Yeast sterol C8-C7 isomerase: Identification and characterization of a high-affinity binding site for enzyme inhibitors

Biochemistry

Volumn 35, Issue 51, 1996, Pages 16871-16878

  Moebius, Fabian F ^a   Bermoser, Katrin ^a   Reiter, Raphael J ^a   Hanner, Markus ^a   Glossmann, Hartmut ^a  

^a UNIVERSITY OF INNSBRUCK   (Austria)

Author keywords

[No Author keywords available]

Indexed keywords

1,4 BIS(2 CHLOROBENZYLAMINOMETHYL)CYCLOHEXANE; 3 (3 HYDROXYPHENYL)PIPERIDINE PROPYL ESTER; AMIODARONE; AZIDOPAMIL; CORTICOSTERONE; DITOLYLGUANIDINE; DRUG BINDING PROTEIN; EMOPAMIL; FENPROPIMORPH; GUANIDINE DERIVATIVE; HALOPERIDOL; IFENPRODIL; ISOMERASE; ISOMERASE INHIBITOR; MDL 28815; METAZOCINE; N [(1,5,9) TRIMETHYLDECYL] 4,10 DIMETHYL 8 AZA DECAL 3BETA OL; NORALLYLMETAZOCINE; OPIPRAMOL; PENTAZOCINE; PIPERIDINE DERIVATIVE; PROGESTERONE; SIGMA RECEPTOR LIGAND; STEROID; TESTOSTERONE; TESTOSTERONE PROPIONATE; TRIDEMORPH; TRIFLUOPERAZINE; TRIFLUPERIDOL; TRIPARANOL; UNCLASSIFIED DRUG; UNINDEXED DRUG; DELTA(8) DELTA(7) STEROL ISOMERASE; DELTA(8)-DELTA(7)-STEROL ISOMERASE; ENZYME INHIBITOR; ERGOSTEROL; LIGAND; PRIMER DNA; SIGMA OPIATE RECEPTOR; STEROID DELTA ISOMERASE;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG BINDING SITE; FUNGUS GROWTH; GENE MUTATION; NONHUMAN; ONCOGENE C MYC; PRIORITY JOURNAL; SACCHAROMYCES CEREVISIAE; STEROL SYNTHESIS; ANIMAL; BINDING SITE; BIOSYNTHESIS; CHEMISTRY; DRUG ANTAGONISM; DRUG EFFECT; ENZYMOLOGY; GENETICS; GUINEA PIG; KINETICS; METABOLISM; MUTATION; NUCLEOTIDE SEQUENCE;

CAVIA PORCELLUS; FUNGI; MAMMALIA; SACCHAROMYCES CEREVISIAE; SUS SCROFA;

ANIMALS; BASE SEQUENCE; BINDING SITES; DNA PRIMERS; ENZYME INHIBITORS; ERGOSTEROL; GUINEA PIGS; HALOPERIDOL; KINETICS; LIGANDS; MUTATION; PIPERIDINES; RECEPTORS, SIGMA; SACCHAROMYCES CEREVISIAE; STEROID ISOMERASES; TRIFLUPERIDOL;

EID: 0030300156     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi961996m     Document Type: Article

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