-
1
-
-
0002976015
-
-
Filler, R., Kobayashi, Y., Eds.; Kodansha: Tokyo
-
1. (a) Kollonitsch, J. In Biomedical Aspects of Fluorine Chemistry; Filler, R., Kobayashi, Y., Eds.; Kodansha: Tokyo, 1982, pp. 93-122.
-
(1982)
Biomedical Aspects of Fluorine Chemistry
, pp. 93-122
-
-
Kollonitsch, J.1
-
2
-
-
0012005107
-
-
Kobayashi, Y., Kumadaki, I., Taguchi, T., Eds.; Hirokawa Publishing: Tokyo, (in Japanese)
-
(b) Tsushima, T.; Kawada, K. In Fluorine Chemistry in Pharmaceutical Sciences, Basic and Experimental; Kobayashi, Y., Kumadaki, I., Taguchi, T., Eds.; Hirokawa Publishing: Tokyo, 1993, pp. 55-72 (in Japanese),
-
(1993)
Fluorine Chemistry in Pharmaceutical Sciences, Basic and Experimental
, pp. 55-72
-
-
Tsushima, T.1
Kawada, K.2
-
4
-
-
0002696051
-
-
2. (a) Tsushima, T.; Kawada, K.; Shiratori, O.; Uchida, N. Heterocycles 1985, 23, 45.
-
(1985)
Heterocycles
, vol.23
, pp. 45
-
-
Tsushima, T.1
Kawada, K.2
Shiratori, O.3
Uchida, N.4
-
5
-
-
0023735973
-
-
(b) Tsushima, T.; Kawada, K.; Ishihara, S.; Uchida, N.; Shiratori, O; Higaki, J.; Hirata, M. Tetrahedron 1988, 44, 5375.
-
(1988)
Tetrahedron
, vol.44
, pp. 5375
-
-
Tsushima, T.1
Kawada, K.2
Ishihara, S.3
Uchida, N.4
Shiratori, O.5
Higaki, J.6
Hirata, M.7
-
6
-
-
0004060819
-
-
American Chemical Society: Washington, D.C.
-
3. For a recent review on fluorine chemistry, see: (a) Chemistry of Organic Fluorine Compounds II, A Critical Review, Hudlicky, M.; Pavlath, A. E. Eds.; American Chemical Society: Washington, D.C., 1995.
-
(1995)
Chemistry of Organic Fluorine Compounds II, a Critical Review
-
-
Hudlicky, M.1
Pavlath, A.E.2
-
7
-
-
0001834676
-
Fluoroorganic chemistry: Synthetic challenges and biomedical rewards
-
Tetrahedron Symposium-in-Print
-
For recent results in this field, see: (b) Fluoroorganic Chemistry: Synthetic Challenges and Biomedical Rewards (Tetrahedron Symposium-in-Print); Tetrahedron 1996, 52, 1-330.
-
(1996)
Tetrahedron
, vol.52
, pp. 1-330
-
-
-
8
-
-
0000964836
-
-
4. (a) Galivan, J.; Ingless, J.; McGuire, J. J.; Nimec, Z; Coward, J. K. Proc. Natl. Acad. Sci., U.S.A. 1985, 82, 2598.
-
(1985)
Proc. Natl. Acad. Sci., U.S.A.
, vol.82
, pp. 2598
-
-
Galivan, J.1
Ingless, J.2
McGuire, J.J.3
Nimec, Z.4
Coward, J.K.5
-
9
-
-
0011983281
-
-
Welch, J. T. Ed.; American Chemical Society: Washington, D.C.
-
(b) Coward, J. K.; McGuire, J. J.; Galivan, J. In Selective Fluorination in Organic and Bioorganic Chemistry, Welch, J. T. Ed.; American Chemical Society: Washington, D.C., 1991; pp. 196-204.
-
(1991)
Selective Fluorination in Organic and Bioorganic Chemistry
, pp. 196-204
-
-
Coward, J.K.1
McGuire, J.J.2
Galivan, J.3
-
13
-
-
0027953530
-
-
6. For general reviews, see: (a) Bannwarth, B.; Labat, L.; Moride, Y.; Schaeverbeke, T. Drugs 1994, 47, 25.
-
(1994)
Drugs
, vol.47
, pp. 25
-
-
Bannwarth, B.1
Labat, L.2
Moride, Y.3
Schaeverbeke, T.4
-
14
-
-
0029164467
-
-
(b) DeGraw, J. I.; Colwell, W. T.; Pipe, J. R.; Sirotnak, F. M.; Smith, R. L. Curr. Med. Chem. 1995, 2, 630.
-
(1995)
Curr. Med. Chem.
, vol.2
, pp. 630
-
-
DeGraw, J.I.1
Colwell, W.T.2
Pipe, J.R.3
Sirotnak, F.M.4
Smith, R.L.5
-
15
-
-
0021363704
-
-
7. MTX analogue containing D-glutamic acid was reported to be a poor inhibitor of cell growth, see: (a) Cramer, S. M.; Schomagel, J. H.; Kalghatgi, K. K.; Bertino, J. R.; Horvath, C. Cancer Res. 1984, 44, 1843.
-
(1984)
Cancer Res.
, vol.44
, pp. 1843
-
-
Cramer, S.M.1
Schomagel, J.H.2
Kalghatgi, K.K.3
Bertino, J.R.4
Horvath, C.5
-
16
-
-
0030026396
-
-
The in vitro activity of L-threo-3 has been reported recently, see: (b) Hart, B. P.; Haile, W. H.; Licato, N. J.; Bolanowska, W. E.; McGuire, J. J.; Coward, J. K. J. Med. Chem. 1996, 39, 56.
