Cyclic morphiceptin analogs: Cyclization studies and opioid activities in vitro

International Journal of Peptide and Protein Research

Volumn 48, Issue 6, 1996, Pages 495-502

  Vogel, D ^a,b   Schmidt, R ^b   Hartung K ^b,c,d   Demuth, H U ^b,d   Chung, N N ^a,b   Schiller, P W ^a  

^a Hans Knoell Inst Nat Prod Res J   (Germany)

^b CLIN RESEARCH INSTITUTE OF MONTREAL   (Canada)

^c Federal Institute of Neurobiology   (Germany)

^d Astra Research Centre Montreal   (Canada)

Author keywords

In vitro opioid activity; Morphiceptin analogs; Peptide cyclization

Indexed keywords

DELTA OPIATE RECEPTOR; MORPHICEPTIN DERIVATIVE; MU OPIATE RECEPTOR;

ANIMAL TISSUE; ARTICLE; BIOASSAY; CHIRALITY; CONTROLLED STUDY; CRYSTALLIZATION; CYCLIZATION; DRUG SYNTHESIS; GUINEA PIG; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; ILEUM; IN VITRO STUDY; LIQUID CHROMATOGRAPHY; MASS SPECTROMETRY; MOUSE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; REACTION ANALYSIS; SMOOTH MUSCLE CONTRACTION; STRUCTURE ACTIVITY RELATION; THIN LAYER CHROMATOGRAPHY; VAS DEFERENS;

ANIMALIA; CAVIA PORCELLUS; SUS SCROFA;

EID: 0030454931     PISSN: 03678377     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1399-3011.1996.tb00868.x     Document Type: Article

References (4)

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4. Di Maio, J. & Schiller, P.W. (1980) Proc. Natl. Acad. Sci. USA 77