-
1
-
-
0024567173
-
Very long-acting narcotic antagonists: The 14β-p-substituted cinnamoylaminomorphinones and their partial mu agonist codeinone relatives
-
ACETO, M. D., BOWMAN, E. R., MAY, E. L., HARRIS, L. S., WOODS, J. H., SMITH, C. B., MEDZIHRADSKY, F. AND JACOBSON, A. E.: Very long-acting narcotic antagonists: The 14β-p-substituted cinnamoylaminomorphinones and their partial mu agonist codeinone relatives. Arzneim. Forsch./Drug Res. 39: 570-575, 1989.
-
(1989)
Arzneim. Forsch./Drug Res.
, vol.39
, pp. 570-575
-
-
Aceto, M.D.1
Bowman, E.R.2
May, E.L.3
Harris, L.S.4
Woods, J.H.5
Smith, C.B.6
Medzihradsky, F.7
Jacobson, A.E.8
-
2
-
-
0021058380
-
Operational models of pharmacological agonism
-
BLACK, J. W. AND LEFF, P.: Operational models of pharmacological agonism. Proc. R. Soc. Lond. B 220: 141-162, 1983.
-
(1983)
Proc. R. Soc. Lond. B
, vol.220
, pp. 141-162
-
-
Black, J.W.1
Leff, P.2
-
3
-
-
0017184389
-
A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding
-
BRADFORD, M. M.: A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding. Anal. Biochem. 72: 248-254, 1976.
-
(1976)
Anal. Biochem.
, vol.72
, pp. 248-254
-
-
Bradford, M.M.1
-
4
-
-
0027960605
-
Irreversible opioid antagonist effects of clocinnamox on opioid analgesia and mu receptor binding in mice
-
BURKE, T. F., WOODS, J. H., LEWIS, J. W. AND MEDZIHRADSKY, F.: Irreversible opioid antagonist effects of clocinnamox on opioid analgesia and mu receptor binding in mice. J. Pharmacol. Exp. Ther. 271: 715-721, 1994.
-
(1994)
J. Pharmacol. Exp. Ther.
, vol.271
, pp. 715-721
-
-
Burke, T.F.1
Woods, J.H.2
Lewis, J.W.3
Medzihradsky, F.4
-
5
-
-
0026792917
-
Clocinnamox: A novel, systemically active irreversible opioid antagonist
-
COMER, S. D., BURKE, T. F., LEWIS, J. W. AND WOODS, J. H.: Clocinnamox: A novel, systemically active irreversible opioid antagonist. J. Pharmacol. Exp. Ther. 262: 1051-1056, 1992.
-
(1992)
J. Pharmacol. Exp. Ther.
, vol.262
, pp. 1051-1056
-
-
Comer, S.D.1
Burke, T.F.2
Lewis, J.W.3
Woods, J.H.4
-
6
-
-
0019466744
-
Scatchard analysis of opiate receptor binding
-
FISCHEL, S. V. AND MEDZIHRADSKY, F.: Scatchard analysis of opiate receptor binding. Mol. Pharmacol. 20: 269-279, 1981.
-
(1981)
Mol. Pharmacol.
, vol.20
, pp. 269-279
-
-
Fischel, S.V.1
Medzihradsky, F.2
-
7
-
-
0015337637
-
Log-normal distribution of equieffective doses of norepinephrine and acetylcholine in several tissues
-
FLEMING, W. W., WESTFALL, D. P., DE LA LANDE, I. S. AND JELLETT, L. B.: Log-normal distribution of equieffective doses of norepinephrine and acetylcholine in several tissues. J. Pharmacol. Exp. Ther. 181: 339-345, 1972.
-
(1972)
J. Pharmacol. Exp. Ther.
, vol.181
, pp. 339-345
-
-
Fleming, W.W.1
Westfall, D.P.2
De La Lande, I.S.3
Jellett, L.B.4
-
8
-
-
0002355204
-
The use of β-haloalkylamines in the differentiation of receptors and in the determination of dissociation constants of receptor-agonist complexes
-
FURCHGOTT, R. F.: The use of β-haloalkylamines in the differentiation of receptors and in the determination of dissociation constants of receptor-agonist complexes. Adv. Drug Res. 3: 21-56, 1966.
-
(1966)
Adv. Drug Res.
, vol.3
, pp. 21-56
-
-
Furchgott, R.F.1
-
9
-
-
0024433616
-
Hydrophobic calcium channel ligands: Methodical problems and their solution
-
GRAZIADEI, I., ZERNIG, G., GRASSEGGER, A., BOER, R., SCHUDT, C. AND GLOSSMANN, H.: Hydrophobic calcium channel ligands: Methodical problems and their solution. Am. J. Cardiol. 64: 43I-50I, 1989.
-
(1989)
Am. J. Cardiol.
, vol.64
-
-
Graziadei, I.1
Zernig, G.2
Grassegger, A.3
Boer, R.4
Schudt, C.5
Glossmann, H.6
-
10
-
-
0026612763
-
3 aromatic ring in cyclic delta opioid receptor-selective dermorphin/deltorphin tetrapeptide analogues: Electronic and lipophilic requirements for receptor affinity
-
3 aromatic ring in cyclic delta opioid receptor-selective dermorphin/deltorphin tetrapeptide analogues: Electronic and lipophilic requirements for receptor affinity. J. Med. Chem. 35: 1535-1541, 1992.
