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Volumn 277, Issue 3, 1996, Pages 1444-1453

Tamoxifen (estrogen antagonist) inhibits voltage-gated calcium current and contractility in vascular smooth muscle from rats1

Author keywords

[No Author keywords available]

Indexed keywords

ANTIESTROGEN; CALCIUM CHANNEL; TAMOXIFEN;

EID: 0030439246     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (68)

References (34)
  • 1
    • 0025333499 scopus 로고
    • Interaction of antiestrogens with binding sites for muscarinic cholinergic drugs and calcium channel blockers in cell membranes
    • BATRA, S.: Interaction of antiestrogens with binding sites for muscarinic cholinergic drugs and calcium channel blockers in cell membranes. Cancer Chemother. Pharmacol. 26: 310-312, 1990.
    • (1990) Cancer Chemother. Pharmacol. , vol.26 , pp. 310-312
    • Batra, S.1
  • 2
    • 0021141476 scopus 로고
    • A comparison of two doses of tamoxifen (Nolvadex) in postmenopausal women with advanced breast cancer: 10 mg bd versus 20 mg bd
    • BRATHERTON, D. G., BROWN, C. H., BUCHANAN, R., HALL, V., PILLERS, E. M. K., WHEELER, T. K. AND WILLIAMS, C. J.: A comparison of two doses of tamoxifen (Nolvadex) in postmenopausal women with advanced breast cancer: 10 mg bd versus 20 mg bd. Br. J. Cancer 50: 199-205, 1984.
    • (1984) Br. J. Cancer , vol.50 , pp. 199-205
    • Bratherton, D.G.1    Brown, C.H.2    Buchanan, R.3    Hall, V.4    Pillers, E.M.K.5    Wheeler, T.K.6    Williams, C.J.7
  • 3
    • 0027469702 scopus 로고
    • Clinical and radiographic response in a minority of patients with recurrent malignant gliomas treated with high-dose tamoxifen
    • COULDWELL, W. T., WEISS, M. H., DEGIORGIO, C. M., WEINER, L. P., HINTON, D. R., EHRESMANN, G. R., CONTI, P. S. AND APUZZO, M. L. J.: Clinical and radiographic response in a minority of patients with recurrent malignant gliomas treated with high-dose tamoxifen. Neurosurgery 32: 485-490, 1993.
    • (1993) Neurosurgery , vol.32 , pp. 485-490
    • Couldwell, W.T.1    Weiss, M.H.2    Degiorgio, C.M.3    Weiner, L.P.4    Hinton, D.R.5    Ehresmann, G.R.6    Conti, P.S.7    Apuzzo, M.L.J.8
  • 4
    • 0022502275 scopus 로고
    • Isolation of smooth muscle cells from swine carotid artery by digestion with papain
    • DRISKA, S. P. AND PORTER, R.: Isolation of smooth muscle cells from swine carotid artery by digestion with papain. Am. J. Physiol. 251: C474-C481, 1986.
    • (1986) Am. J. Physiol. , vol.251
    • Driska, S.P.1    Porter, R.2
  • 5
    • 0024269590 scopus 로고
    • Effects of adjuvant tamoxifen and of cytotoxic therapy in early breast cancer: An overview of 61 randomized trials among 28,896 women
    • Early Breast Cancer Trialiats' Collaborative Group. Effects of adjuvant tamoxifen and of cytotoxic therapy in early breast cancer: An overview of 61 randomized trials among 28,896 women. N. Engl. J. Med. 319: 1681-1692, 1988.
    • (1988) N. Engl. J. Med. , vol.319 , pp. 1681-1692
  • 6
    • 0001666063 scopus 로고
    • Calcium antagonists in the management of hypertension
    • ed. by M. Epstein, Hanley & Belfus, Inc., Philadelphia, PA
    • EPSTEIN, M.: Calcium antagonists in the management of hypertension. In Calcium Antagonists in Clinical Medicine, ed. by M. Epstein, pp. 213-230, Hanley & Belfus, Inc., Philadelphia, PA, 1992.
    • (1992) Calcium Antagonists in Clinical Medicine , pp. 213-230
    • Epstein, M.1
  • 7
    • 0026511698 scopus 로고
    • Opposite regulation of cAMP concentration in the quail oviduct and the mouse uterus by tamoxifen. Correlation with estrogen-antagonist and eatrogen-agonist activity
