Structure-activity relationship studies of novel pyrazolo[1,5-c][1,3]benzoxazines: Synthesis and benzodiazepine receptor affinity

Archiv der Pharmazie

Volumn 329, Issue 12, 1996, Pages 529-534

  Varano, Flavia ^a   Catarzi, Daniela ^a   Colotta, Vittoria ^a   Cecchi, Lucia ^a   Filacchioni, Guido ^a   Galli, Alessandro ^a   Costagli, Chiara ^a  

^a UNIVERSITY OF FLORENCE   (Italy)

Author keywords

benzodiazepine receptor ligands; pharmacophoric descriptors; pyrazolo 1,5 c 1,3 benzoxazines

Indexed keywords

4 AMINOBUTYRIC ACID; BENZODIAZEPINE RECEPTOR; BENZOXAZINE DERIVATIVE; FLUNITRAZEPAM; PYRAZOLO[1,5 C][1,3]BENZOXAZINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; IN VITRO STUDY; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; STRUCTURE ACTIVITY RELATION;

ANIMALS; CEREBRAL CORTEX; LIGANDS; MALE; OXAZINES; PYRAZOLES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, GABA-A; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0030482291     PISSN: 03656233     EISSN: None     Source Type: Journal    
DOI: 10.1002/ardp.19963291204     Document Type: Article

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