-
(1992)
J. Med. Chem.
, vol.35
, pp. 1535-1541
-
-
Heyl, D.L.1
Mosberg, H.I.2
-
11
-
-
84873788346
-
The inhibitory effect of fentanyl and other morphine-like analgesics on the warm water induced tail withdrawal reflex in rats
-
JANSSEN, P. A. J., NIEMEGEERS, J. E. AND DONY, J. G. H.: The inhibitory effect of fentanyl and other morphine-like analgesics on the warm water induced tail withdrawal reflex in rats. Arzneim. Forsch./Drug Res. 13: 502-507, 1963.
-
(1963)
Arzneim. Forsch./Drug Res.
, vol.13
, pp. 502-507
-
-
Janssen, P.A.J.1
Niemegeers, J.E.2
Dony, J.G.H.3
-
14
-
-
0024164085
-
New 14-aminomorphinones and codeinones
-
LEWIS, J. W., SMITH, C., MCCARTHY, P., WALTER, D., KOBYLECKI, R., MYERS, M., HAYNES, A., LEWIS, C. AND WALTHAM, K.: New 14-aminomorphinones and codeinones. NIDA Res. Monogr. 90: 136-143, 1988.
-
(1988)
NIDA Res. Monogr.
, vol.90
, pp. 136-143
-
-
Lewis, J.W.1
Smith, C.2
Mccarthy, P.3
Walter, D.4
Kobylecki, R.5
Myers, M.6
Haynes, A.7
Lewis, C.8
Waltham, K.9
-
15
-
-
0020446693
-
Calculating the dissociation constant of an unlabeled compound from the concentration required to displace radiolabel binding by 50%
-
LINDEN, J.: Calculating the dissociation constant of an unlabeled compound from the concentration required to displace radiolabel binding by 50%. J. Cycl. Nucl. Res. 8: 163-172, 1982.
-
(1982)
J. Cycl. Nucl. Res.
, vol.8
, pp. 163-172
-
-
Linden, J.1
-
17
-
-
0002253655
-
Anatomical distribution of opioid receptors in mammalians: An overview
-
Opioids I, ed. by A. Herz, Springer, New York
-
MANSOUR, A. AND WATSON, S. J.: Anatomical distribution of opioid receptors in mammalians: An overview, In: Handbook of Experimental Pharmacology: Opioids I, ed. by A. Herz, pp. 79-105, Springer, New York, 1993.
-
(1993)
Handbook of Experimental Pharmacology
, pp. 79-105
-
-
Mansour, A.1
Watson, S.J.2
-
18
-
-
0027471855
-
Pharmacological mechanisms of opioid analgesics
-
PASTERNAK, G. W.: Pharmacological mechanisms of opioid analgesics. Clin. Neuropharmacol. 16: 1-18, 1993.
-
(1993)
Clin. Neuropharmacol.
, vol.16
, pp. 1-18
-
-
Pasternak, G.W.1
-
19
-
-
0018900991
-
A novel opioid receptor site directed alkylating agent with irreversible narcotic antagonistic and reversible agonistic activities
-
PORTOGHESE, P. S., LARSON, D. L., SAYRE, L. M., FRIES, D. S. AND TAKEMORI, A. E.: A novel opioid receptor site directed alkylating agent with irreversible narcotic antagonistic and reversible agonistic activities. J. Med. Chem. 23: 233-234, 1980.
-
(1980)
J. Med. Chem.
, vol.23
, pp. 233-234
-
-
Portoghese, P.S.1
Larson, D.L.2
Sayre, L.M.3
Fries, D.S.4
Takemori, A.E.5
-
20
-
-
0017643957
-
Memory impairment correlates closely with cycloheximide dose and degree of inhibition of protein synthesis
-
QUINTON, E. E. AND KRAMARCY, N. R.: Memory impairment correlates closely with cycloheximide dose and degree of inhibition of protein synthesis. Brain Res. 131: 184-190, 1977.
-
(1977)
Brain Res.
, vol.131
, pp. 184-190
-
-
Quinton, E.E.1
Kramarcy, N.R.2
-
21
-
-
0026050898
-
Resolution of biphasic binding of the opioid antagonist naltrexone in brain membranes
-
REMMERS, A. E. AND MEDZIHRADSKY, F: Resolution of biphasic binding of the opioid antagonist naltrexone in brain membranes. J. Neurochem. 57: 1265-1269, 1991.
-
(1991)
J. Neurochem.
, vol.57
, pp. 1265-1269
-
-
Remmers, A.E.1
Medzihradsky, F.2
-
22
-
-
0018070660
-
Inhibition of 5,7-dihydrotryptamine-induced supersensitivity to 5-hydroxytryptophan in mice by treatment with cycloheximide
-
SPERK, G., STEWART, R. M., CAMPBELL, A. AND BALDESSARINI, R. J.: Inhibition of 5,7-dihydrotryptamine-induced supersensitivity to 5-hydroxytryptophan in mice by treatment with cycloheximide. Brain Res. 159: 183-194, 1978.