    • FANIDI, A., AHNADI, C., FAYARD, J. M., PAGEAUX, J. F. AND LAUGIER, C.: Opposite regulation of cAMP concentration in the quail oviduct and the mouse uterus by tamoxifen. Correlation with estrogen-antagonist and eatrogen-agonist activity. J, Steroid Biochem. Molec. Biol. 41: 571-577, 1992.
    • (1992) J, Steroid Biochem. Molec. Biol. , vol.41 , pp. 571-577
    • Fanidi, A.1    Ahnadi, C.2    Fayard, J.M.3    Pageaux, J.F.4    Laugier, C.5
  • 8
    • 0026730666 scopus 로고
    • Tamoxifen induced changes in MCF7 human breast cancer: In vitro and in vivo studies using nuclear magnetic resonance spectroscopy and imaging
    • FURMAN, E., RUSHKIN, E., MARGALIT, R., BENDEL, P. AND DEGANI, H.: Tamoxifen induced changes in MCF7 human breast cancer: In vitro and in vivo studies using nuclear magnetic resonance spectroscopy and imaging. J. Steroid Biochem. Mol. Biol. 43: 189-195, 1992.
    • (1992) J. Steroid Biochem. Mol. Biol. , vol.43 , pp. 189-195
    • Furman, E.1    Rushkin, E.2    Margalit, R.3    Bendel, P.4    Degani, H.5
  • 9
    • 0025365292 scopus 로고
    • Potassium channels and vascular reactivity in genetically hypertensive rats
    • FURSPAN, P. B. AND WEBB, R. C.: Potassium channels and vascular reactivity in genetically hypertensive rats. Hypertension 15: 687-691, 1990.
    • (1990) Hypertension , vol.15 , pp. 687-691
    • Furspan, P.B.1    Webb, R.C.2
  • 10
    • 0025281705 scopus 로고
    • Contribution of two types of calcium channels to membrane conductance of single myocytes from guinea-pig coronary artery
    • GANITKEVICH, V. YA. AND ISENBERG, G.: Contribution of two types of calcium channels to membrane conductance of single myocytes from guinea-pig coronary artery. J. Physiol. 426: 19-42, 1990.
    • (1990) J. Physiol. , vol.426 , pp. 19-42
    • Ganitkevich, V.Ya.1    Isenberg, G.2
  • 11
    • 0027184395 scopus 로고
    • Tamoxifen decreases the rate of proliferation of rat vascular smooth-muscle cells in culture by inducing production of transforming growth factor B
    • GRAINGER, D. J., WEISSBERG, P. L. AND METCALFE, J. C.: Tamoxifen decreases the rate of proliferation of rat vascular smooth-muscle cells in culture by inducing production of transforming growth factor B. Biochem. J. 294: 109-112, 1993.
    • (1993) Biochem. J. , vol.294 , pp. 109-112
    • Grainger, D.J.1    Weissberg, P.L.2    Metcalfe, J.C.3
  • 12
    • 0028291850 scopus 로고
    • Potentiation of tamoxifen activity by verapamil in a human breast cancer cell line
    • GUPTA, V., KAMATH, N., TKALCEVIC, G. T. AND SINGH, S. V.: Potentiation of tamoxifen activity by verapamil in a human breast cancer cell line. Biochem. Pharmacol. 47: 1701-1704, 1994.
    • (1994) Biochem. Pharmacol. , vol.47 , pp. 1701-1704
    • Gupta, V.1    Kamath, N.2    Tkalcevic, G.T.3    Singh, S.V.4
  • 13
    • 0028080918 scopus 로고
    • Tamoxifen enhances cell death in implanted MCF7 breast cancer by inhibiting endothelium growth
    • HARAN, E. F., MARETZEK, A. F., GOLDBERG, I., HOROWITZ, A. AND DEGANI, H.: Tamoxifen enhances cell death in implanted MCF7 breast cancer by inhibiting endothelium growth. Cancer Res. 21: 5511-5514, 1994.
    • (1994) Cancer Res. , vol.21 , pp. 5511-5514
    • Haran, E.F.1    Maretzek, A.F.2    Goldberg, I.3    Horowitz, A.4    Degani, H.5
  • 14
    • 0020566189 scopus 로고
    • Identification and biological activity of tamoxifen metabolites in human serum
