a) Pandey, R. K.; Shiau, F. Y.; Dougherty, T. J. and Smith, K. M., U. S. Patent, 1996, in press,
11. (b) Kozyrev, A. N.; Evimov, A. V.; Efremova, O. A.; Perepyolkin, P. Y.; Mironov, A. F., Proc. SPIE, 1994, 2325, 297.
12. Rb. sphaeroides (green paste) was obtained from Porphyrin Products, Logan, Utah, USA.
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15. 1H NMR (400 MHz, expressed in δ ppm) and Mass Spectrometry Data:
16. 5: 675. Found: 676 (M+l).
17. 5: 707.9 Found: 707.9 (M+1).