-
(1978)
Brain Res.
, vol.159
, pp. 183-194
-
-
Sperk, G.1
Stewart, R.M.2
Campbell, A.3
Baldessarini, R.J.4
-
23
-
-
0019427430
-
The irreversible narcotic antagonistic and reversible agonistic properties of the fumarate methyl ester derivative of naltrexone
-
TAKEMORI, A. E., LARSON, D. L. AND PORTOGHESE, P. S.: The irreversible narcotic antagonistic and reversible agonistic properties of the fumarate methyl ester derivative of naltrexone. Eur. J. Pharmacol. 70: 445-451, 1981.
-
(1981)
Eur. J. Pharmacol.
, vol.70
, pp. 445-451
-
-
Takemori, A.E.1
Larson, D.L.2
Portoghese, P.S.3
-
25
-
-
0028991723
-
Methoclocinnamox: A mu-partial agonist with pharmacotherapeutic potential for heroin abuse
-
WOODS, J. H., LEWIS, J. W., WINGER, G., BUTELMAN, E., BROADBEAR, J. AND ZERNIG, G.: Methoclocinnamox: A mu-partial agonist with pharmacotherapeutic potential for heroin abuse. NIDA Res. Monogr. 147: 195-219, 1995.
-
(1995)
NIDA Res. Monogr.
, vol.147
, pp. 195-219
-
-
Woods, J.H.1
Lewis, J.W.2
Winger, G.3
Butelman, E.4
Broadbear, J.5
Zernig, G.6
-
26
-
-
0028829429
-
Opioid agonist effects on mouse writhing after irreversible mu receptor blockade with clocinnamox
-
ZERNIG, G., BROADBEAR, J. H., LEWIS, J. W., BRINE, G. A. AND WOODS, J. H.: Opioid agonist effects on mouse writhing after irreversible mu receptor blockade with clocinnamox. Exp. Clin. Psychopharmacol. 3: 323-329, 1995a.
-
(1995)
Exp. Clin. Psychopharmacol.
, vol.3
, pp. 323-329
-
-
Zernig, G.1
Broadbear, J.H.2
Lewis, J.W.3
Brine, G.A.4
Woods, J.H.5
-
27
-
-
0028293519
-
In vivo determination of mu opiod receptor turnover in rhesus monkeys after irreversible blockade with clocinnamox
-
ZERNIG, G., BUTELMAN, E. R., LEWIS, J. W., WALKER, E. A. AND WOODS, J. H.: In vivo determination of mu opiod receptor turnover in rhesus monkeys after irreversible blockade with clocinnamox. J. Pharmacol. Exp. Ther. 269: 57-65, 1994.
-
(1994)
J. Pharmacol. Exp. Ther.
, vol.269
, pp. 57-65
-
-
Zernig, G.1
Butelman, E.R.2
Lewis, J.W.3
Walker, E.A.4
Woods, J.H.5
-
28
-
-
0028831265
-
Receptor reserve and affinity of mu opioid agonists in mouse antinociception: Correlation with receptor binding
-
ZERNIG, G., ISSAEVITCH, T., BROADBEAR, J., BURKE, T., LEWIS, J. W., BRINE, G. A. AND WOODS, J. H.: Receptor reserve and affinity of mu opioid agonists in mouse antinociception: Correlation with receptor binding. Life Sci. 57:2113-2125, 1995b.
-
(1995)
Life Sci.
, vol.57
, pp. 2113-2125
-
-
Zernig, G.1
Issaevitch, T.2
Broadbear, J.3
Burke, T.4
Lewis, J.W.5
Brine, G.A.6
Woods, J.H.7
-
29
-
-
0030221796
-
Calculation of agonist efficacy, apparent affinity and receptor population changes: Comparison of different analytical approaches
-
ZERNIG, G., ISSAEVITCH, T. AND WOODS, J. H.: Calculation of agonist efficacy, apparent affinity and receptor population changes: Comparison of different analytical approaches. J. Pharmacol. Toxicol. Methods, 35:223-237, 1996a.
-
(1996)
J. Pharmacol. Toxicol. Methods
, vol.35
, pp. 223-237
-
-
Zernig, G.1
Issaevitch, T.2
Woods, J.H.3
-
31
-
-
0011998038
-
Clocinnamox effects on intravenous self-administration of mu opioid agonists and cocaine by rhesus monkeys: Agonist efficacy and affinity estimates
-
ZERNIG, G., WINGER, G. D., ISSAEVITCH, T., LEWIS, J. W. AND WOODS, J. H.: Clocinnamox effects on intravenous self-administration of mu opioid agonists and cocaine by rhesus monkeys: Agonist efficacy and affinity estimates. NIDA Res. Monogr., 162:341, 1996b.
-
(1996)
NIDA Res. Monogr.
, vol.162
, pp. 341
-
-
Zernig, G.1
Winger, G.D.2
Issaevitch, T.3
Lewis, J.W.4
Woods, J.H.5
|