-
(1996)
J. Med. Chem.
, vol.39
, pp. 56
-
-
Hart, B.P.1
Haile, W.H.2
Licato, N.J.3
Bolanowska, W.E.4
McGuire, J.J.5
Coward, J.K.6
-
18
-
-
0026590329
-
-
(b) Avent, A. G.; Bowler, A. N.; Doyle, P. M.; Marchand, C. M.; Young, D. W. Tetrahedron Lett. 1992, 33, 1509.
-
(1992)
Tetrahedron Lett.
, vol.33
, pp. 1509
-
-
Avent, A.G.1
Bowler, A.N.2
Doyle, P.M.3
Marchand, C.M.4
Young, D.W.5
-
21
-
-
37049109218
-
-
(b) Bory, S.; Dubois, J.; Gaudry, M.; Marquet, A.; Lacombe, L.; Weinstein, S. J. Chem. Soc., Perkin Trans. 1 1984, 475.
-
(1984)
J. Chem. Soc., Perkin Trans.
, vol.1
, pp. 475
-
-
Bory, S.1
Dubois, J.2
Gaudry, M.3
Marquet, A.4
Lacombe, L.5
Weinstein, S.6
-
22
-
-
0000729413
-
-
and references cited therein
-
10. Tolman V. J. Fluorine Chem. 1993, 60, 179, and references cited therein.
-
(1993)
J. Fluorine Chem.
, vol.60
, pp. 179
-
-
Tolman, V.1
-
23
-
-
0011948429
-
-
Several kilograms of the adduct were purchased from Daikin Industries, Ltd., see: ref. 12
-
11. Several kilograms of the adduct were purchased from Daikin Industries, Ltd., see: ref. 12.
-
-
-
-
27
-
-
0011975143
-
-
Kukhar, V. P., Soloshonok, V. A., Eds.; John Wiley & Sons: New York
-
For reviews on enzymatic preparation of fluorine-containing amino acids, see: (b) Matsumura, Y.; Urushihara, M. In Fluorine-containing Amino Acids: Synthesis and Properties; Kukhar, V. P., Soloshonok, V. A., Eds.; John Wiley & Sons: New York, 1995; pp 243-265.
-
(1995)
Fluorine-containing Amino Acids: Synthesis and Properties
, pp. 243-265
-
-
Matsumura, Y.1
Urushihara, M.2
-
29
-
-
0011950146
-
-
14. Burde, N. L.; Alekseeva, L. V.; Lundin, B. N. Zh. Obshch. Khim. 1968, 38, 439.
-
(1968)
Zh. Obshch. Khim.
, vol.38
, pp. 439
-
-
Burde, N.L.1
Alekseeva, L.V.2
Lundin, B.N.3
-
30
-
-
0019038017
-
-
15. (a) Gentzen, I.; Löffler, H.-G.; Schneider, F. Z. Naturforsch. 1980, 35c, 544.
-
(1980)
Z. Naturforsch.
, vol.35 C
, pp. 544
-
-
Gentzen, I.1
Löffler, H.-G.2
Schneider, F.3
-
31
-
-
33845183768
-
-
(b) Chenault, H. K.; Dahmer, J.; Whitesides, G. M. J. Am. Chem. Soc. 1989, 111, 6354.
-
(1989)
J. Am. Chem. Soc.
, vol.111
, pp. 6354
-
-
Chenault, H.K.1
Dahmer, J.2
Whitesides, G.M.3
-
32
-
-
0000812849
-
-
16. Vidal-Cros, A.; Gaudry, M.; Marquet, A. J. Org. Chem. 1985, 50, 3163.
-
(1985)
J. Org. Chem.
, vol.50
, pp. 3163
-
-
Vidal-Cros, A.1
Gaudry, M.2
Marquet, A.3
-
35
-
-
0011989128
-
-
Data of X-ray crystallographic analysis of both 1a and 1b can be obtained from Mr. H. Nakai of these Laboratories. The X-ray crystal structures of 1b and 1c were also reported by Hudlicky and Merola, see: ref. 8a
-
19. Data of X-ray crystallographic analysis of both 1a and 1b can be obtained from Mr. H. Nakai of these Laboratories. The X-ray crystal structures of 1b and 1c were also reported by Hudlicky and Merola, see: ref. 8a.
-
-
-
-
36
-
-
0000416098
-
-
20. Tolman et al. reported that DL-threo-8·HCl was secured in high diastereomeric purity by recrystallization from acetone, see: Tolman, V.; Vlasakova, V.; Nemecek, J. Fluorine Chem. 1993, 60, 185.
-
(1993)
J. Fluorine Chem.
, vol.60
, pp. 185
-
-
Tolman, V.1
Vlasakova, V.2
Nemecek3
-
37
-
-
0000509230
-
-
21. (a) Benson, J. R.; Hare, P. E. Proc. Natl. Acad. Sci., U.S.A. 1975, 72, 619.
-
(1975)
Proc. Natl. Acad. Sci., U.S.A.
, vol.72
, pp. 619
-
-
Benson, J.R.1
Hare, P.E.2
-
38
-
-
0012049198
-
-
(b) Gil-Av, E.; Tishbee, A.; Hare, P. E. J. Am. Chem. Soc. 1980, 102, 5115.
-
(1980)
J. Am. Chem. Soc.
, vol.102
, pp. 5115
-
-
Gil-Av, E.1
Tishbee, A.2
Hare, P.E.3
|