    • KEMP, J. V., ADAM, H. K., WAKELING, A. E. AND SLATER, R.: Identification and biological activity of tamoxifen metabolites in human serum. Biochem. Pharmacol. 32: 2045-2052, 1983.
    • (1983) Biochem. Pharmacol. , vol.32 , pp. 2045-2052
    • Kemp, J.V.1    Adam, H.K.2    Wakeling, A.E.3    Slater, R.4
  • 15
    • 0021321610 scopus 로고
    • Tamoxifen is a calmodulin antagonist in the activation of cAMP phosphodiesterase
    • LAM, P. H.-Y.: Tamoxifen is a calmodulin antagonist in the activation of cAMP phosphodiesterase. Biochem. Biophys. Res. Commun. 118: 27-32, 1984.
    • (1984) Biochem. Biophys. Res. Commun. , vol.118 , pp. 27-32
    • Lam, P.H.-Y.1
  • 16
    • 0021244764 scopus 로고
    • Antiproliferative actions of tamoxifen of human ovarian carcinomas in vitro
    • LAZO, J. S., SCHWARTZ, P. E., MACLUSKY, M. J., LABAREE, D. C. AND EISENFELD, A. J.: Antiproliferative actions of tamoxifen of human ovarian carcinomas in vitro. Cancer Res. 44: 2266-2271, 1984.
    • (1984) Cancer Res. , vol.44 , pp. 2266-2271
    • Lazo, J.S.1    Schwartz, P.E.2    Maclusky, M.J.3    Labaree, D.C.4    Eisenfeld, A.J.5
  • 17
    • 0026425653 scopus 로고
    • Distribution of tamoxifen and its metabolites in rat and human tissues during steady-state treatment
    • LIEN, E. A., SOLHEIM, E. AND UELAND, P. M.: Distribution of tamoxifen and its metabolites in rat and human tissues during steady-state treatment. Cancer Research 51: 4837-4844, 1991.
    • (1991) Cancer Research , vol.51 , pp. 4837-4844
    • Lien, E.A.1    Solheim, E.2    Ueland, P.M.3
  • 18
    • 0023261746 scopus 로고
    • The anti-oestrogen tamoxifen is a calcium antagonist in perfused rat mesentery
    • LIPTON, A.: The anti-oestrogen tamoxifen is a calcium antagonist in perfused rat mesentery. Cancer Chemother. Pharmacol. 20: 125-127, 1987.
    • (1987) Cancer Chemother. Pharmacol. , vol.20 , pp. 125-127
    • Lipton, A.1
  • 19
    • 0025193824 scopus 로고
    • 2+-dependent binding of tamoxifen to calmodulin isolated from bovine brain
    • 2+-dependent binding of tamoxifen to calmodulin isolated from bovine brain. Cancer Research 50: 2753-2758, 1990.
    • (1990) Cancer Research , vol.50 , pp. 2753-2758
    • Lopes, M.C.F.1    Vale, M.G.P.2    Carvalho, A.P.3
  • 20
    • 0000373590 scopus 로고
    • Metabolism of nonsteroidal antiestrogens
    • ed. by V. C. Jordan, University of Wisconsin Press, Madison, WI
    • LYMAN S. D. AND JORDAN, V. C.: Metabolism of nonsteroidal antiestrogens. In Estrogen/Antiestrogen Action and Breast Cancer Therapy, ed. by V. C. Jordan, pp. 191-219, University of Wisconsin Press, Madison, WI, 1986.
    • (1986) Estrogen/Antiestrogen Action and Breast Cancer Therapy , pp. 191-219
    • Lyman, S.D.1    Jordan, V.C.2
  • 21
    • 0026573866 scopus 로고
    • Calcium-dependent enhancement of calcium current in smooth muscle by calmodulin-dependent protein kinase II
    • MCCARRON, J. G., MCGEOWN, J. G., REAEDON, S., IKEBE, M., FAY, F. S. AND WALSH JR., J. V.: Calcium-dependent enhancement of calcium current in smooth muscle by calmodulin-dependent protein kinase II. Nature 357: 74-77, 1992.
    • (1992) Nature , vol.357 , pp. 74-77
    • Mccarron, J.G.1    Mcgeown, J.G.2    Reaedon, S.3    Ikebe, M.4    Fay, F.S.5    Walsh Jr., J.V.6
  • 23
    • 0343832591 scopus 로고
    • Calcium function in vascular smooth muscle and its relationship to hypertension
    • ed. by M. Epstein, Hanley & Belfus, Inc., Philadelphia, PA
    • RAM, J. L., STANDLEY, P. R. AND SOWERS, J. R.: Calcium function in vascular smooth muscle and its relationship to hypertension. In Calcium Antagonists in Clinical Medicine, ed. by M. Epstein, pp. 29-48, Hanley & Belfus, Inc., Philadelphia, PA, 1992.
    • (1992) Calcium Antagonists in Clinical Medicine , pp. 29-48
    • Ram, J.L.1    Standley, P.R.2    Sowers, J.R.3
  • 24
    • 0028569143 scopus 로고
    • In vitro relaxation of phenylephrine- and angiotensin II-contracted aortic rings by β-estradiol
    • RAVI, J., MANTZOROS, C. S., PRABHU, A. S., RAM, J. L. AND SOWERS, J. R.: In vitro relaxation of phenylephrine- and angiotensin II-contracted aortic rings by β-estradiol. Am. J. Hypertens. 7: 1065-1069, 1994.
    • (1994) Am. J. Hypertens. , vol.7 , pp. 1065-1069
    • Ravi, J.1    Mantzoros, C.S.2    Prabhu, A.S.3    Ram, J.L.4    Sowers, J.R.5
  • 25
    • 0018387286 scopus 로고
    • Absence of correlation between antioestrogenic activity and binding affinity for the oestrogen receptor
    • ROCHEFORT, H., GARCIA, M. AND BORGNA, J. L.: Absence of correlation between antioestrogenic activity and binding affinity for the oestrogen receptor. Biochem. Biophys. Res. Commun. 88: 351-357, 1979.
    • (1979) Biochem. Biophys. Res. Commun. , vol.88 , pp. 351-357
    • Rochefort, H.1    Garcia, M.2    Borgna, J.L.3
  • 26
    • 0027325734 scopus 로고
    • Cardiac and thromboembolic morbidity among postmenopausal women with early-stage breast cancer in a randomized trial of adjuvant tamoxifen
    • RUTQVIST, L. E. AND MATTSSON, A: Cardiac and thromboembolic morbidity among postmenopausal women with early-stage breast cancer in a randomized trial of adjuvant tamoxifen. J. Natl. Cancer Inst. 85: 1398-1406, 1993.
    • (1993) J. Natl. Cancer Inst. , vol.85 , pp. 1398-1406
    • Rutqvist, L.E.1    Mattsson, A.2
  • 28
    • 0025953809 scopus 로고
    • Insulin attenuates vasopressin-induced calcium transients and a voltage-dependent calcium response in rat vascular smooth muscle
    • STANDLEY, P. R., ZHANG, F., RAM, J. L., ZEMEL, M. B. AND SOWERS, J. R.: Insulin attenuates vasopressin-induced calcium transients and a voltage-dependent calcium response in rat vascular smooth muscle. J. Clin. Invest. 88: 1230-1236, 1991.
    • (1991) J. Clin. Invest. , vol.88 , pp. 1230-1236
    • Standley, P.R.1    Zhang, F.2    Ram, J.L.3    Zemel, M.B.4    Sowers, J.R.5
  • 30
    • 0027994674 scopus 로고
    • Calmodulin and the regulation of smooth muscle contraction
    • WALSH, M. P.: Calmodulin and the regulation of smooth muscle contraction. Mole. Cell. Biochem. 135: 21-41, 1994.
    • (1994) Mole. Cell. Biochem. , vol.135 , pp. 21-41
    • Walsh, M.P.1
  • 32
    • 0027296162 scopus 로고
    • Tamoxifen and related compounds decrease membrane fluidity in liposomes. Mechanism for the antioxidant action of tamoxifen and relevance to its anticancer and cardioprotective actions?
    • WISEMAN, H., QUINN, P. AND HALLIWELL, B.: Tamoxifen and related compounds decrease membrane fluidity in liposomes. Mechanism for the antioxidant action of tamoxifen and relevance to its anticancer and cardioprotective actions? FEBS Lett. 330: 53-56, 1993.
    • (1993) FEBS Lett. , vol.330 , pp. 53-56
    • Wiseman, H.1    Quinn, P.2    Halliwell, B.3
  • 34
    • 0028124577 scopus 로고
    • Effects of pioglitazone on L-type calcium channels in vascular smooth muscle
    • ZHANG, F., SOWERS, J. R., RAM, J. L., STANDLEY, P. R. AND PECLER, J. D.: Effects of pioglitazone on L-type calcium channels in vascular smooth muscle. Hypertension 24: 170-175, 1994b.
    • (1994) Hypertension , vol.24 , pp. 170-175
    • Zhang, F.1    Sowers, J.R.2    Ram, J.L.3    Standley, P.R.4    Pecler, J.D.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.